Copper-Catalyzed Direct Secondary and Tertiary CH Alkylation of Azoles through a Heteroarene-Amine-Aldehyde/Ketone Coupling Reaction

Regio- and Stereocontrolled Introduction of Secondary Alkyl Groups to Electron-Deficient Arenes through Copper-Catalyzed Allylic Alkylation

(2012) Yusuke Makida et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A walk around the A3-coupling

(2012) Vsevolod A. Peshkov et al.   CHEMICAL SOCIETY REVIEWS

Pd/Cu-Catalyzed C–H Arylation of 1,3,4-Thiadiazoles with (Hetero)aryl Iodides, Bromides, and Triflates

(2012) Dipak D. Vachhani et al.   JOURNAL OF ORGANIC CHEMISTRY

Direct Heteroarylation of Tautomerizable Heterocycles into Unsymmetrical and Symmetrical Biheterocycles via Pd/Cu-Catalyzed Phosphonium Coupling

(2012) Abhishek Sharma et al.   ORGANIC LETTERS

Copper-Catalyzed Alkylation of Benzoxazoles with Secondary Alkyl Halides

(2012) Peng Ren et al.   ORGANIC LETTERS

Structure Determination and Interception of Biosynthetic Intermediates for the Plantazolicin Class of Highly Discriminating Antibiotics

(2011) Katie J. Molohon et al.   ACS Chemical Biology

User-Friendly [(Diglyme)NiBr2]-Catalyzed Direct Alkylations of Heteroarenes with Unactivated Alkyl Halides through CH Bond Cleavages

(2011) Lutz Ackermann et al.   ADVANCED SYNTHESIS & CATALYSIS

Nickel- and Cobalt-Catalyzed Direct Alkylation of Azoles with N-Tosylhydrazones Bearing Unactivated Alkyl Groups

(2011) Tomoyuki Yao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Room-Temperature Synthesis of Tetra-ortho-Substituted Biaryls by NHC-Catalyzed Suzuki-Miyaura Couplings

(2011) Linglin Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Metal-Free Route to 2-Aminooxazoles by Taking Advantage of the Unique Ring Opening of Benzoxazoles and Oxadiazoles with Secondary Amines

(2011) Jomy Joseph et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

(2011) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Direct Benzylation or Allylation of 1,3-Azoles withN-Tosylhydrazones

(2011) Xia Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Discovery of a Potent Thiadiazole Class of Histamine H3 Receptor Antagonist for the Treatment of Diabetes

(2011) Ashwin U. Rao et al.   ACS Medicinal Chemistry Letters

The Development of Catalytic Nucleophilic Additions of Terminal Alkynes in Water†

(2010) Chao-Jun Li   ACCOUNTS OF CHEMICAL RESEARCH

Concise and Diversity-Oriented Route toward Polysubstituted 2-Aminoimidazole Alkaloids and Their Analogues

(2010) Denis S. Ermolat'ev et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed Hydroheteroarylation of Vinylarenes

(2010) Yoshiaki Nakao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Formal Inverse Sonogashira Reaction: Direct Alkynylation of Arenes and Heterocycles with Alkynyl Halides

(2010) Alexander S. Dudnik et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Nickel/Copper-Catalyzed Direct Alkylation of Heterocyclic CH Bonds

(2010) Oleg Vechorkin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-catalyzed direct alkylations of (hetero)arenes via C–H bond cleavages with unactivated alkyl halides

(2010) Lutz Ackermann   CHEMICAL COMMUNICATIONS

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

(2010) Thomas W. Lyons et al.   CHEMICAL REVIEWS

Efficient Microwave-Assisted Synthesis of Secondary Alkylpropargylamines by Using A3-Coupling with Primary Aliphatic Amines

(2010) Jitender B. Bariwal et al.   CHEMISTRY-A EUROPEAN JOURNAL

Palladium- and Nickel-Catalyzed Direct Alkylation of Azoles with Unactivated Alkyl Bromides and Chlorides

(2010) Tomoyuki Yao et al.   CHEMISTRY-A EUROPEAN JOURNAL

Selective C-4 Alkylation of Pyridine by Nickel/Lewis Acid Catalysis

(2010) Yoshiaki Nakao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diversity-Oriented Synthesis of Dibenzoazocines and Dibenzoazepines via a Microwave-Assisted Intramolecular A3-Coupling Reaction

(2010) Jitender B. Bariwal et al.   ORGANIC LETTERS

Unprecedented Cu(I)-Catalyzed Microwave-Assisted Three-Component Coupling of a Ketone, an Alkyne, and a Primary Amine

(2010) Olga P. Pereshivko et al.   ORGANIC LETTERS

Palladium-Catalyzed Direct Benzylation of Azoles with Benzyl Carbonates

(2010) Tomoya Mukai et al.   ORGANIC LETTERS

Transition-Metal-Catalyzed Regioselective Arylation and Vinylation of Carboxylic Acids

(2010) Tetsuya Satoh et al.   SYNTHESIS-STUTTGART

Palladium- and Copper-Catalyzed Arylation of Carbon−Hydrogen Bonds

(2009) Olafs Daugulis et al.   ACCOUNTS OF CHEMICAL RESEARCH

Ruthenium-Catalyzed Regioselective Direct Alkylation of Arenes with Unactivated Alkyl Halides through CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophore

(2009) Brian A. Johns et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Rhenium-Catalyzed Regioselective Alkylation of Phenols

(2009) Yoichiro Kuninobu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Consecutive Intramolecular Hydroamination/Asymmetric Transfer Hydrogenation under Relay Catalysis of an Achiral Gold Complex/Chiral Brønsted Acid Binary System

(2009) Zhi-Yong Han et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Mediated Direct Arylation of 1,3,4-Oxadiazoles and 1,2,4-Triazoles with Aryl Iodides

(2009) Tsuyoshi Kawano et al.   ORGANIC LETTERS

Palladium-Catalyzed Benzylation of Heterocyclic Aromatic Compounds

(2009) David Lapointe et al.   ORGANIC LETTERS

Optimization of the Central Heterocycle of α-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase

(2008) Joie Garfunkle et al.   JOURNAL OF MEDICINAL CHEMISTRY

Relay Catalysis by a Metal-Complex/Brønsted Acid Binary System in a Tandem Isomerization/Carbon−Carbon Bond Forming Sequence

(2008) Keiichi Sorimachi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Reactive and Regenerable Fluorinating Agent for Oxidative Fluorination of Aromatics

(2008) Krishna Murthy Janmanchi et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT