Structure-Activity Relationship Studies on (R )-PFI-2 Analogues as Inhibitors of Histone Lysine Methyltransferase SETD7
出版年份 2018 全文链接
标题
Structure-Activity Relationship Studies on (R
)-PFI-2 Analogues as Inhibitors of Histone Lysine Methyltransferase SETD7
作者
关键词
-
出版物
ChemMedChem
Volume 13, Issue 14, Pages 1405-1413
出版商
Wiley
发表日期
2018-06-05
DOI
10.1002/cmdc.201800242
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Inhibition of histone lysine methyltransferases G9a and GLP by ejection of structural Zn(II)
- (2018) Danny C. Lenstra et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Steric structure–activity relationship of cyproheptadine derivatives as inhibitors of histone methyltransferase Set7/9
- (2016) Takashi Fujiwara et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Identification of Cyproheptadine as an Inhibitor of SET Domain Containing Lysine Methyltransferase 7/9 (Set7/9) That Regulates Estrogen-Dependent Transcription
- (2016) Yasushi Takemoto et al. JOURNAL OF MEDICINAL CHEMISTRY
- Methylation by Set9 modulates FoxO3 stability and transcriptional activity
- (2016) Daniel R. Calnan et al. Aging-US
- Regulation of Transcription Factor Yin Yang 1 by SET7/9-mediated Lysine Methylation
- (2016) Wen-juan Zhang et al. Scientific Reports
- SET7/9 regulates cancer cell proliferation by influencing β-catenin stability
- (2015) Changchun Shen et al. FASEB JOURNAL
- Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening
- (2015) Fanwang Meng et al. JOURNAL OF MEDICINAL CHEMISTRY
- MicroRNA-153 functions as a tumor suppressor by targeting SET7 and ZEB2 in ovarian cancer cells
- (2015) JUN ZHOU et al. ONCOLOGY REPORTS
- Adverse Epigenetic Signatures by Histone Methyltransferase Set7 Contribute to Vascular Dysfunction in Patients With Type 2 Diabetes MellitusCLINICAL PERSPECTIVE
- (2014) Francesco Paneni et al. Circulation-Cardiovascular Genetics
- Selective Inhibitors of Protein Methyltransferases
- (2014) H. Ümit Kaniskan et al. JOURNAL OF MEDICINAL CHEMISTRY
- (R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells
- (2014) D. Barsyte-Lovejoy et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- SET7/9-dependent methylation of ARTD1 at K508 stimulates poly-ADP-ribose formation after oxidative stress
- (2013) I. Kassner et al. Open Biology
- Histone methylation: a dynamic mark in health, disease and inheritance
- (2012) Eric L. Greer et al. NATURE REVIEWS GENETICS
- Regulation of chromatin by histone modifications
- (2011) Andrew J Bannister et al. CELL RESEARCH
- Regulation of the androgen receptor by SET9-mediated methylation
- (2010) Luke Gaughan et al. NUCLEIC ACIDS RESEARCH
- Regulation of DNMT1 stability through SET7-mediated lysine methylation in mammalian cells
- (2009) P.-O. Esteve et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Role of histone modifications in defining chromatin structure and function
- (2008) Kathy A. Gelato et al. BIOLOGICAL CHEMISTRY
- Regulation of Estrogen Receptor α by the SET7 Lysine Methyltransferase
- (2008) Krithika Subramanian et al. MOLECULAR CELL
- Methylation of p53 by Set7/9 Mediates p53 Acetylation and Activity In Vivo
- (2008) Julia K. Kurash et al. MOLECULAR CELL
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