Identification of novel positive allosteric modulators and null modulators at the GABAAreceptor α+β− interface

Subtype selectivity of α+β− site ligands of GABAAreceptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors

(2013) Zdravko Varagic et al.   BRITISH JOURNAL OF PHARMACOLOGY

Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands

(2012) Lars Richter et al.   Nature Chemical Biology

A novel GABAA receptor pharmacology: drugs interacting with the α+β- interface

(2011) Werner Sieghart et al.   BRITISH JOURNAL OF PHARMACOLOGY

The GABAA Receptor  + - Interface: A Novel Target for Subtype Selective Drugs

(2011) J. Ramerstorfer et al.   JOURNAL OF NEUROSCIENCE

Valerenic acid derivatives as novel subunit-selective GABAA receptor ligands -in vitro and in vivo characterization

(2010) S Khom et al.   BRITISH JOURNAL OF PHARMACOLOGY

The point mutation γ2F77I changes the potency and efficacy of benzodiazepine site ligands in different GABAA receptor subtypes

(2010) Joachim Ramerstorfer et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Covalent modification of GABAAreceptor isoforms by a diazepam analogue provides evidence for a novel benzodiazepine binding site that prevents modulation by these drugs

(2008) Roland Baur et al.   JOURNAL OF NEUROCHEMISTRY

International Union of Pharmacology. LXX. Subtypes of  -Aminobutyric AcidA Receptors: Classification on the Basis of Subunit Composition, Pharmacology, and Function. Update

(2008) R. W. Olsen et al.   PHARMACOLOGICAL REVIEWS