Synthesis of Cyclopropylamines through an Electro-Induced Hofmann Rearrangement

Synthesis of 1- and 1,2-Substituted Cyclopropylamines from Ketone Homoenolates

(2022) Michael S. West et al.   ORGANIC LETTERS

Synthesis of 1-Substituted Cyclopropylamines via Formal Tertiary Csp3–H Amination of Cyclopropanes

(2021) Kui Liu et al.   ORGANIC LETTERS

Selective Carbon–Carbon Bond Cleavage of Cyclopropylamine Derivatives

(2020) Olga O. Sokolova et al.   CHEMICAL REVIEWS

Rhodium(III)-Catalyzed Cyclopropane C–H/C–C Activation Sequence Provides Diastereoselective Access to α-Alkoxylated γ-Lactams

(2020) Benoit Audic et al.   ORGANIC LETTERS

Discovery of a Hepatitis C Virus NS5B Replicase Palm Site Allosteric Inhibitor (BMS-929075) Advanced to Phase 1 Clinical Studies

(2017) Kap-Sun Yeung et al.   JOURNAL OF MEDICINAL CHEMISTRY

The “Cyclopropyl Fragment” is a Versatile Player that Frequently Appears in Preclinical/Clinical Drug Molecules

(2016) Tanaji T. Talele   JOURNAL OF MEDICINAL CHEMISTRY

Transition-Metal-Free Synthesis of Tertiary Aminocyclopropanes

(2016) Patrick Cyr et al.   ORGANIC LETTERS

Transition-Metal-Free Cyclopropanation of 2-Aminoacrylates with N-Tosylhydrazones: A General Route to Cyclopropane α-Amino Acid with Contiguous Quaternary Carbon Centers

(2016) Chuanle Zhu et al.   ORGANIC LETTERS

Critical Intermediates Reveal New Biosynthetic Events in the Enigmatic Colibactin Pathway

(2015) Zhong-Rui Li et al.   CHEMBIOCHEM

Palladium(II)-Catalyzed Intramolecular Tandem Aminoalkylation via Divergent C(sp3)–H Functionalization

(2015) Wei Du et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Stereoselective Synthesis of (Borylmethyl)cyclopropylamines by Copper-Catalyzed Aminoboration of Methylenecyclopropanes

(2014) Ryosuke Sakae et al.   ORGANIC LETTERS

Experimental Evidence for the All-Up Reactive Conformation of Chiral Rhodium(II) Carboxylate Catalysts: Enantioselective Synthesis ofcis-Cyclopropane α-Amino Acids

(2009) Vincent N. G. Lindsay et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY