Recent progress for the synthesis of selected carbocyclic nucleosides

Total synthesis of carbocyclic nucleoside (+)-neplanocin A

(2015) Young Hoon Jung et al.   TETRAHEDRON

Stereoselective Synthesis of 2′-Fluoro-6′-methylene Carbocyclic Adenosine via Vince Lactam

(2014) Uma S. Singh et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Neplanocin A and Its 3′-Epimer via an Intramolecular Baylis–Hillman Reaction

(2014) Yun Xuan Tan et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Antiviral Evaluation of Novel 2′,2′-Difluoro 5′-Norcarbocyclic Phosphonic Acid Nucleosides as Antiviral Agents

(2014) Guang Huan Shen et al.   NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS

Advances in the enantioselective synthesis of carbocyclic nucleosides

(2013) Omar Boutureira et al.   CHEMICAL SOCIETY REVIEWS

Total Synthesis of Entecavir

(2013) Javier Velasco et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Evaluation of Novel 6′,6′-Difluoro 5′-Deoxycarbocyclic Phosphonic Acid Nucleosides as Antiviral Agents

(2013) Eunae Kim et al.   NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS

Fluorocyclopentenyl-cytosine with Broad Spectrum and Potent Antitumor Activity

(2012) Won Jun Choi et al.   JOURNAL OF MEDICINAL CHEMISTRY

Stereoselective Synthesis of Fluoro-homoneplanocin A as a Potential Antiviral Agent

(2012) Girish Chandra et al.   ORGANIC LETTERS

2′-Fluoro-3-deazaaristeromycin

(2012) Chun Chen et al.   TETRAHEDRON

A novel and efficient synthesis of Entecavir

(2012) Xiaoyu Liu et al.   TETRAHEDRON LETTERS

Synthesis of the 5′-Fluoro-2′β-methyl Analogues of Neplanocin

(2011) Hiroki Kumamoto et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

X-ray Crystal Structure and Binding Mode Analysis of HumanS-Adenosylhomocysteine Hydrolase Complexed with Novel Mechanism-Based Inhibitors, Haloneplanocin A Analogues

(2011) Kang Man Lee et al.   JOURNAL OF MEDICINAL CHEMISTRY

Design and Synthesis of Carbocyclic Versions of Furanoid Nucleoside Phosphonic Acid Analogues as Potential Anti-Hiv Agents

(2011) Eunae Kim et al.   NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS

Synthesis of 2′,3′-dideoxy-6′-fluorocarbocyclic nucleosides via Reformatskii–Claisen rearrangement

(2011) Yi Yang et al.   TETRAHEDRON

(+)-Neplanocin F, 2′-fluoroneplanocin, and a 6′-isoneplanocin via a common versatile cyclopentenol precursor

(2011) Chong Liu et al.   TETRAHEDRON LETTERS

Hepatitis B Virus Resistance to Nucleos(t)ide Analogues

(2009) Fabien Zoulim et al.   GASTROENTEROLOGY

Long-term monitoring shows hepatitis B virus resistance to entecavir in nucleoside-naïve patients is rare through 5 years of therapy

(2009) Daniel J. Tenney et al.   HEPATOLOGY

Synthesis of Nucleoside Di- and Triphosphates and Dinucleoside Polyphosphates withcycloSal-Nucleotides

(2009) Svenja Warnecke et al.   JOURNAL OF ORGANIC CHEMISTRY

A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions

(2009) Marco Radi et al.   NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS

Truncated Fluorocyclopentenyl Pyrimidines asS-Adenosylhomocysteine Hydrolase Inhibitors

(2009) Yeon Hee Park et al.   NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS

Radical-mediated stannylation of vinyl sulfones: access to novel 4′-modified neplanocin A analogues

(2009) Hiroki Kumamoto et al.   TETRAHEDRON