期刊
JOURNAL OF ORGANIC CHEMISTRY
卷 82, 期 12, 页码 6366-6372出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.joc.7b00948
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资金
- UGC-New Delhi
- CSIR-New Delhi
- DST-SERB
- CSIR-ORIGIN, New Delhi
The Pd-catalyzed quinazolinone-directed regioselective monoarylation of aromatic rings by C-H bond activation is developed. A broad substrate scope is demonstrated for both quinazolinone as well as diary-liodonium triflates. The use of a base was found to be crucial for this transformation, unlike for the known nitrogen-directed arylations. All of the novel quinazolinones of biological interest were synthesized by using the operationally simple Pd(II)-catalyzed arylation reaction.
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