Copper-Mediated C6-Selective Dehydrogenative Heteroarylation of 2-Pyridones with 1,3-Azoles

Copper-catalyzed ortho-C–H amination of protected anilines with secondary amines

(2014) Ángel Manu Martínez et al.   CHEMICAL COMMUNICATIONS

Palladium catalyzed C3-arylation of 4-hydroxy-2-pyridones

(2014) Elissavet E. Anagnostaki et al.   CHEMICAL COMMUNICATIONS

Manganese-Mediated C3-Selective Direct Alkylation and Arylation of 2-Pyridones with Diethyl Malonates and Arylboronic Acids

(2014) Akihiro Nakatani et al.   JOURNAL OF ORGANIC CHEMISTRY

Cu(II)-Mediated C–H Amidation and Amination of Arenes: Exceptional Compatibility with Heterocycles

(2014) Ming Shang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Boron–Heck Reaction of Cyclic Enaminones: Regioselective Direct Arylation via Oxidative Palladium(II) Catalysis

(2014) Yong Wook Kim et al.   ORGANIC LETTERS

Synthesis of Carbazoles by Copper-Catalyzed Intramolecular C–H/N–H Coupling

(2014) Kazutaka Takamatsu et al.   ORGANIC LETTERS

Copper-Catalyzed Carboxamide-Directed Ortho Amination of Anilines with Alkylamines at Room Temperature

(2014) Qiong Li et al.   ORGANIC LETTERS

Copper-Mediated Direct Arylation of Azole Compounds

(2014) Koji Hirano et al.   TOPICS IN CATALYSIS

Directed Amination of Non-Acidic Arene CH Bonds by a Copper-Silver Catalytic System

(2013) Ly Dieu Tran et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Mediated CH/CH Biaryl Coupling of Benzoic Acid Derivatives and 1,3-Azoles

(2013) Mayuko Nishino et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-catalyzed ortho-halogenation of protected anilines

(2013) Beatriz Urones et al.   CHEMICAL COMMUNICATIONS

Nickel-Catalyzed Direct Alkylation of Heterocycles with α-Bromo Carbonyl Compounds: C3-Selective Functionalization of 2-Pyridones

(2013) Akihiro Nakatani et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Mediated Regioselective Homocoupling of Thiophenes and Indoles via Directed C–H Cleavage

(2013) Masahiro Miura et al.   HETEROCYCLES

Copper-Mediated Dehydrogenative Biaryl Coupling of Naphthylamines and 1,3-Azoles

(2013) Riko Odani et al.   JOURNAL OF ORGANIC CHEMISTRY

Removal of the Pyridine Directing Group from α-Substituted N-(Pyridin-2-yl)piperidines Obtained via Directed Ru-Catalyzed sp3 C–H Functionalization

(2013) Veerle Smout et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed, Directing Group-Assisted Fluorination of Arene and Heteroarene C–H Bonds

(2013) Thanh Truong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Etherification of Arene C–H Bonds

(2013) James Roane et al.   ORGANIC LETTERS

Rhodium or Ruthenium-Catalyzed Oxidative CH/CH Cross-Coupling: Direct Access to Extended π-Conjugated Systems

(2012) Jiaxing Dong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Mediated and Copper-Catalyzed Cross-Coupling of Indoles and 1,3-Azoles: Double CH Activation

(2012) Mayuko Nishino et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Alkylation of Pyridone Derivatives By Nickel/Lewis Acid Catalysis

(2012) Ryuichi Tamura et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

[RhIIICp*]-Catalyzed Dehydrogenative ArylAryl Bond Formation

(2012) Joanna Wencel-Delord et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals

(2012) Junichiro Yamaguchi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-mediated oxidative direct C–C (hetero)aromatic cross-coupling

(2012) Koji Hirano et al.   CHEMICAL COMMUNICATIONS

Discovery of 2-(2-Oxo-1-phenyl-5-pyridin-2-yl-1,2-dihydropyridin-3-yl)benzonitrile (Perampanel): A Novel, Noncompetitive α-Amino-3-hydroxy-5-methyl-4-isoxazolepropanoic Acid (AMPA) Receptor Antagonist

(2012) Shigeki Hibi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed C–H Azidation of Anilines under Mild Conditions

(2012) Conghui Tang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Promoted Sulfenylation of sp2 C–H Bonds

(2012) Ly Dieu Tran et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-catalyzed selective oxidative olefination and arylation of 2-pyridones

(2012) Yuye Chen et al.   Chemical Science

Efficient synthesis of biazoles by aerobic oxidative homocoupling of azoles catalyzed by a copper(i)/2-pyridonate catalytic system

(2011) Mingwen Zhu et al.   CHEMICAL COMMUNICATIONS

Bond Formations between Two Nucleophiles: Transition Metal Catalyzed Oxidative Cross-Coupling Reactions

(2011) Chao Liu et al.   CHEMICAL REVIEWS

Oxidative C–H/C–H Coupling of Azine and Indole/Pyrrole Nuclei: Palladium Catalysis and Synthesis of Eudistomin U

(2011) Atsushi D. Yamaguchi et al.   CHEMISTRY LETTERS

Copper-Mediated Intermolecular Direct Biaryl Coupling

(2011) Masanori Kitahara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Nucleophilic Aryl Fluorination and Aryl Halide Exchange Mediated by a CuI/CuIIICatalytic Cycle

(2011) Alicia Casitas et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Highly Regioselective Oxidative CH Bond Amidation of 2-Arylpyridine Derivatives and 1-Methylindoles

(2010) Qi Shuai et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis and biological evaluation of N-difluoromethyl-1,2-dihydropyrid-2-one acetic acid regioisomers: Dual Inhibitors of cyclooxygenases and 5-lipoxygenase

(2010) Gang Yu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Pd-catalyzed oxidative coupling with organometallic reagents via C–H activation

(2010) Chang-Liang Sun et al.   CHEMICAL COMMUNICATIONS

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

(2010) Thomas W. Lyons et al.   CHEMICAL REVIEWS

Overview of the Mechanistic Work on the Concerted Metallation–Deprotonation Pathway

(2010) David Lapointe et al.   CHEMISTRY LETTERS

Oxidative Coupling of Aromatic Substrates with Alkynes and Alkenes under Rhodium Catalysis

(2010) Tetsuya Satoh et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper(II)-Catalyzed Ortho-Acyloxylation of the 2-Arylpyridines sp2C−H Bonds with Anhydrides, Using O2as Terminal Oxidant

(2010) Wenhui Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd(OAc)2-Catalyzed Oxidative C−H/C−H Cross-Coupling of Electron-Deficient Polyfluoroarenes with Simple Arenes

(2010) Ye Wei et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Aerobic Oxidative Functionalization of an Arene C−H Bond: Evidence for an Aryl-Copper(III) Intermediate

(2010) Amanda E. King et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

4-Hydroxy-2-pyridone alkaloids: Structures and synthetic approaches

(2010) Henning Jacob Jessen et al.   NATURAL PRODUCT REPORTS

Rational design of small-molecule inhibitors of the LEDGF/p75-integrase interaction and HIV replication

(2010) Frauke Christ et al.   Nature Chemical Biology

Regioselective syntheses of fully-substituted 1,2,3-triazoles: the CuAAC/C–H bond functionalization nexus

(2010) Lutz Ackermann et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Nickel, Manganese, Cobalt, and Iron-Catalyzed Deprotonative Arene Dimerization

(2010) Thanh Truong et al.   ORGANIC LETTERS

Cu(II)-Mediated Methylthiolation of Aryl C−H Bonds with DMSO

(2010) Lingling Chu et al.   ORGANIC LETTERS

Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds

(2009) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium(II)-Catalyzed CH Activation/CC Cross-Coupling Reactions: Versatility and Practicality

(2009) Xiao Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cu(ii)-mediated oxidative intermolecular ortho C–H functionalisation using tetrahydropyrimidine as the directing group

(2009) Tsukasa Mizuhara et al.   CHEMICAL COMMUNICATIONS

Regioselective Halogenations and Subsequent Suzuki−Miyaura Coupling onto Bicyclic 2-Pyridones

(2009) Christoffer Bengtsson et al.   JOURNAL OF ORGANIC CHEMISTRY

Mechanistic Study of Copper-Catalyzed Aerobic Oxidative Coupling of Arylboronic Esters and Methanol: Insights into an Organometallic Oxidase Reaction

(2009) Amanda E. King et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Direct Alkenylation and Alkylation of Pyridone Derivatives by Ni/AlMe3Catalysis

(2009) Yoshiaki Nakao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxidative dimerization of azoles via copper(II)/silver(I)-catalyzed CH homocoupling

(2009) Daiki Monguchi et al.   TETRAHEDRON LETTERS

Direct Functionalization of Nitrogen Heterocycles via Rh-Catalyzed C−H Bond Activation

(2008) Jared C. Lewis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Metal−Organic Cooperative Catalysis in C−H and C−C Bond Activation and Its Concurrent Recovery

(2008) Young Jun Park et al.   ACCOUNTS OF CHEMICAL RESEARCH

New Strategies for the Synthesis of Pyrimidine Derivatives

(2008) Matthew D. Hill et al.   CHEMISTRY-A EUROPEAN JOURNAL

Carbon−Nitrogen Bond Formation Involving Well-Defined Aryl−Copper(III) Complexes

(2008) Lauren M. Huffman et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transition-Metal-Catalyzed Carbon-Carbon Bond Formation via Carbon-Hydrogen Bond Cleavage

(2008) Fumitoshi Kakiuchi et al.   SYNTHESIS-STUTTGART