A cascade approach to fused indolizinones through Lewis acid–copper(i) relay catalysis

Rhodium(III)-Catalyzed Intramolecular Annulation through CH Activation: Total Synthesis of (±)-Antofine, (±)-Septicine, (±)-Tylophorine, and Rosettacin

(2012) Xianxiu Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Lewis Acid Catalyzed Intramolecular [4+2] and [3+2] Cross-Cycloaddition of Alkynylcyclopropane Ketones with Carbonyl Compounds and Imines

(2012) Yu Bai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Pyrido[1,2-a]indole Malonates and Amines through Aryne Annulation

(2012) Donald C. Rogness et al.   JOURNAL OF ORGANIC CHEMISTRY

Cu(OTf)2-catalysed Ritter reaction: efficient synthesis of amides from nitriles and halohydrocarbons in water

(2012) Gui-Rong Qu et al.   RSC Advances

Lewis Acid Catalyzed Intramolecular [3+2] Cross-Cycloaddition of Donor-Acceptor Cyclopropanes with Carbonyls: A General Strategy for the Construction of Acetal[n.2.1] Skeletons

(2011) Siyang Xing et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Palladium-Catalyzed Aminoalkynylation Strategy towards Bicyclic Heterocycles: Synthesis of (±)-Trachelanthamidine

(2011) Stefano Nicolai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rh(I)-Catalyzed Formal [5 + 1]/[2 + 2 + 1] Cycloaddition of 1-Yne-vinylcyclopropanes and Two CO Units: One-Step Construction of Multifunctional Angular Tricyclic 5/5/6 Compounds

(2011) Mu Lin et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Rh(I)-Catalyzed Intramolecular [3 + 2] Cycloaddition of 1-Yne-vinylcyclopropanes for Bicyclo[3.3.0] Compounds with a Chiral Quaternary Carbon Stereocenter and Density Functional Theory Study of the Origins of Enantioselectivity

(2011) Mu Lin et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Brønsted acid assisted activation of imide carbonyl group: regioselective synthesis of isoindoloisoquinolinone alkaloid (±)-nuevamine

(2011) Jayaraman Selvakumar et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Highly Diastereoselective Synthesis of 1-PyrrolinesviaSnCl4-Promoted [3 + 2] Cycloaddition between Activated Donor–Acceptor Cyclopropanes and Nitriles

(2011) Gopal Sathishkannan et al.   ORGANIC LETTERS

Cyclopropane−Aldehyde Annulations at Quaternary Donor Sites: Stereoselective Access to Highly Substituted Tetrahydrofurans

(2011) Austin G. Smith et al.   ORGANIC LETTERS

Rhodium(I)-Catalyzed Intramolecular [5+2] Cycloaddition Reactions of Alkynes and Allenylcyclopropanes: Construction of Bicyclo[5.4.0]undecatrienes and Bicyclo[5.5.0]dodecatrienes

(2010) Fuyuhiko Inagaki et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient Construction of Oxa- and Aza-[n.2.1] Skeletons: Lewis Acid Catalyzed Intramolecular [3+2] Cycloaddition of Cyclopropane 1,1-Diesters with Carbonyls and Imines

(2010) Siyang Xing et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dynamic Kinetic Asymmetric Synthesis of Substituted Pyrrolidines from Racemic Cyclopropanes and Aldimines: Reaction Development and Mechanistic Insights

(2010) Andrew T. Parsons et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Density Functional Theory Study of the Mechanisms and Stereochemistry of the Rh(I)-Catalyzed Intramolecular [3+2] Cycloadditions of 1-Ene- and 1-Yne-Vinylcyclopropanes

(2010) Lei Jiao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 5-Azaindoles via a Cycloaddition Reaction between Nitriles and Donor−Acceptor Cyclopropanes

(2010) Mahmoud M. Abd Rabo Moustafa et al.   ORGANIC LETTERS

Reaction of α-Ene-Vinylcyclopropanes: Type II Intramolecular [5+2] Cycloaddition or [3+2] Cycloaddition?

(2010) Qian Li et al.   ORGANIC LETTERS

Rh(I)-Catalyzed [(3 + 2) + 1] Cycloaddition of 1-Yne/Ene-vinylcyclopropanes and CO: Homologous Pauson−Khand Reaction and Total Synthesis of (±)-α-Agarofuran

(2010) Lei Jiao et al.   ORGANIC LETTERS

Synthesis and SAR of Benzisothiazole- and Indolizine-β-d-glucopyranoside Inhibitors of SGLT2

(2010) Huiqiang Zhou et al.   ACS Medicinal Chemistry Letters

Total Synthesis of Indolizidine Alkaloid (−)-209D: Overriding Substrate Bias in the Asymmetric Rhodium-Catalyzed [2+2+2] Cycloaddition

(2009) Robert T. Yu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Copper-Catalyzed Tandem Synthesis of Indolo- and Pyrrolo[2,1-a]isoquinolines

(2009) Akhilesh Kumar Verma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Identification and Characterization of Novel Small Molecules as Potent Inhibitors of the Plasmodial Calcium-Dependent Protein Kinase 1

(2009) Guillaume Lemercier et al.   BIOCHEMISTRY

Heterocycles from cyclopropanes: applications in natural product synthesis

(2009) Cheryl A. Carson et al.   CHEMICAL SOCIETY REVIEWS

Synthesis of Tetrahydropyrans from Propargyl Alcohols and 1,1-Cyclopropanediesters: A One-Pot Ring-Opening/Conia-ene Protocol

(2009) Andrew B. Leduc et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Schmidt Reaction Involving Primary Azidoalcohols under Nonacidic Conditions: Synthesis of Indolizidine (−)-167B

(2009) Ajoy Kapat et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Enantioselective Synthesis of Tetrahydrofurans: A Dynamic Kinetic Asymmetric [3 + 2] Cycloaddition of Racemic Cyclopropanes and Aldehydes

(2009) Andrew T. Parsons et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Brønsted Acid-CatalyzedN-Acyliminium Cyclization Cascades

(2009) Michael E. Muratore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Zn(II)-Catalyzed Synthesis of Piperidines from Propargyl Amines and Cyclopropanes

(2009) Terry P. Lebold et al.   ORGANIC LETTERS

Ritter-type amidation of alkylboron derivatives with nitriles

(2009) Clément Cazorla et al.   TETRAHEDRON LETTERS

Solid-Phase Synthesis of Aryl-Substituted Thienoindolizines: Sequential Pictet−Spengler, Bromination and Suzuki Cross-Coupling Reactions of Thiophenes

(2008) Sebastian T. Le Quement et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

Stereodivergent Methodology for the Synthesis of Complex Pyrrolidines

(2008) Stephen K. Jackson et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rh(I)-Catalyzed Intramolecular [3 + 2] Cycloaddition oftrans-Vinylcyclopropane-enes

(2008) Lei Jiao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Scope and Mechanism for Lewis Acid-Catalyzed Cycloadditions of Aldehydes and Donor−Acceptor Cyclopropanes: Evidence for a Stereospecific Intimate Ion Pair Pathway

(2008) Patrick D. Pohlhaus et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (±)-Goniomitine via a Formal Nitrile/Donor−Acceptor Cyclopropane [3 + 2] Cyclization

(2007) Christian L. Morales et al.   ORGANIC LETTERS