Benzoylphosphonate-Based Photoactive Phosphopeptide Mimetics for Modulation of Protein Tyrosine Phosphatases and Highly Specific Labeling of SH2 Domains

Dynamic Substrate Enhancement for the Identification of Specific, Second-Site-Binding Fragments Targeting a Set of Protein Tyrosine Phosphatases

(2011) Marco F. Schmidt et al.   CHEMBIOCHEM

Cell Signaling by Receptor Tyrosine Kinases

(2010) Mark A. Lemmon et al.   CELL

Selective Identification of Cooperatively Binding Fragments in a High-Throughput Ligation Assay Enables Development of a Picomolar Caspase-3 Inhibitor

(2009) Marco F. Schmidt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Drug Discovery and Protein Tyrosine Phosphatases

(2009) Mark Blaskovich   CURRENT MEDICINAL CHEMISTRY

Profiling protein tyrosine phosphatase activity with mechanistic probes

(2009) Divya Krishnamurthy et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Dynamic template-assisted strategies in fragment-based drug discovery

(2009) Marco F. Schmidt et al.   TRENDS IN BIOTECHNOLOGY

Sensitized Detection of Inhibitory Fragments and Iterative Development of Non-Peptidic Protease Inhibitors by Dynamic Ligation Screening

(2008) Marco Florian Schmidt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Protein phosphatase inhibitory activity of tautomycin photoaffinity probes evaluated at femto-molar level

(2007) Magne O. Sydnes et al.   BIOORGANIC & MEDICINAL CHEMISTRY