B-Ring-Modified isoCombretastatin A-4 Analogues Endowed with Interesting Anticancer Activities

Copper-Catalyzed Direct Amination of Halo(hetero)arenes with Sodium Azide as the Amino Source

(2012) S. Messaoudi et al.   MINI-REVIEWS IN ORGANIC CHEMISTRY

Discovery of Isoerianin Analogues as Promising Anticancer Agents

(2011) Samir Messaoudi et al.   ChemMedChem

An Expeditious Copper-Catalyzed Access to 3-Aminoquinolinones, 3-Aminocoumarins and Anilines using Sodium Azide

(2010) Samir Messaoudi et al.   ADVANCED SYNTHESIS & CATALYSIS

Substituted 2-(3′,4′,5′-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitors

(2010) Romeo Romagnoli et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and Evaluation of Azetidinone Analogues of Combretastatin A-4 as Tubulin Targeting Agents

(2010) Niamh M. O’Boyle et al.   JOURNAL OF MEDICINAL CHEMISTRY

p-Toluenesulfonic acid-promoted selective functionalization of unsymmetrical arylalkynes: a regioselective access to various arylketones and heterocycles

(2010) Maud Jacubert et al.   TETRAHEDRON

Synthesis, Biological Evaluation of 1,1-Diarylethylenes as a Novel Class of Antimitotic Agents

(2009) Abdallah Hamze et al.   ChemMedChem

A review and update of the current status of the vasculature-disabling agent combretastatin-A4 phosphate (CA4P)

(2009) Dietmar W Siemann et al.   EXPERT OPINION ON INVESTIGATIONAL DRUGS

Isocombretastatins A versus Combretastatins A: The ForgottenisoCA-4 Isomer as a Highly Promising Cytotoxic and Antitubulin Agent

(2009) Samir Messaoudi et al.   JOURNAL OF MEDICINAL CHEMISTRY

p-Toluenesulfonic acid-mediated cyclization of o-(1-alkynyl)anisoles or thioanisoles: synthesis of 2-arylsubstituted benzofurans and benzothiophenes

(2009) Maud Jacubert et al.   TETRAHEDRON LETTERS

Expeditious synthesis of 1,1-diarylethylenes related to isocombretastatin A-4 (isoCA-4) via palladium-catalyzed arylation of N-tosylhydrazones with aryl triflates

(2009) Bret Tréguier et al.   TETRAHEDRON LETTERS

1,5-Disubstituted 1,2,3-triazoles as cis-restricted analogues of combretastatin A-4: Synthesis, molecular modeling and evaluation as cytotoxic agents and inhibitors of tubulin

(2008) Kristin Odlo et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and antitumor activity of benzils related to combretastatin A-4

(2008) Céline Mousset et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Blood Vessel Maturation and Response to Vascular-Disrupting Therapy in Single Vascular Endothelial Growth Factor-A Isoform-Producing Tumors

(2008) G. M. Tozer et al.   CANCER RESEARCH

DMSO–PdI2 as a powerful oxidizing couple of alkynes into benzils: one-pot synthesis of nitrogen-containing five- or six-membered heterocycles

(2008) Céline Mousset et al.   TETRAHEDRON

One-pot hydrosilylation–protodesilylation of functionalized diarylalkynes: a highly selective access to Z-stilbenes. Application to the synthesis of combretastatin A-4

(2007) Anne Giraud et al.   TETRAHEDRON LETTERS