The Concise Guide to PHARMACOLOGY 2013/14: Nuclear Hormone Receptors

T0901317, a potent LXR agonist, is an inverse agonist of CAR

(2013) Yuichiro Kanno et al.   JOURNAL OF TOXICOLOGICAL SCIENCES

HNF4α Antagonists Discovered by a High-Throughput Screen for Modulators of the Human Insulin Promoter

(2012) Alice Kiselyuk et al.   CHEMISTRY & BIOLOGY

GSK4112, a Small Molecule Chemical Probe for the Cell Biology of the Nuclear Heme Receptor Rev-erbα

(2010) Daniel Grant et al.   ACS Chemical Biology

The Orphan Nuclear Receptor TR4 Is a Vitamin A-activated Nuclear Receptor

(2010) X. Edward Zhou et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Profile of ligand specificity of the vitamin D binding protein for 1α,25-dihydroxyvitamin d3 and its analogs

(2010) June E. Bishop et al.   JOURNAL OF BONE AND MINERAL RESEARCH

Differential Action on Coregulator Interaction Defines Inverse Retinoid Agonists and Neutral Antagonists

(2009) Pierre Germain et al.   CHEMISTRY & BIOLOGY

Non-genomic signaling by steroids

(2009) Eric R. Prossnitz et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Identification of an Endogenous Ligand Bound to a Native Orphan Nuclear Receptor

(2009) Xiaohui Yuan et al.   PLoS One

Rapid signaling by steroid receptors

(2008) Ellis R. Levin   AMERICAN JOURNAL OF PHYSIOLOGY-REGULATORY INTEGRATIVE AND COMPARATIVE PHYSIOLOGY

Estrogen Signaling through the Transmembrane G Protein–Coupled Receptor GPR30

(2008) Eric R. Prossnitz et al.   Annual Review of Physiology

Rational Design and Synthesis of 4-((1R,2R)-2-Hydroxycyclohexyl)-2(trifluoromethyl)benzonitrile (PF-998425), a Novel, Nonsteroidal Androgen Receptor Antagonist Devoid of Phototoxicity for Dermatological Indications

(2008) Jie Jack Li et al.   JOURNAL OF MEDICINAL CHEMISTRY

Potent, Selective and Cell Penetrant Inhibitors of SF-1 by Functional Ultra-High-Throughput Screening

(2008) F. Madoux et al.   MOLECULAR PHARMACOLOGY

Molecular Characterization of Novel and Selective Peroxisome Proliferator-Activated Receptor   Agonists with Robust Hypolipidemic Activity in Vivo

(2008) C. D. Kane et al.   MOLECULAR PHARMACOLOGY

Cytosporone B is an agonist for nuclear orphan receptor Nur77

(2008) Yanyan Zhan et al.   Nature Chemical Biology

Heterologous expression of human mPRα, mPRβ and mPRγ in yeast confirms their ability to function as membrane progesterone receptors

(2008) Jessica L. Smith et al.   STEROIDS

Identification and Characterization of a Selective Peroxisome Proliferator-Activated Receptor β/δ (NR1C2) Antagonist

(2007) Barry G. Shearer et al.   MOLECULAR ENDOCRINOLOGY

Biological activities of a novel selective oestrogen receptor modulator derived from raloxifene (Y134)

(2006) M Ning et al.   BRITISH JOURNAL OF PHARMACOLOGY