Metal-mediated post-Ugi transformations for the construction of diverse heterocyclic scaffolds

Diversely Substituted Indoloazepinones and Indoloazocinones: A Post-Ugi Gold-Catalyzed Regioselective Carbocyclization Approach

(2015) Sachin Modha et al.   SYNTHESIS-STUTTGART

Isocyanide-based multicomponent reactions towards cyclic constrained peptidomimetics

(2014) Gijs Koopmanschap et al.   Beilstein Journal of Organic Chemistry

Regioselective Synthesis of Diversely Substituted Diazoninones Through a Post-Ugi Gold-Catalyzed Intramolecular Hydroarylation Process

(2014) Zhenghua Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Facile Access to Functionalized Spiro[indoline-3,2′-pyrrole]-2,5′-diones via Post-Ugi Domino Buchwald–Hartwig/Michael Reaction

(2014) Nandini Sharma et al.   ORGANIC LETTERS

Microwave-assisted synthesis of 4H-benzo[f]imidazo[1,4]diazepin-6-ones via a post-Ugi copper-catalyzed intramolecular Ullmann coupling

(2014) Zhenghua Li et al.   TETRAHEDRON LETTERS

Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines

(2013) Amit Kumar et al.   Beilstein Journal of Organic Chemistry

Rapid and selective access to three distinct sets of indole-based heterocycles from a single set of Ugi-adducts under microwave heating

(2013) Lei Zhang et al.   CHEMICAL COMMUNICATIONS

Switching the regioselectivity via indium(iii) and gold(i) catalysis: a post-Ugi intramolecular hydroarylation to azepino- and azocino-[c,d]indolones

(2013) Amit Kumar et al.   CHEMICAL COMMUNICATIONS

Synthesis of (spiro)cyclopentapyridinones via Csp3–H functionalization: a post-Ugi gold-catalyzed regioselective tandem cyclization

(2013) Dipak D. Vachhani et al.   CHEMICAL COMMUNICATIONS

Diversely Substituted Triazolo[1,5-a][1,4]benzodiazepinones: A Post-Ugi Copper-Catalyzed Tandem Azide-Alkyne Cycloaddition/Ullmann C-N Coupling Approach

(2013) Dipak D. Vachhani et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Selective Synthesis of 5,6-Dihydroindolo[1,2-a]quinoxalines and 6,7-Dihydroindolo[2,3-c]quinolines by Orthogonal Copper and Palladium Catalysis

(2013) Lei Zhang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Gold(I)-Catalyzed Post-Ugi Hydroarylation: An Approach to Pyrrolopyridines and Azepinoindoles

(2013) Amit Kumar et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

An Expedient Route to Imidazo[1,4]diazepin-7-ones via A Post-Ugi Gold-Catalyzed Heteroannulation

(2013) Amit Kumar et al.   ORGANIC LETTERS

Ligand-free palladium-catalyzed intramolecular arylation of chromones: an expedient synthesis of 1-benzopyrano[3,2-c]quinolines

(2013) Jaydip Ghosh et al.   TETRAHEDRON LETTERS

A Diversity-Oriented Approach to Spiroindolines: Post-Ugi Gold-Catalyzed Diastereoselective Domino Cyclization

(2012) Sachin G. Modha et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A concise route to indoloazocines via a sequential Ugi–gold-catalyzed intramolecular hydroarylation

(2012) Sachin G. Modha et al.   CHEMICAL COMMUNICATIONS

Gold(i) and platinum(ii) switch: a post-Ugi intramolecular hydroarylation to pyrrolopyridinones and pyrroloazepinones

(2012) Sachin G. Modha et al.   CHEMICAL COMMUNICATIONS

A Ligand-Free Pd-Catalyzed Cascade Reaction: An Access to the Highly Diverse Isoquinolin-1(2H)-one Derivatives via Isocyanide and Ugi-MCR Synthesized Amide Precursors

(2012) Vikas Tyagi et al.   ORGANIC LETTERS

Ugi post-condensation copper-triggered oxidative cascade towards pyrazoles

(2011) Aurélie Dos Santos et al.   Beilstein Journal of Organic Chemistry

Straightforward four-component access to spiroindolines

(2011) Laurent El Kaïm et al.   CHEMICAL COMMUNICATIONS

Palladium-catalyzed stereoselective synthesis of 3-(aminomethylene)-oxindoles

(2011) Morteza Bararjanian et al.   TETRAHEDRON LETTERS

Six-Component Reactions for the Stereoselective Synthesis of 3-Arylidene-2-oxindoles via Sequential One-Pot Ugi/Heck Carbocyclization/Sonogashira/Nucleophilic Addition

(2010) Morteza Bararjanian et al.   JOURNAL OF ORGANIC CHEMISTRY

A Highly Convergent Synthesis of Tricyclic N-Heterocycles Coupling an Ugi Reaction with a Tandem SN2′-Heck Double Cyclization

(2010) Renata Riva et al.   JOURNAL OF ORGANIC CHEMISTRY

Ugi-Post Functionalization, from a Single Set of Ugi-Adducts to Two Distinct Heterocycles by Microwave-Assisted Palladium-Catalyzed Cyclizations: Tuning the Reaction Pathways by Ligand Switch

(2009) William Erb et al.   JOURNAL OF ORGANIC CHEMISTRY

Emerging molecular diversity from the intra-molecular Ugi reaction: iterative efficiency in medicinal chemistry

(2009) Christopher Hulme et al.   MOLECULAR DIVERSITY

Palladium-Catalyzed IntramolecularC-Arylation of Benzylic Carbon: Synthesis of 3-Benzoxazolylisoindolinones by a Sequence of Ugi-4CR/Postfunctionalization

(2008) Angela Salcedo et al.   JOURNAL OF ORGANIC CHEMISTRY

Polyfunctionalized Pyrrolidines by Ugi Multicomponent Reaction Followed by Palladium-Mediated SN2‘ Cyclizations

(2008) Luca Banfi et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Domino Intramolecular N-Arylation/Intermolecular C−C Bond Formation for the Synthesis of Functionalized Benzodiazepinediones

(2008) Angela Salcedo et al.   ORGANIC LETTERS

A Tandem One-Pot, Microwave-Assisted Synthesis of Regiochemically Differentiated 1,2,4,5-Tetrahydro-1,4-benzodiazepin-3-ones

(2008) Ravindra A. De Silva et al.   ORGANIC LETTERS

Synthesis of 3-Arylideneindolin-2-ones from 2-Aminophenols by Ugi Four-Component Reaction and Heck Carbocyclization

(2008) Wei-Min Dai et al.   SYNLETT