Data-Driven Global Assessment of Protein Kinase Inhibitors with Emphasis on Covalent Compounds
出版年份 2023 全文链接
标题
Data-Driven Global Assessment of Protein Kinase Inhibitors with Emphasis on Covalent Compounds
作者
关键词
-
出版物
Journal of Medicinal Chemistry
Volume 66, Issue 11, Pages 7657-7665
出版商
American Chemical Society (ACS)
发表日期
2023-05-22
DOI
10.1021/acs.jmedchem.3c00621
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- From traditional to data-driven medicinal chemistry: A case study
- (2022) Ryo Kunimoto et al. DRUG DISCOVERY TODAY
- Advances in covalent drug discovery
- (2022) Lydia Boike et al. NATURE REVIEWS DRUG DISCOVERY
- Systematic Exploration of Privileged Warheads for Covalent Kinase Drug Discovery
- (2022) Zheng Zhao et al. Pharmaceuticals
- UniProt: the Universal Protein Knowledgebase in 2023
- (2022) et al. NUCLEIC ACIDS RESEARCH
- Reactivity of Covalent Fragments and Their Role in Fragment Based Drug Discovery
- (2022) Kirsten McAulay et al. Pharmaceuticals
- Structure- and Similarity-Based Survey of Allosteric Kinase Inhibitors, Activators, and Closely Related Compounds
- (2021) Oliver Laufkötter et al. JOURNAL OF MEDICINAL CHEMISTRY
- Recent advances in development of hetero-bivalent kinase inhibitors
- (2021) Seungbeom Lee et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Kinase drug discovery 20 years after imatinib: progress and future directions
- (2021) Philip Cohen et al. NATURE REVIEWS DRUG DISCOVERY
- Trends in kinase drug discovery: targets, indications and inhibitor design
- (2021) Misty M. Attwood et al. NATURE REVIEWS DRUG DISCOVERY
- Small Molecule Kinase Inhibitor Drugs (1995–2021): Medical Indication, Pharmacology, and Synthesis
- (2021) Cecilia C. Ayala-Aguilera et al. JOURNAL OF MEDICINAL CHEMISTRY
- Kinase inhibition in autoimmunity and inflammation
- (2020) Ali A. Zarrin et al. NATURE REVIEWS DRUG DISCOVERY
- CovalentInDB: a comprehensive database facilitating the discovery of covalent inhibitors
- (2020) Hongyan Du et al. NUCLEIC ACIDS RESEARCH
- Evolving Concept of Activity Cliffs
- (2019) Dagmar Stumpfe et al. ACS Omega
- New Promise and Opportunities for Allosteric Kinase Inhibitors
- (2019) Xiaoyun Lu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- The Cysteinome of Protein Kinases as a Target in Drug Development
- (2018) Apirat Chaikuad et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Redundancy in two major compound databases
- (2018) Dimitar Yonchev et al. DRUG DISCOVERY TODAY
- Kinase inhibitors: the road ahead
- (2018) Fleur M. Ferguson et al. NATURE REVIEWS DRUG DISCOVERY
- Emerging and Re-Emerging Warheads for Targeted Covalent Inhibitors: Applications in Medicinal Chemistry and Chemical Biology
- (2018) Matthias Gehringer et al. JOURNAL OF MEDICINAL CHEMISTRY
- The role of hypoxia-inducible factors in metabolic diseases
- (2018) Frank J. Gonzalez et al. Nature Reviews Endocrinology
- Determining Cysteines Available for Covalent Inhibition Across the Human Kinome
- (2017) Zheng Zhao et al. JOURNAL OF MEDICINAL CHEMISTRY
- Covalent-Allosteric Kinase Inhibitors
- (2015) Jörn Weisner et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- The ins and outs of selective kinase inhibitor development
- (2015) Susanne Müller et al. Nature Chemical Biology
- Bivalent inhibitors of protein kinases
- (2014) Carrie M. Gower et al. CRITICAL REVIEWS IN BIOCHEMISTRY AND MOLECULAR BIOLOGY
- Current Compound Coverage of the Kinome
- (2014) Ye Hu et al. JOURNAL OF MEDICINAL CHEMISTRY
- Approaches to discover non-ATP site kinase inhibitors
- (2012) Lori Krim Gavrin et al. MedChemComm
- ChEMBL: a large-scale bioactivity database for drug discovery
- (2011) A. Gaulton et al. NUCLEIC ACIDS RESEARCH
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