Discovery of 1-{4-[3-Fluoro-4-((3S,6R)-3-methyl-1,1-dioxo-6-phenyl-[1,2]thiazinan-2-ylmethyl)-phenyl]-piperazin-1-yl}-ethanone (GNE-3500): a Potent, Selective, and Orally Bioavailable Retinoic Acid Receptor-Related Orphan Receptor C (RORc or RORγ) Inverse Agonist
JOURNAL OF MEDICINAL CHEMISTRY (2015)
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JOURNAL OF MEDICINAL CHEMISTRY
卷 58, 期 13, 页码 5308-5322出版社
AMER CHEMICAL SOC
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- US NIH Shared Instrumentation grant [S10-RR027172]
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