期刊
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
卷 19, 期 24, 页码 6935-6938出版社
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.bmcl.2009.10.067
关键词
Serotonin; 5-HT6 receptor; Pyrrolo[2,3-c]pyridine; Pyrrolo[3,2-b]pyridine; Pyrrolo[3,2-c]pyridine; Agonist; Antagonist; Sulfone
1-(2-Aminoethyl)-3-(arylsulfonyl)-1H-pyrrolopyridines were prepared. Binding assays indicated they are 5-HT6 receptor ligands, among which 6f and 6g showed high affinity for 5-HT6 receptors with K-i = 3.9 and 1.7 nM, respectively. (C) 2009 Elsevier Ltd. All rights reserved.
作者
我是这篇论文的作者
点击您的名字以认领此论文并将其添加到您的个人资料中。
推荐
暂无数据