Reaction of Alkynes and Azides: Not Triazoles Through Copper-Acetylides but Oxazoles Through Copper-Nitrene Intermediates

Direct Evidence of a Dinuclear Copper Intermediate in Cu(I)-Catalyzed Azide-Alkyne Cycloadditions

(2013) B. T. Worrell et al.   SCIENCE

Direct Functionalization Processes: A Journey from Palladium to Copper to Iron to Nickel to Metal-Free Coupling Reactions

(2012) James J. Mousseau et al.   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis of Oxazoles through Copper-Mediated Aerobic Oxidative Dehydrogenative Annulation and Oxygenation of Aldehydes and Amines

(2012) Zejun Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

1,3-Azoles from ortho-naphthoquinones: Synthesis of aryl substituted imidazoles and oxazoles and their potent activity against Mycobacterium tuberculosis

(2012) Kelly C.G. Moura et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Efficient synthesis of oxazoles by dirhodium(ii)-catalyzed reactions of styryl diazoacetate with oximes

(2012) Xinfang Xu et al.   CHEMICAL COMMUNICATIONS

New Polyamides and Polyoxazoles Based on Diphenyl Ether Segments in the Polymers' Backbone

(2012) Mahmoud A. Hussein et al.   International Journal of Polymeric Materials and Polymeric Biomaterials

Room Temperature Copper(II)-Catalyzed Oxidative Cyclization of Enamides to 2,5-Disubstituted Oxazoles via Vinylic C–H Functionalization

(2012) Chi Wai Cheung et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Oxazoles from Enamides via Phenyliodine Diacetate-Mediated Intramolecular Oxidative Cyclization

(2012) Yunhui Zheng et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2,5-Disubstituted Oxazoles and Oxazolines Catalyzed by Ruthenium(II) Porphyrin and Simple Copper Salts

(2012) Chuan Long Zhong et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper(ii)-mediated oxidative cyclization of enamides to oxazoles

(2012) Alison E. Wendlandt et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Catalyst-Free Intramolecular Oxidative Cyclization of N-Allylbenzamides: A New Route to 2,5-Substituted Oxazoles

(2012) Wei Zhou et al.   ORGANIC LETTERS

Facile, Selective, and Regiocontrolled Synthesis of Oxazolines and Oxazoles Mediated by ZnI2 and FeCl3

(2012) Gopal Chandru Senadi et al.   ORGANIC LETTERS

Ugi/Robinson–Gabriel reactions directed toward the synthesis of 2,4,5-trisubstituted oxazoles

(2012) Arthur Y. Shaw et al.   TETRAHEDRON LETTERS

Copper-catalyzed oxidative [2 + 2 + 1] cycloaddition: regioselective synthesis of 1,3-oxazoles from internal alkynes and nitriles

(2012) Xianwei Li et al.   Chemical Science

The Synthesis of Aromatic Heterocycles from Propargylic Compounds

(2012) Wen Jia-Jie et al.   Asian Journal of Organic Chemistry

Three Ring Posttranslational Circuses: Insertion of Oxazoles, Thiazoles, and Pyridines into Protein-Derived Frameworks

(2011) Christopher T. Walsh et al.   ACS Chemical Biology

Intermolecular and Selective Synthesis of 2,4,5-Trisubstituted Oxazoles by a Gold-Catalyzed Formal [3+2] Cycloaddition

(2011) Paul W. Davies et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Strategies for the Construction of Optically Active Imidazoles, Oxazoles, and Thiazoles

(2011) Łukasz Albrecht et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Silver-Mediated One-Step Synthesis of Oxazoles

(2011) Dougal J. Ritson et al.   JOURNAL OF ORGANIC CHEMISTRY

An Efficient [2 + 2 + 1] Synthesis of 2,5-Disubstituted Oxazoles via Gold-Catalyzed Intermolecular Alkyne Oxidation

(2011) Weimin He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Muscarine, imidazole, oxazole, and thiazole alkaloids

(2011) Zhong Jin   NATURAL PRODUCT REPORTS

Synthesis of a family of cyclic peptide-based anion receptors

(2011) Stephen J. Butler et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Environmental-benign oxidation of 2-oxazolines to oxazoles by dioxygen as the sole oxidant

(2011) Yue Huang et al.   TETRAHEDRON

Metal-catalyzed direct alkylations of (hetero)arenes via C–H bond cleavages with unactivated alkyl halides

(2010) Lutz Ackermann   CHEMICAL COMMUNICATIONS

Copper-catalyzed azide–alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(i) acetylides

(2010) Jason E. Hein et al.   CHEMICAL SOCIETY REVIEWS

Macrocyclic Pyridyl Polyoxazoles: Selective RNA and DNA G-Quadruplex Ligands as Antitumor Agents

(2010) Suzanne G. Rzuczek et al.   JOURNAL OF MEDICINAL CHEMISTRY

Tailored Ligand Acceleration of the Cu-Catalyzed Azide−Alkyne Cycloaddition Reaction: Practical and Mechanistic Implications

(2010) Stanislav I. Presolski et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regioselective Formation of 2,5-Disubstituted Oxazoles Via Copper(I)-Catalyzed Cycloaddition of Acyl Azides and 1-Alkynes

(2010) Israel Cano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Telomestatin: Formal Total Synthesis and Cation-Mediated Interaction of Itsseco-Derivatives with G-Quadruplexes

(2010) Jörg Linder et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Direct Synthesis of Oxazoles from Aldehydes

(2010) Thomas H. Graham   ORGANIC LETTERS

Simple and Efficient Preparation of 2,5-Disubstituted Oxazoles via a Metal-Free-Catalyzed Cascade Cyclization

(2010) Changfeng Wan et al.   ORGANIC LETTERS

Efficient Synthesis of 1-Sulfonyl-1,2,3-triazoles

(2010) Jessica Raushel et al.   ORGANIC LETTERS

TBHP/I2-Mediated Domino Oxidative Cyclization for One-Pot Synthesis of Polysubstituted Oxazoles

(2010) Huanfeng Jiang et al.   ORGANIC LETTERS

Intramolecular Fe(II)-Catalyzed N−O or N−N Bond Formation from Aryl Azides

(2010) Benjamin J. Stokes et al.   ORGANIC LETTERS

Fluorinated high-performance polymers: Poly(arylene ether)s and aromatic polyimides containing trifluoromethyl groups

(2010) Mahua G. Dhara et al.   PROGRESS IN POLYMER SCIENCE

Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds

(2009) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Isothiourea-Catalyzed Enantioselective Carboxy Group Transfer

(2009) Caroline Joannesse et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and antifungal activity of benzo[d]oxazole-4,7-diones

(2009) Chung-Kyu Ryu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Recent Applications of Oxazoline-Containing Ligands in Asymmetric Catalysis

(2009) Gráinne C. Hargaden et al.   CHEMICAL REVIEWS

Three-Component Synthesis of Highly Functionalized 5-Acetyloxazoles

(2009) Tilman Lechel et al.   CHEMISTRY-A EUROPEAN JOURNAL

Cyclization of Propargylic Amides: Mild Access to Oxazole Derivatives

(2009) Jan P. Weyrauch et al.   CHEMISTRY-A EUROPEAN JOURNAL

Highly active copper-catalysts for azide-alkynecycloaddition

(2009) Zsombor Gonda et al.   DALTON TRANSACTIONS

Copper Complexes with Neutral N4 Tripodal Ligands: Influence of the Number of Nitrogen Donors on Their Structures, Properties, and Reactivity

(2009) Kiyoshi Fujisawa et al.   EUROPEAN JOURNAL OF INORGANIC CHEMISTRY

Novel 2,4,5-trisubstituted oxazole derivatives: Synthesis and antiproliferative activity

(2009) Xin-Hua Liu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

An expeditious synthesis and anticancer activity of novel 4-(3′-indolyl)oxazoles

(2009) Dalip Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Establishment of Broadly Applicable Reaction Conditions for the Palladium-Catalyzed Direct Arylation of Heteroatom-Containing Aromatic Compounds

(2009) Benoît Liégault et al.   JOURNAL OF ORGANIC CHEMISTRY

Brønsted Acid-Catalyzed Propargylation/Cycloisomerization Tandem Reaction: One-Pot Synthesis of Substituted Oxazoles from Propargylic Alcohols and Amides

(2009) Ying-ming Pan et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium Carbene Routes to Oxazoles and Thiazoles. Catalyst Effects in the Synthesis of Oxazole and Thiazole Carboxylates, Phosphonates, and Sulfones

(2009) Baolu Shi et al.   JOURNAL OF ORGANIC CHEMISTRY

A Combined Theoretical and Experimental Study on the Role of Spin States in the Chemistry of Fe(CO)5Photoproducts

(2009) Maria Besora et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Facile Synthesis of 2,4-Disubstituted Thiazoles Using MnO2

(2009) Yan-Bo Yu et al.   MOLECULES

Muscarine, imidazole, oxazole and thiazole alkaloids

(2009) Zhong Jin   NATURAL PRODUCT REPORTS

Copper(i) complexes as catalysts for the synthesis of N-sulfonyl-1,2,3-triazoles from N-sulfonylazides and alkynes

(2009) Israel Cano et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Dehydrative cyclization of serine, threonine, and cysteine residues catalyzed by molybdenum(VI) oxo compounds

(2009) Akira Sakakura et al.   TETRAHEDRON

Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed C−H Bond Activation

(2008) Jared C. Lewis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Copper-Catalyzed Cycloaddition of Sulfonyl Azides with Alkynes to SynthesizeN-Sulfonyltriazoles ‘on Water’ at Room Temperature

(2008) Feng Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Mechanistic study on dimerization of acetylene with a Nieuwland catalyst

(2008) Takashi Tachiyama et al.   APPLIED ORGANOMETALLIC CHEMISTRY

A versatile synthesis of 2,4-substituted oxazoles

(2008) Vijay Chudasama et al.   CHEMICAL COMMUNICATIONS

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Modular Synthesis of Tetrasubstituted Imidazoles and Trisubstituted Oxazoles by Aldimine Cross-Coupling

(2008) Coralie Kison et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Natural Product Derivatives Containing 2,4‐Concatenated Oxazoles

(2008) Delia Hernández et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Mechanistic Studies on the Cu-Catalyzed Three-Component Reactions of Sulfonyl Azides, 1-Alkynes and Amines, Alcohols, or Water: Dichotomy via a Common Pathway

(2008) Eun Jeong Yoo et al.   JOURNAL OF ORGANIC CHEMISTRY

Polymer “Clicking” by CuAAC Reactions

(2008) Morten Meldal   MACROMOLECULAR RAPID COMMUNICATIONS

Total synthesis of siphonazole and its O-methyl derivative, structurally unusual bis-oxazole natural products

(2008) Jörg Linder et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Triflic anhydride-mediated synthesis of oxazoles

(2008) Armin Thalhammer et al.   TETRAHEDRON LETTERS