标题
New Insights on the Mechanism of Quinoline-based DNA Methyltransferase Inhibitors
作者
关键词
-
出版物
JOURNAL OF BIOLOGICAL CHEMISTRY
Volume 290, Issue 10, Pages 6293-6302
出版商
American Society for Biochemistry & Molecular Biology (ASBMB)
发表日期
2014-12-19
DOI
10.1074/jbc.m114.594671
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- Design, Synthesis and Biological Evaluation of 4-Amino-N-(4-aminophenyl)benzamide Analogues of Quinoline-Based SGI-1027 as Inhibitors of DNA Methylation
- (2014) Elodie Rilova et al. ChemMedChem
- Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells
- (2014) Sergio Valente et al. JOURNAL OF MEDICINAL CHEMISTRY
- Structure–activity relationships for 4-anilinoquinoline derivatives as inhibitors of the DNA methyltransferase enzyme DNMT1
- (2013) Swarna A. Gamage et al. BIOORGANIC & MEDICINAL CHEMISTRY
- DNA Methyltransferase-1 Inhibitors as Epigenetic Therapy for Cancer
- (2013) Varinder Singh et al. CURRENT CANCER DRUG TARGETS
- New anticancer active and selective phenylene-bisbenzothiazoles: Synthesis, antiproliferative evaluation and DNA binding
- (2013) Livio Racané et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Laccaic Acid A Is a Direct, DNA-competitive Inhibitor of DNA Methyltransferase 1
- (2013) Rebecca L. Fagan et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- The future of epigenetic therapy in solid tumours—lessons from the past
- (2013) Nilofer Azad et al. Nature Reviews Clinical Oncology
- Development of a universal radioactive DNA methyltransferase inhibition test for high-throughput screening and mechanistic studies
- (2013) Christina Gros et al. NUCLEIC ACIDS RESEARCH
- Clinical outcome of treatment with a combined regimen of decitabine and aclacinomycin/cytarabine for patients with refractory acute myeloid leukemia
- (2012) Lu Xi Song et al. ANNALS OF HEMATOLOGY
- DNA methylation inhibitors in cancer: Recent and future approaches
- (2012) Christina Gros et al. BIOCHIMIE
- Towards the Chemoinformatic-Based Identification of DNA Methyltransferase Inhibitors: 2D- and 3D-Similarity Profile of Screening Libraries
- (2012) Jakyung Yoo et al. Current Computer-Aided Drug Design
- DNA methyltransferase inhibitors in cancer: a chemical and therapeutic patent overview and selected clinical studies
- (2012) Jacques Fahy et al. EXPERT OPINION ON THERAPEUTIC PATENTS
- The Replication Focus Targeting Sequence (RFTS) Domain Is a DNA-competitive Inhibitor of Dnmt1
- (2011) Farisa Syeda et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Structural insight into maintenance methylation by mouse DNA methyltransferase 1 (Dnmt1)
- (2011) K. Takeshita et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Combination Epigenetic Therapy Has Efficacy in Patients with Refractory Advanced Non-Small Cell Lung Cancer
- (2011) R. A. Juergens et al. Cancer Discovery
- Structure and Function of Mammalian DNA Methyltransferases
- (2010) Renata Zofia Jurkowska et al. CHEMBIOCHEM
- Targeting DNA methylation for epigenetic therapy
- (2010) Xiaojing Yang et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- A New Class of Quinoline-Based DNA Hypomethylating Agents Reactivates Tumor Suppressor Genes by Blocking DNA Methyltransferase 1 Activity and Inducing Its Degradation
- (2009) J. Datta et al. CANCER RESEARCH
- Photochemical electrocyclisation of 3-vinylindoles to pyrido[2,3-a]-, pyrido[4,3-a]- and thieno[2,3-a]-carbazoles: Design, synthesis, DNA binding and antitumor cell cytotoxicity
- (2009) Thomas Lemster et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
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