Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs

标题
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs
作者
关键词
-
出版物
JOURNAL OF MEDICINAL CHEMISTRY
Volume 60, Issue 10, Pages 4304-4315
出版商
American Chemical Society (ACS)
发表日期
2017-05-11
DOI
10.1021/acs.jmedchem.7b00247

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