A One-Pot Tandem Ugi Multicomponent Reaction (MCR)/Click Reaction as an Efficient Protecting-Group-Free Route to 1H-1,2,3-Triazole-Modified α-Amino Acid Derivatives and Peptidomimetics

1,2,3-Triazoles in Peptidomimetic Chemistry

(2011) Daniel Sejer Pedersen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Anion-Binding Properties of a Cyclic Pseudohexapeptide Containing 1,5-Disubstituted 1,2,3-Triazole Subunits

(2011) Martin R. Krause et al.   JOURNAL OF ORGANIC CHEMISTRY

Design and synthesis of bile acid–peptide conjugates linked via triazole moiety

(2011) Nadezhda V. Sokolova et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Three-Component Synthesis of Neoglycopeptides Using a Cu(II)-Triggered Aminolysis of Peptide Hydrazide Resin and an Azide–Alkyne Cycloaddition Sequence

(2011) Jean-Philippe Ebran et al.   ORGANIC LETTERS

Evaluation of amphiphilic aminoglycoside–peptide triazole conjugates as antibacterial agents

(2010) Smritilekha Bera et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Click chemistry: function follows form

(2010) M. G. Finn et al.   CHEMICAL SOCIETY REVIEWS

Tricks with clicks: modification of peptidomimetic oligomers via copper-catalyzed azide-alkyne [3 + 2] cycloaddition

(2010) Justin M. Holub et al.   CHEMICAL SOCIETY REVIEWS

Efficient Multicomponent Reaction Synthesis of the Schistosomiasis Drug Praziquantel

(2010) Haiping Cao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and dual PPARα/δ agonist effects of 1,4-disubstituted 1,2,3-triazole analogues of GW 501516

(2010) Calin C. Ciocoiu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Chiral Isocyanoazides: Efficient Bifunctional Reagents for Bioconjugation

(2010) Valentine G. Nenajdenko et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Ugi reaction for the synthesis of 4-aminopiperidine-4-carboxylic acid derivatives. Application to the synthesis of carfentanil and remifentanil

(2010) Sandra Malaquin et al.   TETRAHEDRON LETTERS

Multiple Multicomponent Macrocyclizations (MiBs): A Strategic Development Toward Macrocycle Diversity

(2009) Ludger A. Wessjohann et al.   CHEMICAL REVIEWS

Natural Product Synthesis Using Multicomponent Reaction Strategies

(2009) Barry B. Touré et al.   CHEMICAL REVIEWS

Rapid Discovery of Triazolobenzylidene-Thiazolopyrimidines (TBTP) as CDC25 Phosphatase Inhibitors by Parallel Click Chemistry and in Situ Screening

(2009) Romain Duval et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Synthesis of Fish Antifreeze Neoglycopeptides Using Microwave-Assisted “Click Chemistry”

(2009) Nicole Miller et al.   ORGANIC LETTERS

Synthesis and Conformational Analysis of a Cyclic Peptide Obtained viaitoi+4 Intramolecular Side-Chain to Side-Chain Azide−Alkyne 1,3-Dipolar Cycloaddition

(2008) Sonia Cantel et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and antibiotic activity of a small molecules library of 1,2,3-triazole derivatives

(2007) Marie Aufort et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS