Nature-inspired cascade catalysis: reaction control through substrate concentration—double vs. quadruple domino reactions

Organocatalytic asymmetric synthesis of polyfunctionalized 3-(cyclohexenylmethyl)-indoles via a quadruple domino Friedel–Crafts-type/Michael/Michael/aldol condensation reaction

(2010) Dieter Enders et al.   CHEMICAL COMMUNICATIONS

Organocatalytic Tandem Reaction to Construct Six-Membered Spirocyclic Oxindoles with Multiple Chiral Centres through a Formal [2+2+2] Annulation

(2010) Kun Jiang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric Domino Michael-Henry Reaction: Enantioselective Access to Bicycles with Consecutive Quaternary Centers by Using Bifunctional Catalysts

(2010) Magnus Rueping et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric Mannich-Ketalization Reaction: Highly Enantioselective Synthesis of Aminobenzopyrans

(2010) Magnus Rueping et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric organocatalysis in total synthesis – a trial by fire

(2010) Eugenia Marqués-López et al.   NATURAL PRODUCT REPORTS

Organocatalytic cascade reactions as a new tool in total synthesis

(2010) Christoph Grondal et al.   Nature Chemistry

Enantioselective Total Synthesis of (+)-Conicol via Cascade Three-Component Organocatalysis

(2010) Bor-Cherng Hong et al.   ORGANIC LETTERS

Asymmetric Quadruple Aminocatalytic Domino Reactions to Fused Carbocycles Incorporating a Spirooxindole Motif

(2010) Kun Jiang et al.   ORGANIC LETTERS

Fast, Efficient, Mild, and Metal-Free Synthesis of Pyrroles by Domino Reactions in Water

(2010) Magnus Rueping et al.   ORGANIC LETTERS

Catalytic Asymmetric Domino Michael Addition−Alkylation Reaction: Enantioselective Synthesis of Dihydrofurans

(2010) Magnus Rueping et al.   ORGANIC LETTERS

Thieme Chemistry Journal Awardees - Where Are They Now? Asymmetric Brønsted Acid Catalyzed Transfer Hydrogenations

(2010) Magnus Rueping et al.   SYNLETT

Hydride-Donor Abilities of 1,4-Dihydropyridines: A Comparison with π Nucleophiles and Borohydride Anions

(2009) Dorothea Richter et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Organocatalytic Domino Michael/Aldol Reactions: Enantioselective Synthesis of Chiral Cycloheptanones, Tetrahydrochromenones, and Polyfunctionalized Bicyclo[3.2.1]octanes

(2009) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Targeting Structural and Stereochemical Complexity by Organocascade Catalysis: Construction of Spirocyclic Oxindoles Having Multiple Stereocenters

(2009) Giorgio Bencivenni et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Principles, implementation, and application of biology-oriented synthesis (BIOS)

(2009) Wolfram Wilk et al.   BIOLOGICAL CHEMISTRY

Asymmetric Organocatalytic Four-Component Quadruple Domino Reaction Initiated by Oxa-Michael Addition of Alcohols to Acrolein

(2009) Fang-Lin Zhang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic Domino Reactions

(2009) Andrea-Nekane Alba et al.   CURRENT ORGANIC CHEMISTRY

Asymmetric Synthesis of Polyfunctionalized Mono-, Bi-, and Tricyclic Carbon Frameworksvia Organocatalytic Domino Reactions

(2008) Dieter Enders et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Organocatalytic Reactions of 4-Hydroxycoumarin and 4-Hydroxypyrone with α,β-Unsaturated Aldehydes - An Efficient Michael Addition-Acetalization Cascade to Chromenones, Quinolinones and Pyranones

(2008) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

Biology-inspired synthesis of compound libraries

(2008) M. Kaiser et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

Quaternary Stereogenic Carbon Atoms in Complex Molecules by an Asymmetric, Organocatalytic, Triple-Cascade Reaction

(2008) Oriol Penon et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric Organocatalysis: An Efficient Enantioselective Access to Benzopyranes and Chromenes

(2008) Magnus Rueping et al.   CHEMISTRY-A EUROPEAN JOURNAL

Broader, Greener, and More Efficient: Recent Advances in Asymmetric Transfer Hydrogenation

(2008) Chao Wang et al.   Chemistry-An Asian Journal

α,α-Diarylprolinol Ethers: New Tools for Functionalization of Carbonyl Compounds

(2008) Antonia Mielgo et al.   Chemistry-An Asian Journal

Organocatalysis: asymmetric cascade reactions catalysed by chiral secondary amines

(2008) Xinhong Yu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective synthesis of the tetrahydro-6H-benzo[c]chromenes via Domino Michael–Aldol condensation: control of five stereocenters in a quadruple-cascade organocatalytic multi-component reaction

(2008) Prakash Kotame et al.   TETRAHEDRON LETTERS

Towards the Optimal Screening Collection: A Synthesis Strategy

(2007) Thomas E. Nielsen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

MacMillan’s Imidazolidinones: Powerful Chiral Organocatalysts

(2007) Thomas Poisson   SYNLETT