Design of inhibitors of BCRP/ABCG2

Characterization of 3-methoxy flavones for their interaction with ABCG2 as suggested by ATPase activity

(2014) Jennifer Gallus et al.   BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES

Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2)

(2013) Kapil Juvale et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and biological evaluation of flavones and benzoflavones as inhibitors of BCRP/ABCG2

(2013) Kapil Juvale et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Identification of Novel Breast Cancer Resistance Protein (BCRP) Inhibitors by Virtual Screening

(2013) Yongmei Pan et al.   MOLECULAR PHARMACEUTICS

Tyrosine Kinase Inhibitors Influence ABCG2 Expression in EGFR-Positive MDCK BCRP Cells via the PI3K/Akt Signaling Pathway

(2012) Anne Pick et al.   ChemMedChem

Investigation of Chalcones as Selective Inhibitors of the Breast Cancer Resistance Protein: Critical Role of Methoxylation in both Inhibition Potency and Cytotoxicity

(2012) Glaucio Valdameri et al.   JOURNAL OF MEDICINAL CHEMISTRY

Investigation of chalcones and benzochalcones as inhibitors of breast cancer resistance protein

(2011) Kapil Juvale et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The sulfated conjugate of biochanin A is a substrate of breast cancer resistant protein (ABCG2)

(2011) Guohua An et al.   BIOPHARMACEUTICS & DRUG DISPOSITION

Substituted Chromones as Highly Potent Nontoxic Inhibitors, Specific for the Breast Cancer Resistance Protein

(2011) Glaucio Valdameri et al.   JOURNAL OF MEDICINAL CHEMISTRY

Breast cancer resistance protein (BCRP/ABCG2): its role in multidrug resistance and regulation of its gene expression

(2011) Takeo Nakanishi et al.   Chinese Journal of Cancer

Structure–activity relationships of flavonoids as inhibitors of breast cancer resistance protein (BCRP)

(2010) Anne Pick et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Restricted brain penetration of the tyrosine kinase inhibitor erlotinib due to the drug transporters P-gp and BCRP

(2010) Nienke A. de Vries et al.   INVESTIGATIONAL NEW DRUGS

Modulation of breast cancer resistance protein (BCRP/ABCG2) by non-basic chalcone analogues

(2008) Yi Han et al.   EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES

Functionalized chalcones as selective inhibitors of P-glycoprotein and breast cancer resistance protein

(2007) Xiao-Ling Liu et al.   BIOORGANIC & MEDICINAL CHEMISTRY