期刊
ORGANIC LETTERS
卷 18, 期 7, 页码 1554-1557出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.6b00356
关键词
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资金
- NIH [GM63188]
- NSF [GOALI-1012883]
- Merck
- ACS/GCI Pharmaceutical Roundtable
- Thomas J. Pinnavaia Fellowship
Bismuth(III) acetate is a safe, inexpensive, and selective facilitator of sequential protodeboronations, which when used in conjunction with Ir-catalyzed borylations allows access to a diversity of borylated indoles. The versatility of combining Ir-catalyzed borylations with Bi(III)-catalyzed protodeboronation is demonstrated by selectively converting 6-fluoroindole into products with Bpin groups at the 4-, 5-, 7-, 2,7-, 4,7-, 3,5-, and 2,4,7-positions and the late-stage functionalization of sumatriptan.
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