Discovery and Optimization of 1,3,4-Trisubstituted-pyrazolone Derivatives as Novel, Potent, and Nonsteroidal Farnesoid X Receptor (FXR) Selective Antagonists

标题
Discovery and Optimization of 1,3,4-Trisubstituted-pyrazolone Derivatives as Novel, Potent, and Nonsteroidal Farnesoid X Receptor (FXR) Selective Antagonists
作者
关键词
-
出版物
JOURNAL OF MEDICINAL CHEMISTRY
Volume 55, Issue 16, Pages 7037-7053
出版商
American Chemical Society (ACS)
发表日期
2012-08-04
DOI
10.1021/jm3002718

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