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Luminescent Lanthanide Cryptates: from the Bench to the Bedside

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Selective Actions of Novel Allosteric Modulators Reveal Functional Heteromers of Metabotropic Glutamate Receptors in the CNS

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(2014) Li Xue et al.   Nature Chemical Biology

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The Druggable Genome: Evaluation of Drug Targets in Clinical Trials Suggests Major Shifts in Molecular Class and Indication

(2013) Mathias Rask-Andersen et al.   Annual Review of Pharmacology and Toxicology

Inhibition of Tumor Angiogenesis and Growth by a Small-Molecule Multi-FGF Receptor Blocker with Allosteric Properties

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Small-molecule modulation of neurotrophin receptors: a strategy for the treatment of neurological disease

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Illuminating the activation mechanisms and allosteric properties of metabotropic glutamate receptors

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A Fluorescent Sensor for GABA and Synthetic GABAB Receptor Ligands

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Semisynthesis of Fluorescent Metabolite Sensors on Cell Surfaces

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(2011) Søren G. F. Rasmussen et al.   NATURE

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(2011) Christy F Landes et al.   Nature Chemical Biology

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A new approach to analyze cell surface protein complexes reveals specific heterodimeric metabotropic glutamate receptors

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Spatial control of EGF receptor activation by reversible dimerization on living cells

(2010) Inhee Chung et al.   NATURE

Crosstalk between GABAB and mGlu1a receptors reveals new insight into GPCR signal integration

(2009) Marie-Laure Rives et al.   EMBO JOURNAL

BRET3: a red-shifted bioluminescence resonance energy transfer (BRET)-based integrated platform for imaging protein-protein interactions from single live cells and living animals

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An Engineered Protein Tag for Multiprotein Labeling in Living Cells

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Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to GPCR oligomerization

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Structural diversity of G protein-coupled receptors and significance for drug discovery

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