In vitro expression and analysis of the 826 human G protein-coupled receptors

Mammalian odorant receptors: functional evolution and variation

(2015) Yue Jiang et al.   CURRENT OPINION IN NEUROBIOLOGY

Role of post-translational modifications on structure, function and pharmacology of class C G protein-coupled receptors

(2015) Lenea Nørskov-Lauritsen et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

N-glycosylation and disulfide bonding affects GPRC6A receptor expression, function, and dimerization

(2015) Lenea Nørskov-Lauritsen et al.   FEBS LETTERS

G protein-coupled odorant receptors: From sequence to structure

(2015) Claire A. de March et al.   PROTEIN SCIENCE

Generic GPCR residue numbers – aligning topology maps while minding the gaps

(2015) Vignir Isberg et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Agonist-bound structure of the human P2Y12 receptor

(2014) Jin Zhang et al.   NATURE

Molecular control of δ-opioid receptor signalling

(2014) Gustavo Fenalti et al.   NATURE

Promotion of Cancer Cell Invasiveness and Metastasis Emergence Caused by Olfactory Receptor Stimulation

(2014) Guenhaël Sanz et al.   PLoS One

The Druggable Genome: Evaluation of Drug Targets in Clinical Trials Suggests Major Shifts in Molecular Class and Indication

(2013) Mathias Rask-Andersen et al.   Annual Review of Pharmacology and Toxicology

Structure of the human glucagon class B G-protein-coupled receptor

(2013) Fai Yiu Siu et al.   NATURE

Structural Features for Functional Selectivity at Serotonin Receptors

(2013) D. Wacker et al.   SCIENCE

Ice breaking in GPCR structural biology

(2012) Qiang Zhao et al.   ACTA PHARMACOLOGICA SINICA

Structure-Function of the G Protein–Coupled Receptor Superfamily

(2012) Vsevolod Katritch et al.   Annual Review of Pharmacology and Toxicology

The GPCR Network: a large-scale collaboration to determine human GPCR structure and function

(2012) Raymond C. Stevens et al.   NATURE REVIEWS DRUG DISCOVERY

Crystal Structure of a Lipid G Protein-Coupled Receptor

(2012) M. A. Hanson et al.   SCIENCE

Structural Basis for Allosteric Regulation of GPCRs by Sodium Ions

(2012) W. Liu et al.   SCIENCE

Fusion Partner Toolchest for the Stabilization and Crystallization of G Protein-Coupled Receptors

(2012) Eugene Chun et al.   STRUCTURE

Diversity and modularity of G protein-coupled receptor structures

(2011) Vsevolod Katritch et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Structures of the CXCR4 Chemokine GPCR with Small-Molecule and Cyclic Peptide Antagonists

(2010) B. Wu et al.   SCIENCE