Ruthenium-Catalyzed Cycloadditions of 1-Haloalkynes with Nitrile Oxides and Organic Azides: Synthesis of 4-Haloisoxazoles and 5-Halotriazoles

Copper(I)-Catalyzed Cycloaddition of Bismuth(III) Acetylides with Organic Azides: Synthesis of Stable Triazole Anion Equivalents

(2013) Brady T. Worrell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Tandem Reaction of 1-Copper(I) Alkynes for the Synthesis of 1,4,5-Trisubstituted 5-Chloro-1,2,3-triazoles

(2013) Bo Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Fused Polycyclic Compounds via Cycloaddition of 4-(1′-Cyclohexenyl)-5-iodo-1,2,3-triazoles with 4-Phenyl-1,2,4-triazoline-3,5-dione: The Importance of a Sacrificial Iodide Leaving Group

(2013) Heather A. Michaels et al.   JOURNAL OF ORGANIC CHEMISTRY

Transannulation of 1-Sulfonyl-1,2,3-triazoles with Heterocumulenes

(2013) Stepan Chuprakov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Iridium-Catalyzed Cycloaddition of Azides and 1-Bromoalkynes at Room Temperature

(2013) Evelia Rasolofonjatovo et al.   ORGANIC LETTERS

Heterocycle–Heterocycle Strategies: (2-Nitrophenyl)isoxazole Precursors to 4-Aminoquinolines, 1H-Indoles, and Quinolin-4(1H)-ones

(2013) Keith C. Coffman et al.   ORGANIC LETTERS

Palladium-Catalyzed Cross-Coupling of 1,4-Disubstituted 5-Iodo-1,2,3-tri­azoles with Organotin Reagents

(2013) Jérôme Thibonnet et al.   SYNTHESIS-STUTTGART

Halogen Exchange (Halex) Reaction of 5-Iodo-1,2,3-triazoles: Synthesis and Applications of 5-Fluorotriazoles

(2012) Brady T. Worrell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Braces for the Peptide Backbone: Insights into Structure-Activity Relationships of Protease Inhibitor Mimics with Locked Amide Conformations

(2012) Marco Tischler et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design, synthesis and biological evaluation of novel 2-methylpyrimidine-4-ylamine derivatives as inhibitors of Escherichia coli pyruvate dehydrogenase complex E1

(2012) Junbo He et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Design and synthesis of potent, isoxazole-containing renin inhibitors

(2012) Pierre-André Fournier et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and evaluation of 4-(substituted styryl/alkenyl)-3,5-bis(4-hydroxyphenyl)-isoxazoles as ligands for the estrogen receptor

(2012) Terra Haddad et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

(Iminophosphorane)copper(I) Complexes as Highly Efficient Catalysts for 1,3-Dipolar Cycloaddition of Azides with Terminal and 1-Iodoalkynes in Water: One-Pot Multi-Component Reaction from Alkynes and in situ Generated Azides

(2012) Joaquín García-Álvarez et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Synthesis of 5-Iodo-1,4-disubstituted-1,2,3-triazoles Mediated by in Situ Generated Copper(I) Catalyst and Electrophilic Triiodide Ion

(2012) Wendy S. Brotherton et al.   JOURNAL OF ORGANIC CHEMISTRY

Reaction mechanism of ruthenium-catalyzed azide–alkyne cycloaddition reaction: A DFT study

(2012) Esra Boz et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Arylation of Rhodium(II) Azavinyl Carbenes with Boronic Acids

(2012) Nicklas Selander et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ruthenium-Catalyzed Transformation of Aryl and Alkenyl Triflates to Halides

(2012) Yusuke Imazaki et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly regioselective nitrile oxide dipolar cycloadditions with ortho-nitrophenyl alkynes

(2012) Melissa L. McIntosh et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Coordinatively Unsaturated Ruthenium Complexes As Efficient Alkyne–Azide Cycloaddition Catalysts

(2012) Marina Lamberti et al.   ORGANOMETALLICS

Triazole Appending Agent (TAAG): A New Synthon for Preparing Iodine-Based Molecular Imaging and Radiotherapy Agents

(2012) Alla Darwish et al.   ACS Medicinal Chemistry Letters

“Triazole Bridge”: Disulfide-Bond Replacement by Ruthenium-Catalyzed Formation of 1,5-Disubstituted 1,2,3-Triazoles

(2011) Martin Empting et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Isoxazole Functionalization Technologies Enable Construction of Tetracycline Derivatives

(2011) Brian Heasley   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Triazole: a unique building block for the construction of functional materials

(2011) Michal Juríček et al.   CHEMICAL COMMUNICATIONS

Catalytic Asymmetric C–H Insertions of Rhodium(II) Azavinyl Carbenes

(2011) Stepan Chuprakov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 5-Iodo-1,2,3-triazole-Containing Macrocycles Using Copper Flow Reactor Technology

(2011) Andrew R. Bogdan et al.   ORGANIC LETTERS

Direct Synthesis of 1,4-Disubstituted-5-alumino-1,2,3-triazoles: Copper-Catalyzed Cycloaddition of Organic Azides and Mixed Aluminum Acetylides

(2010) Yuhan Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structure–activity studies of a novel series of isoxazole-3-carboxamide derivatives as TRPV1 antagonists

(2010) Ronald Palin et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Copper-catalyzed azide–alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(i) acetylides

(2010) Jason E. Hein et al.   CHEMICAL SOCIETY REVIEWS

A Versatile Iron-Catalyzed Protocol for the One-Pot Synthesis of Isoxazoles or Isoxazolines from the Same Propargylic Alcohols

(2010) Olivier Debleds et al.   CHEMISTRY-A EUROPEAN JOURNAL

A highly efficient copper(i) catalyst for the 1,3-dipolar cycloaddition of azides with terminal and 1-iodoalkynes in water: regioselective synthesis of 1,4-disubstituted and 1,4,5-trisubstituted 1,2,3-triazoles

(2010) Joaquín García-Álvarez et al.   GREEN CHEMISTRY

An Alkynyliodide Cycloaddition Strategy for the Construction of Iodoisoxazoles

(2010) James A. Crossley et al.   JOURNAL OF ORGANIC CHEMISTRY

Development of Stable Phosphohistidine Analogues

(2010) Jung-Min Kee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of Sporolide B and 9-epi-Sporolide B

(2010) K. C. Nicolaou et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Electronic effects of ruthenium-catalyzed [3+2]-cycloaddition of alkynes and azides

(2010) Duen-Ren Hou et al.   TETRAHEDRON

Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes

(2009) Jason E. Hein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Probing the Bioactive Conformation of an Archetypal Natural Product HDAC Inhibitor with Conformationally Homogeneous Triazole-Modified Cyclic Tetrapeptides

(2009) W. Seth Horne et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of highly enantiomerically enriched planar chiral ruthenium complexes via Pd-catalysed asymmetric hydrogenolysis

(2009) Audrey Mercier et al.   CHEMICAL COMMUNICATIONS

Synthesis and Characterization of Isomeric Vinyl-1,2,3-triazole Materials by Azide−Alkyne Click Chemistry

(2009) Hunaid Nulwala et al.   MACROMOLECULES

Ruthenium-Catalyzed Cycloaddition of Nitrile Oxides and Alkynes: Practical Synthesis of Isoxazoles

(2008) Scott Grecian et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A cycloaddition route to novel triazole boronic esters

(2008) Jianhui Huang et al.   CHEMICAL COMMUNICATIONS

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Ruthenium Complexes Bearing Bulky Pentasubstituted Cyclopentadienyl Ligands and Evaluation of [Ru(η5‐C5Me4R)(MeCN)3][PF6] Precatalysts in Nucleophilic Allylic Substitution Reactions

(2008) Hui‐Jun Zhang et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Alkynyl Halides in Ruthenium(II)-Catalyzed [2+2] Cycloadditions of Bicyclic Alkenes

(2008) Anna Allen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Rhodium-Catalyzed Transannulation of 1,2,3-Triazoles with Nitriles

(2008) Tony Horneff et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hyperbranched Polytriazoles: Click Polymerization, Regioisomeric Structure, Light Emission, and Fluorescent Patterning

(2008) Anjun Qin et al.   MACROMOLECULES

Divergent synthesis of chiral spiro (isoxazole–isoxazoline) hybrid ligands

(2008) Kazuhiro Takenaka et al.   TETRAHEDRON-ASYMMETRY

Synthesis of multiply functionalized benzenes via ruthenium-catalyzed cycloaddition of diiododiynes

(2007) Yoshihiko Yamamoto et al.   TETRAHEDRON