期刊
CHEMICAL BIOLOGY & DRUG DESIGN
卷 82, 期 5, 页码 477-499出版社
WILEY
DOI: 10.1111/cbdd.12180
关键词
anticancer activity; blister beetles; cantharidin analogs; Diels-Alder cycloaddition reactions; drug design and development; protein phosphatases inhibitory activity
资金
- Patrimonio Autonomo Fondo Nacional de Financiamiento para la Ciencia, la Tecnologia y la Innovacion, Francisco Jose de Caldas [RC-0572-2012]
- COLCIENCIAS
Chemical and pharmacological information on cantharidin-based small molecules was analyzed. The review summarizes new facts about blister beetles' metabolites for the period 2006-2012. General synthetic approaches to cantharidin-based small molecules as well as their chemical transformations and biological activities related to cantharidin, norcantharidin, cantharidimide, and norcantharimide analogs, especially their inhibitory activity of phosphoprotein phosphatases in cancer treatment, were discussed in this mini review, which could help to design new small molecule modulators for other biological models.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据