Synthesis of Indoles through Highly Efficient Cascade Reactions of Sulfur Ylides and N-(ortho-Chloromethyl)aryl Amides

Gold-Catalyzed Carbene Transfer to Alkynes: Access to 2,4-Disubstituted Furans

(2012) Søren Kramer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Hydrogen-Bond-Mediated Asymmetric Cascade Reaction of Stable Sulfur Ylides with Nitroolefins: Scope, Application and Mechanism

(2012) Liang-Qiu Lu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective Synthesis of Dihydropyrazoles by Formal [4+1] Cycloaddition of in Situ-Derived Azoalkenes and Sulfur Ylides

(2012) Jia-Rong Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium-Catalyzed Synthesis of 2,3-Disubstituted Indoles from β,β-Disubstituted Stryryl Azides

(2011) Ke Sun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structure and activity relationship of 2-(substituted benzoyl)-hydroxyindoles as novel CaMKII inhibitors

(2011) Masafumi Komiya et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Au-catalyzed synthesis of 2-alkylindoles from N-arylhydroxylamines and terminal alkynes

(2011) Yanzhao Wang et al.   CHEMICAL COMMUNICATIONS

Two-Step Route to Indoles and Analogues from Haloarenes: A Variation on the Fischer Indole Synthesis

(2011) Martyn Inman et al.   JOURNAL OF ORGANIC CHEMISTRY

Ionic Diamine Rhodium Complex Catalyzed Reductive N-Heterocyclization of 2-Nitrovinylarenes

(2011) Kazumi Okuro et al.   JOURNAL OF ORGANIC CHEMISTRY

Rh2(II)-Catalyzed Nitro-Group Migration Reactions: Selective Synthesis of 3-Nitroindoles from β-Nitro Styryl Azides

(2011) Benjamin J. Stokes et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Catalytic Asymmetric Fischer Indolization

(2011) Steffen Müller et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Total Synthesis of the Crinine Alkaloid Hamayne via a Pd[0]-Catalyzed Intramolecular Alder-Ene Reaction

(2011) Laurent Petit et al.   ORGANIC LETTERS

Direct annulation and alkylation of indoles with 2-aminobenzyl alcohols catalyzed by TFA

(2011) Forest J. Robertson et al.   TETRAHEDRON

Fischer Indole Synthesis with Organozinc Reagents

(2010) Benjamin A. Haag et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Tuning Electronic and Steric Effects: Highly Enantioselective [4+1] Pyrroline Annulation of Sulfur Ylides with α,β-Unsaturated Imines

(2010) Liang-Qiu Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A two step route to indoles from haloarenes—a versatile variation on the Fischer indole synthesis

(2010) Martyn Inman et al.   CHEMICAL COMMUNICATIONS

Palladium-Catalyzed Amination of Aromatic C−H Bonds with Oxime Esters

(2010) Yichen Tan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (+)-Perophoramidine and Determination of the Absolute Configuration

(2010) Haoxing Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(III)-Catalyzed Arene and Alkene C−H Bond Functionalization Leading to Indoles and Pyrroles

(2010) David R. Stuart et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper catalysis in the construction of indole and benzo[b]furan rings

(2010) Sandro Cacchi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Total Synthesis of (+)-Haplophytine

(2009) Hirofumi Ueda et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Construction of Fused Heterocyclic Architectures by Formal [4+1]/[3+2] Cycloaddition Cascade of Sulfur Ylides and Nitroolefins

(2009) Liang-Qiu Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Concise One-Pot Tandem Synthesis of Indoles and Isoquinolines from Amides

(2009) Noriko Okamoto et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed CC Bond Formation through CH Functionalization: Synthesis of Multisubstituted Indoles fromN-Aryl Enaminones

(2009) Roberta Bernini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Synthesis of 2,2-Disubstituted Oxetanes from Ketones by Using a One-Pot Sequential Addition of Sulfur Ylide

(2009) Toshihiko Sone et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indoles from Simple Anilines and Alkynes: Palladium-Catalyzed CH Activation Using Dioxygen as the Oxidant

(2009) Zhuangzhi Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Functionalized 4-Alkylidenebicyclo[3.1.0]hex-2-enes by Tandem Michael Addition and Annulation of Electron-Deficient Enynes

(2009) Zuliang Chen et al.   Chemistry-An Asian Journal

Modular Synthesis of Indoles from Imines ando-Dihaloarenes oro-Chlorosulfonates by a Pd-Catalyzed Cascade Process

(2009) José Barluenga et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Ylide-Initiated Michael Addition−Cyclization Reactions beyond Cyclopropanes

(2008) Xiu-Li Sun et al.   ACCOUNTS OF CHEMICAL RESEARCH

Catalytic Synthesis of Indoles from Alkynes

(2008) Karolin Krüger (née Alex) et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Indolines and Tetrahydroisoquinolines from Arylethylamines by PdII-Catalyzed CH Activation Reactions

(2008) Jiao-Jie Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Oxidative Cyclization ofN-Aryl Enamines: From Anilines to Indoles

(2008) Sebastian Würtz et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dirhodium(II)-Catalyzed Intramolecular CH Amination of Aryl Azides

(2008) Meihua Shen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Diastereoselective and Enantioselective Formal [4 + 1] Ylide Annulation for the Synthesis of Optically Active Dihydrofurans

(2008) Jun-Cheng Zheng et al.   JOURNAL OF ORGANIC CHEMISTRY

Tandem Michael Addition/Ylide Epoxidation for the Synthesis of Highly Functionalized Cyclohexadiene Epoxide Derivatives

(2008) Qing-Gang Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Indoles via Domino Reaction ofN-Aryl Amides and Ethyl Diazoacetate

(2008) Sun-Liang Cui et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A New Entry to Cascade Organocatalysis: Reactions of Stable Sulfur Ylides and Nitroolefins Sequentially Catalyzed by Thiourea and DMAP

(2008) Liang-Qiu Lu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indole Synthesis via Rhodium Catalyzed Oxidative Coupling of Acetanilides and Internal Alkynes

(2008) David R. Stuart et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Synthesis of 3-Indolecarboxylic Acid Derivatives

(2008) Björn Söderberg et al.   SYNTHESIS-STUTTGART

Palladium-Catalyzed Aryl Amination–Heck Cyclization Cascade: A One-Flask Approach to 3-Substituted Indoles

(2007) Thomas Jensen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Platinum-Catalyzed Formation of Cyclic-Ketone-Fused Indoles fromN-(2-Alkynylphenyl)lactams

(2007) Guotao Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-Pot Multicomponent Synthesis of Indoles from 2-Iodobenzoic Acid

(2007) Olivier Leogane et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION