Exploring the structural requirements in multiple chemical scaffolds for the selective inhibition of Plasmodium falciparum calcium-dependent protein kinase-1 (PfCDPK-1) by 3D-pharmacophore modelling, and docking studies

In silico Modeling of Antimalarial Protein Kinase Inhibitors

(2015) Rahul Balasaheb Aher et al.   Letters in Drug Design & Discovery

Development of potent and selective Plasmodium falciparum calcium-dependent protein kinase 4 (PfCDPK4) inhibitors that block the transmission of malaria to mosquitoes

(2014) Rama Subba Rao Vidadala et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Optimization of an Imidazopyridazine Series of Inhibitors of Plasmodium falciparum Calcium-Dependent Protein Kinase 1 (PfCDPK1)

(2014) Timothy M. Chapman et al.   JOURNAL OF MEDICINAL CHEMISTRY

Substituted imidazopyridazines are potent and selective inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1)

(2013) Timothy M. Chapman et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Imidazopyridazines as potent inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1): Preparation and evaluation of pyrazole linked analogues

(2013) Jonathan M. Large et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

3,6-Diamino-4-(2-halophenyl)-2-benzoylthieno[2,3-b]pyridine-5-carbonitriles Are Selective Inhibitors of Plasmodium falciparum Glycogen Synthase Kinase-3

(2012) Wiebke Fugel et al.   JOURNAL OF MEDICINAL CHEMISTRY

Selective inhibition of Pfmrk, a Plasmodium falciparum CDK, by antimalarial 1,3-diaryl-2-propenones

(2009) Jeanne A. Geyer et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis of 3-(1,2,3-triazol-1-yl)- and 3-(1,2,3-triazol-4-yl)-substituted pyrazolo[3,4-d]pyrimidin-4-amines via click chemistry: potential inhibitors of the Plasmodium falciparum PfPK7 protein kinase

(2009) Michael Klein et al.   ORGANIC & BIOMOLECULAR CHEMISTRY