Tetrazolium Compounds: Synthesis and Applications in Medicine

1-Substituted-5-[(3,5-dinitrobenzyl)sulfanyl]-1H-tetrazoles and their isosteric analogs: A new class of selective antitubercular agents active against drug-susceptible and multidrug-resistant mycobacteria

(2014) Galina Karabanovich et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Facile synthesis of 1- and 5-substituted 1H-tetrazoles catalyzed by recyclable ligand complex of copper(II) supported on superparamagnetic Fe3O4@SiO2 nanoparticles

(2014) Mohsen Esmaeilpour et al.   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Valence tautomerism of new pyrazolo[4,3-e]tetrazole[4,5-b][1,2,4]triazines

(2014) Mariusz Mojzych et al.   JOURNAL OF MOLECULAR STRUCTURE

Synthesis and activity of novel tetrazole compounds and their pyrazole-4-carbonitrile precursors against Leishmania spp

(2013) Jéssica V. Faria et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Development of 3D-QSAR CoMSIA models for 5-(biphenyl-2-yl)-1H-tetrazole derivatives as angiotensin II receptor type 1 (AT1) antagonists

(2013) Min Ji Choi et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Correlation of hydrogen-bonding propensity and anticancer profile of tetrazole-tethered combretastatin analogues

(2013) Ganesh S. Jedhe et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of tetrazole containing 1,2,3-thiadiazole derivatives via U-4CR and their anti-TMV activity

(2013) Shou-Xin Wang et al.   CHINESE CHEMICAL LETTERS

Hydrothermal synthesis method of 5-(4′-methylbiphenyl-2-yl)-1H-tetrazole

(2013) Wen-Xiang Wang et al.   CHINESE CHEMICAL LETTERS

Synthesis, characterization, X-ray diffraction, antimicrobial and in vitro cytotoxicity studies of 7a-Aza-B-homostigmast-5-eno [7a,7-d] tetrazole

(2013) Mahboob Alam et al.   COMPTES RENDUS CHIMIE

Synthesis, characterization and anticancer screening of some novel piperonyl–tetrazole derivatives

(2013) Mohammad Arshad et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Anticonvulsant Activity Evaluation of 5-Phenyl-[1,2,4]triazolo[4,3-c]quinazolin-3-amines

(2012) Yan Zheng et al.   ARCHIV DER PHARMAZIE

Fimasartan, a novel angiotensin II receptor antagonist

(2012) Je Hak Kim et al.   ARCHIVES OF PHARMACAL RESEARCH

Inhibitors of HIV-1 attachment. Part 9: An assessment of oral prodrug approaches to improve the plasma exposure of a tetrazole-containing derivative

(2012) Kap-Sun Yeung et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Inhibitors of HIV-1 attachment. Part 8: The effect of C7-heteroaryl substitution on the potency, and in vitro and in vivo profiles of indole-based inhibitors

(2012) Kap-Sun Yeung et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Antimicrobial Activity of Newly Synthesized 2,5-Disubstituted 1,3,4-Thiadiaozle Derivatives

(2012) Mahmoud M.M. Ramiz et al.   BULLETIN OF THE KOREAN CHEMICAL SOCIETY

P2X7 Receptors: Channels, Pores and More

(2012) C. Volonte et al.   CNS & Neurological Disorders-Drug Targets

Synthesis and in vitro evaluation of novel tetrazole embedded 1,3,5-trisubstituted pyrazoline derivatives as Entamoeba histolytica growth inhibitors

(2012) Mohmmad Younus Wani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and evaluation of anticonvulsant and antidepressant activities of 5-alkoxytetrazolo[1,5-c]thieno[2,3-e]pyrimidine derivatives

(2012) Shi-Ben Wang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Structure Optimization and Antifungal Screening of Novel Tetrazole Ring Bearing Acyl-Hydrazones

(2012) Maqsood Ahmad Malik et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Isocyanide-based four-component synthesis of ferrocenyl 1,5-disubstituted tetrazoles

(2012) Tayebeh Amanpour et al.   TETRAHEDRON LETTERS

A facile and rapid route for the synthesis of novel 1,5-substituted tetrazole hydantoins and thiohydantoins via a TMSN3-Ugi/RNCX cyclization

(2012) Federico Medda et al.   TETRAHEDRON LETTERS

Synthesis and antimicrobial activity of new 1-[(tetrazol-5-yl)methyl] indole derivatives, their 1,2,4-triazole thioglycosides and acyclic analogs

(2011) Weal A. El-Sayed et al.   ARCHIVES OF PHARMACAL RESEARCH

Synthesis and anti-inflammatory activity of some new 4,5-dihydro-1,5-diaryl-1H-pyrazole-3-substituted-heteroazole derivatives

(2011) Deepak V. Dekhane et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and evaluation of 1,5-diaryl-substituted tetrazoles as novel selective cyclooxygenase-2 (COX-2) inhibitors

(2011) Baker Jawabrah Al-Hourani et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Catecholthioether Derivatives: Preliminary Study of in-Vitro Antimicrobial and Antioxidant Activities

(2011) Hadi Adibi et al.   CHEMICAL & PHARMACEUTICAL BULLETIN

Probing the antiamoebic and cytotoxicity potency of novel tetrazole and triazine derivatives

(2011) Mohmmad Younus Wani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Evaluation of 1,5-Disubstituted Tetrazoles as Rigid Analogues of Combretastatin A-4 with Potent Antiproliferative and Antitumor Activity

(2011) Romeo Romagnoli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of selected 5-thio-substituted tetrazole derivatives and evaluation of their antibacterial and antifungal activities

(2011) V. Dhayanithi et al.   JOURNAL OF THE SERBIAN CHEMICAL SOCIETY

Synthesis and In Vitro Antiproliferative Activity of Novel Androst-5-ene Triazolyl and Tetrazolyl Derivatives

(2011) Zalán Kádár et al.   MOLECULES

Coordination studies of copper(II), cobalt(II) and iron(II) with isomeric pyridyl–tetrazole ligands

(2011) Andrew D. Bond et al.   POLYHEDRON

Synthesis and characterisation of macrocycles containing both tetrazole and pyridine functionalities

(2011) Adrienne Fleming et al.   TETRAHEDRON

Synthesis and biological evaluation of tetrazole containing compounds as possible anticancer agents

(2011) Chebolu Naga Sesha Sai Pavan Kumar et al.   MedChemComm

Synthesis of some new 4-oxo-thiazolidines, tetrazole and triazole derived from 2-SH-benzothiazole and antimicrobial screening of some synthesized

(2011) Suaad M.H. Al-Majidi   Journal of Saudi Chemical Society

Design and synthesis of novel series of pyrrole based chemotypes and their evaluation as selective aldose reductase inhibitors. A case of bioisosterism between a carboxylic acid moiety and that of a tetrazole

(2010) Kyriaki Pegklidou et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of Novel Cyanodihydropyridines as Potent Mineralocorticoid Receptor Antagonists

(2010) Graciela B. Arhancet et al.   JOURNAL OF MEDICINAL CHEMISTRY

Azole antimicrobial pharmacophore-based tetrazoles: Synthesis and biological evaluation as potential antimicrobial and anticonvulsant agents

(2009) Sherif A.F. Rostom et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, in vitro antibacterial and antifungal evaluations of new α-hydroxyphosphonate and new α-acetoxyphosphonate derivatives of tetrazolo [1, 5-a] quinoline

(2009) Amol H. Kategaonkar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Luminescent zinc and cadmium metal-organic frameworks based on tetrazole ligands

(2009) Tuoping Hu et al.   POLYHEDRON

A Simple, Advantageous Synthesis of 5-Substituted 1H-Tetrazoles¹

(2009) Biswanath Das et al.   SYNLETT

A novel synthesis of 1-aryl tetrazoles promoted by employing the synergy of the combined use of DMSO and an ionic liquid as the solvent system at ambient temperature

(2009) Satish N. Dighe et al.   TETRAHEDRON LETTERS

Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profile

(2008) Scott D. Kuduk et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Tetrazole based amides as growth hormone secretagogues

(2008) James J. Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Characterization of angiotensin II antagonism displayed by Ib, a novel nonpeptide angiotensin AT1 receptor antagonist

(2008) Jinhui Wu et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Azido-tetrazole equilibrium in 2-azidothiazole system. Molecular orbital calculations

(2008) Rafie H. Abu-Eittah et al.   JOURNAL OF MOLECULAR STRUCTURE-THEOCHEM

Synthesis and structure guided evaluation of estrogen agonist and antagonist activities of some new tetrazolyl indole derivatives

(2007) Uma Sharan Singh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY