A General Synthesis of Indole-3-carboxylic Esters by Palladium-Catalyzed Direct Oxidative Carbonylation of 2-Alkynylaniline Derivatives

KDR inhibitor with the intramolecular non-bonded interaction: Conformation–activity relationships of novel indole-3-carboxamide derivatives

(2011) Takahiro Honda et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Indole synthesis: a review and proposed classification

(2011) Douglass F. Taber et al.   TETRAHEDRON

Multicomponent Cascade Reactions: A Novel and Expedient Approach to Functionalized Indoles by an Unprecedented Nucleophilic Addition-Heterocyclization-Oxidative Alkoxycarbonylation Sequence

(2010) Bartolo Gabriele et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis and anti-hepatitis C virus activity of novel ethyl 1H-indole-3-carboxylates in vitro

(2010) Grazia Sellitto et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Single Agents with Designed Combination Chemotherapy Potential: Synthesis and Evaluation of Substituted Pyrimido[4,5-b]indoles as Receptor Tyrosine Kinase and Thymidylate Synthase Inhibitors and as Antitumor Agents

(2010) Aleem Gangjee et al.   JOURNAL OF MEDICINAL CHEMISTRY

Naturally Occurring and Synthetic Bioactive Molecules as Novel Non-Nucleoside HBV Inhibitors

(2010) Peng Zhan et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Tandem Blaise–Nenitzescu reaction: one-pot synthesis of 5-hydroxy-α-(aminomethylene)benzofuran-2(3H)-ones from nitriles

(2010) Yu Sung Chun et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Cu-Catalyzed Oxidative Amidation of Propiolic Acids Under Air via Decarboxylative Coupling

(2010) Wei Jia et al.   ORGANIC LETTERS

Discovery of benzo[g]indol-3-carboxylates as potent inhibitors of microsomal prostaglandin E2 synthase-1

(2009) Andreas Koeberle et al.   BIOORGANIC & MEDICINAL CHEMISTRY

1-Indol-1-yl-propan-2-ones and related heterocyclic compounds as dual inhibitors of cytosolic phospholipase A2α and fatty acid amide hydrolase

(2009) Laura Forster et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Structural Optimization and Biological Evaluation of 2-Substituted 5-Hydroxyindole-3-carboxylates as Potent Inhibitors of Human 5-Lipoxygenase

(2009) Eva-Maria Karg et al.   JOURNAL OF MEDICINAL CHEMISTRY

Lewis Acid Catalyzed Indole Synthesis via Intramolecular Nucleophilic Attack of Phenyldiazoacetates to Iminium Ions

(2009) Lei Zhou et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of the new ring system 2-oxo-[1,4]oxazino[3,2-e]indole, heteroanalogue of Angelicin

(2009) Paola Barraja et al.   TETRAHEDRON LETTERS

Synthesis of 1-Amino-1H-indole-3-carboxylates by Copper(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand Melkonyan et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of N-Substituted Indole-3-carboxylic Acid Derivatives via Cu(I)-Catalyzed Intramolecular Amination of Aryl Bromides

(2008) Ferdinand S. Melkonyan et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Indole-3-carboxylic Acid Derivatives by Pd(0)-Catalyzed Intramolecular α-Arylation of β-(2-Iodoanilino) Esters

(2008) Daniel Solé et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Synthesis of 3-Indolecarboxylic Acid Derivatives

(2008) Björn Söderberg et al.   SYNTHESIS-STUTTGART