Transport of drugs by proton-coupled peptide transporters: pearls and pitfalls

Lack of Interaction Between the Peptidomimetic Substrates Captopril and Cephradine

(2009) David R. Foster et al.   JOURNAL OF CLINICAL PHARMACOLOGY

Dipeptide Derivatives of AZT: Synthesis, Chemical Stability, Activation in Human Plasma, hPEPT1 Affinity, and Antiviral Activity

(2008) Cledir Santos et al.   ChemMedChem

High-Affinity Interaction of Sartans with H+/Peptide Transporters

(2008) I. Knutter et al.   DRUG METABOLISM AND DISPOSITION

Transepithelial Transport of the Group II Metabotropic Glutamate 2/3 Receptor Agonist (1S,2S,5R,6S)-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY354740) and Its Prodrug (1S,2S,5R,6S)-2-[(2'S)-(2'-Amino)propionyl]aminobicyclo[3.1.0]hexane-2,6-dicarboxylate (LY544344)

(2008) M. V. S. Varma et al.   DRUG METABOLISM AND DISPOSITION

Role and Relevance of PEPT2 in Drug Disposition, Dynamics, and Toxicity

(2008) Mohamed A. Kamal et al.   Drug Metabolism and Pharmacokinetics

Peptide prodrugs: Improved oral absorption of lopinavir, a HIV protease inhibitor

(2008) Sheetal Agarwal et al.   INTERNATIONAL JOURNAL OF PHARMACEUTICS

Synthesis, metabolism and cellular permeability of enzymatically stable dipeptide prodrugs of acyclovir

(2008) Ravi S. Talluri et al.   INTERNATIONAL JOURNAL OF PHARMACEUTICS

Peptide Derivation of Poorly Absorbable Drug Allows Intestinal Absorption Via Peptide Transporter

(2008) Akihiro Kikuchi et al.   JOURNAL OF PHARMACEUTICAL SCIENCES

Transport of Angiotensin-Converting Enzyme Inhibitors by H+/Peptide Transporters Revisited

(2008) I. Knutter et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Pharmaceutical and pharmacological importance of peptide transporters

(2008) Matthias Brandsch et al.   JOURNAL OF PHARMACY AND PHARMACOLOGY

Targeted Disruption of Peptide TransporterPept1Gene in Mice Significantly Reduces Dipeptide Absorption in Intestine

(2008) Yongun Hu et al.   MOLECULAR PHARMACEUTICS

Synthesis, Transport and Pharmacokinetics of 5′-Amino Acid Ester Prodrugs of 1-β-d-Arabinofuranosylcytosine

(2008) Yongbing Sun et al.   MOLECULAR PHARMACEUTICS

Enhanced Absorption and Growth Inhibition with Amino Acid Monoester Prodrugs of Floxuridine by Targeting hPEPT1 Transporters

(2008) Yasuhiro Tsume et al.   MOLECULES

Quantitative Evaluation of PEPT1 Contribution to Oral Absorption of Cephalexin in Rats

(2008) Takanori Hironaka et al.   PHARMACEUTICAL RESEARCH

The mammalian proton-coupled peptide cotransporter PepT1: sitting on the transporter-channel fence?

(2008) D. Meredith   PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES

Peptide transporters and their roles in physiological processes and drug disposition

(2008) I. Rubio-Aliaga et al.   XENOBIOTICA