Design, synthesis and biological evaluation of fluorescent ligands for MT1 and/or MT2 melatonin receptors

Synthesis of 2-arylfuro[3,2-b]pyridines: Effect of the C2-aryl group on melatoninergic activity

(2016) Audrey Couhert et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

New coumarin-based fluorescent melatonin ligands. Design, synthesis and pharmacological characterization

(2015) Mario de la Fuente Revenga et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II)

(2015) Mohamed Ettaoussi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Novel N-Acetyl Bioisosteres of Melatonin: Melatonergic Receptor Pharmacology, Physicochemical Studies, and Phenotypic Assessment of Their Neurogenic Potential

(2015) Mario de la Fuente Revenga et al.   JOURNAL OF MEDICINAL CHEMISTRY

Melatonin: Physiological effects in humans

(2015) B. Claustrat et al.   NEUROCHIRURGIE

New melatonin (MT1/MT2) ligands: Design and synthesis of (8,9-dihydro-7H-furo[3,2-f]chromen-1-yl) derivatives

(2014) Elodie Landagaray et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Extending the Scope of the Aza-Fischer Synthesis of 4- and 6-Azaindoles

(2013) David Thomae et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

New Radioligands for Describing the Molecular Pharmacology of MT1 and MT2 Melatonin Receptors

(2013) Céline Legros et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

MT1 and MT2 Melatonin Receptors: Ligands, Models, Oligomers, and Therapeutic Potential

(2013) Darius. P. Zlotos et al.   JOURNAL OF MEDICINAL CHEMISTRY

Original Design of Fluorescent Ligands by Fusing BODIPY and Melatonin Neurohormone

(2013) Jérémy Thireau et al.   ACS Medicinal Chemistry Letters

N-Acetyl-5-arylalkoxytryptamine Analogs: Probing the Melatonin Receptors for MT1-Selectivity

(2011) Christian Markl et al.   ARCHIV DER PHARMAZIE

Design and synthesis of 1-(2-alkanamidoethyl)-6-methoxy-7-azaindole derivatives as potent melatonin agonists

(2011) Matthieu Jeanty et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Preparation and pharmacological evaluation of a novel series of 2-(phenylthio)benzo[b]thiophenes as selective MT2 receptor ligands

(2011) Christophe Mésangeau et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design and synthesis of 2-phenylimidazo[1,2-a]pyridines as a novel class of melatonin receptor ligands

(2011) Saïd El Kazzouli et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

1,6-Dihydro-2H-indeno[5,4-b]furan Derivatives: Design, Synthesis, and Pharmacological Characterization of a Novel Class of Highly Potent MT2-Selective Agonists

(2011) Tatsuki Koike et al.   JOURNAL OF MEDICINAL CHEMISTRY

2-[(1,3-Dihydro-2H-isoindol-2-yl)methyl]melatonin – a novel MT2-selective melatonin receptor antagonist

(2011) David Heckman et al.   MedChemComm

Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT1 melatoninergic ligands

(2010) Christophe Mésangeau et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Antiinflammatory Activity of Melatonin in Central Nervous System

(2010) Emanuela Esposito et al.   Current Neuropharmacology

Erratum: Agomelatine, the first melatonergic antidepressant: discovery, characterization and development

(2010) Christian de Bodinat et al.   NATURE REVIEWS DRUG DISCOVERY

Melatonin—A pleiotropic, orchestrating regulator molecule

(2010) Rüdiger Hardeland et al.   PROGRESS IN NEUROBIOLOGY

2-[(2,3-Dihydro-1H-indol-1-yl)methyl]melatonin Analogues: A Novel Class of MT2-Selective Melatonin Receptor Antagonists

(2009) Darius P. Zlotos et al.   JOURNAL OF MEDICINAL CHEMISTRY

Melatonin: A hormone that modulates pain

(2009) Mónica Ambriz-Tututi et al.   LIFE SCIENCES

Synthesis of 4- and 6-Azaindoles via the Fischer Reaction

(2009) Matthieu Jeanty et al.   ORGANIC LETTERS

Fluorescent GPCR Ligands as New Tools in Pharmacology

(2008) Kamil Kuder et al.   CURRENT MEDICINAL CHEMISTRY

Melatonin Receptor Agonists: SAR and Applications to the Treatment of Sleep-Wake Disorders

(2008) Silvia Rivara et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Melatonin, sleep disturbance and cancer risk

(2008) David E. Blask   SLEEP MEDICINE REVIEWS

The Chemistry of Fluorescent Bodipy Dyes: Versatility Unsurpassed

(2007) Gilles Ulrich et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION