标题
Structural basis for subtype-specific inhibition of the P2X7 receptor
作者
关键词
-
出版物
eLife
Volume 5, Issue -, Pages -
出版商
eLife Sciences Organisation, Ltd.
发表日期
2016-12-09
DOI
10.7554/elife.22153
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- The microglial ATP-gated ion channel P2X7 as a CNS drug target
- (2016) Anindya Bhattacharya et al. GLIA
- X-ray structures define human P2X3 receptor gating cycle and antagonist action
- (2016) Steven E. Mansoor et al. NATURE
- Molecular structure and function of P2X receptors
- (2016) Chloé Habermacher et al. NEUROPHARMACOLOGY
- P2X7 receptor: an emerging target in central nervous system diseases
- (2014) Beáta Sperlágh et al. TRENDS IN PHARMACOLOGICAL SCIENCES
- How good are my data and what is the resolution?
- (2013) Philip R. Evans et al. ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY
- Pharmacological characterization of a novel centrally permeable P2X7 receptor antagonist: JNJ-47965567
- (2013) Anindya Bhattacharya et al. BRITISH JOURNAL OF PHARMACOLOGY
- Purinergic mechanisms and pain—An update
- (2013) Geoffrey Burnstock EUROPEAN JOURNAL OF PHARMACOLOGY
- Purinergic signalling: from discovery to current developments
- (2013) Geoffrey Burnstock EXPERIMENTAL PHYSIOLOGY
- Clinical evaluation of the efficacy of the P2X7purinergic receptor antagonist AZD9056 on the signs and symptoms of rheumatoid arthritis in patients with active disease despite treatment with methotrexate or sulphasalazine
- (2012) Edward C Keystone et al. ANNALS OF THE RHEUMATIC DISEASES
- Efficacy and Safety of CE-224,535, an Antagonist of P2X7 Receptor, in Treatment of Patients with Rheumatoid Arthritis Inadequately Controlled by Methotrexate
- (2012) T. C. STOCK et al. JOURNAL OF RHEUMATOLOGY
- Molecular mechanism of ATP binding and ion channel activation in P2X receptors
- (2012) Motoyuki Hattori et al. NATURE
- Overview of theCCP4 suite and current developments
- (2011) Martyn D. Winn et al. ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY
- Modern methods for delivery of drugs across the blood–brain barrier
- (2011) Yan Chen et al. ADVANCED DRUG DELIVERY REVIEWS
- Pain as a global public health priority
- (2011) Daniel S Goldberg et al. BMC PUBLIC HEALTH
- P2X receptor antagonists for pain management: examination of binding and physicochemical properties
- (2011) Rebecca J. Gum et al. Purinergic Signalling
- XDS
- (2010) Wolfgang Kabsch ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY
- PHENIX: a comprehensive Python-based system for macromolecular structure solution
- (2010) Paul D. Adams et al. ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY
- Experimental Characterization and Mathematical Modeling of P2X7 Receptor Channel Gating
- (2010) Z. Yan et al. JOURNAL OF NEUROSCIENCE
- Nociceptor sensitization in pain pathogenesis
- (2010) Michael S Gold et al. NATURE MEDICINE
- The evidence for pharmacological treatment of neuropathic pain
- (2010) Nanna Brix Finnerup et al. PAIN
- Crystal structure of the ATP-gated P2X4 ion channel in the closed state
- (2009) Toshimitsu Kawate et al. NATURE
- Identification of regions of the P2X7 receptor that contribute to human and rat species differences in antagonist effects
- (2008) A D Michel et al. BRITISH JOURNAL OF PHARMACOLOGY
- The P2X7Receptor Channel Pore Dilates under Physiological Ion Conditions
- (2008) Zonghe Yan et al. JOURNAL OF GENERAL PHYSIOLOGY
- [3H]A-804598 ([3H]2-cyano-1-[(1S)-1-phenylethyl]-3-quinolin-5-ylguanidine) is a novel, potent, and selective antagonist radioligand for P2X7 receptors
- (2008) Diana L. Donnelly-Roberts et al. NEUROPHARMACOLOGY
- HOLLOW: Generating Accurate Representations of Channel and Interior Surfaces in Molecular Structures
- (2008) Bosco K Ho et al. BMC STRUCTURAL BIOLOGY
- Negative and positive allosteric modulators of the P2X7receptor
- (2007) A D Michel et al. BRITISH JOURNAL OF PHARMACOLOGY
- Taking The Time To Study Competitive Antagonism
- (2007) D J A Wyllie et al. BRITISH JOURNAL OF PHARMACOLOGY
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