Differential Modulation of Beta-Adrenergic Receptor Signaling by Trace Amine-Associated Receptor 1 Agonists

β-blockers as endocrine disruptors: the potential effects of human β-blockers on aquatic organisms

(2011) Andrey Massarsky et al.   Journal of Experimental Zoology Part A-Ecological Genetics and Physiology

In silico analysis of the binding of agonists and blockers to the β2-adrenergic receptor

(2011) Santiago Vilar et al.   JOURNAL OF MOLECULAR GRAPHICS & MODELLING

The structural basis for agonist and partial agonist action on a β1-adrenergic receptor

(2011) Tony Warne et al.   NATURE

Structure and function of an irreversible agonist-β2 adrenoceptor complex

(2011) Daniel M. Rosenbaum et al.   NATURE

Chemogenomic Analysis of G-Protein Coupled Receptors and Their Ligands Deciphers Locks and Keys Governing Diverse Aspects of Signalling

(2011) Jörg D. Wichard et al.   PLoS One

TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic and hypoglutamatergic activity

(2011) F. G. Revel et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): Discovery of EPPTB (RO5212773)

(2010) Henri Stalder et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Functional evolution of the trace amine associated receptors in mammals and the loss of TAAR1 in dogs

(2010) Eric J Vallender et al.   BMC EVOLUTIONARY BIOLOGY

3-Monoiodothyronamine: The rationale for its action as an endogenous adrenergic-blocking neuromodulator

(2010) Heinrich S. Gompf et al.   BRAIN RESEARCH

Tissue Distribution and Cardiac Metabolism of 3-Iodothyronamine

(2010) Alessandro Saba et al.   ENDOCRINOLOGY

GPCR structure and activation: an essential role for the first extracellular loop in activating the adenosine A2B receptor

(2010) Miriam C. Peeters et al.   FASEB JOURNAL

3-Iodothyronamine (T1AM): a new chapter of thyroid hormone endocrinology?

(2010) Alexandra G. Ianculescu et al.   Molecular BioSystems

Effects of Synephrine andβ-Phenethylamine on Humanα-Adrenoceptor Subtypes

(2010) Guoyi Ma et al.   PLANTA MEDICA

Structural and Functional Evolution of the Trace Amine-Associated Receptors TAAR3, TAAR4 and TAAR5 in Primates

(2010) Claudia Stäubert et al.   PLoS One

TAAR6 variations possibly associated with antidepressant response and suicidal behavior

(2010) Chi-Un Pae et al.   PSYCHIATRY RESEARCH

Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist

(2010) E. Y. T. Chien et al.   SCIENCE

The minor binding pocket: a major player in 7TM receptor activation

(2010) Mette M. Rosenkilde et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Importance of the extracellular loops in G protein-coupled receptors for ligand recognition and receptor activation

(2010) M.C. Peeters et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

The Molecular Basis of Species-Specific Ligand Activation of Trace Amine-Associated Receptor 1 (TAAR1)

(2009) Edwin S. Tan et al.   ACS Chemical Biology

Trace Amine-associated Receptors Are Olfactory Receptors in Vertebrates

(2009) Stephen D. Liberles   Annals of the New York Academy of Sciences

Human and mouse trace amine-associated receptor 1 have distinct pharmacology towards endogenous monoamines and imidazoline receptor ligands

(2009) Liaoyuan A. Hu et al.   BIOCHEMICAL JOURNAL

Amiodarone and its putative metabolites fail to activate wild type hTAAR1

(2009) Anita H. Lewin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Modulation of cardiac ionic homeostasis by 3-iodothyronamine

(2009) Sandra Ghelardoni et al.   JOURNAL OF CELLULAR AND MOLECULAR MEDICINE

Trace Amine-Associated Receptors as Emerging Therapeutic Targets

(2009) T. D. Sotnikova et al.   MOLECULAR PHARMACOLOGY

TAAR 6 and HSP-70 variations associated with bipolar disorder

(2009) Chi-Un Pae et al.   NEUROSCIENCE LETTERS

Trace amine metabolism in Parkinson's disease: Low circulating levels of octopamine in early disease stages

(2009) Giovanni D’Andrea et al.   NEUROSCIENCE LETTERS

International Union of Pharmacology. LXXII. Recommendations for Trace Amine Receptor Nomenclature

(2009) J. J. Maguire et al.   PHARMACOLOGICAL REVIEWS

Comparative Sequence and Structural Analyses of G-Protein-Coupled Receptor Crystal Structures and Implications for Molecular Models

(2009) Catherine L. Worth et al.   PLoS One

Positive Darwinian selection and the birth of an olfactory receptor clade in teleosts

(2009) A. Hussain et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

The selective antagonist EPPTB reveals TAAR1-mediated regulatory mechanisms in dopaminergic neurons of the mesolimbic system

(2009) A. Bradaia et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Mammalian olfactory receptors

(2009) Joerg Fleischer   Frontiers in Cellular Neuroscience

Single amino acid of an octopamine receptor as a molecular switch for distinct G protein couplings

(2008) Jia Huang et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Trace amine-associated receptor 1 (TAAR1) is activated by amiodarone metabolites

(2008) Aaron N. Snead et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Human Olfactory Receptor Families and Their Odorants

(2008) Dietmar Krautwurst   CHEMISTRY & BIODIVERSITY

Toward Deciphering the Code to Aminergic G Protein-Coupled Receptor Drug Design

(2008) Edwin S. Tan et al.   CHEMISTRY & BIOLOGY

3-Iodothyronamine (T1AM): A New Player on the Thyroid Endocrine Team?

(2008) Thomas S. Scanlan   ENDOCRINOLOGY

Cardiac effects of thyronamines

(2008) Riccardo Zucchi et al.   HEART FAILURE REVIEWS

Modulation of Monoamine Transporters by Common Biogenic Amines via Trace Amine-Associated Receptor 1 and Monoamine Autoreceptors in Human Embryonic Kidney 293 Cells and Brain Synaptosomes

(2008) Z. Xie et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Endogenous hallucinogens as ligands of the trace amine receptors: A possible role in sensory perception

(2008) J.V. Wallach   MEDICAL HYPOTHESES

Development of a validated liquid chromatography/tandem mass spectrometry method for the distinction of thyronine and thyronamine constitutional isomers and for the identification of new deiodinase substrates

(2008) Susanne Piehl et al.   RAPID COMMUNICATIONS IN MASS SPECTROMETRY

The 2.6 Angstrom Crystal Structure of a Human A2A Adenosine Receptor Bound to an Antagonist

(2008) V.-P. Jaakola et al.   SCIENCE

Trace amine-associated receptors and their ligands

(2006) R Zucchi et al.   BRITISH JOURNAL OF PHARMACOLOGY