Screening the binding affinity of bile acid derivatives for the glucocorticoid receptor ligand-binding domain

Synthesis of new bile acid-fused tetrazoles using the Schmidt reaction

(2021) Dušan Đ Škorić et al.   Beilstein Journal of Organic Chemistry

Physicochemical characterization of novel 3-carboxymethyl-bile salts, as permeability and solubility enhancers

(2020) Mihalj Poša et al.   JOURNAL OF MOLECULAR LIQUIDS

Dexamethasone in Hospitalized Patients with Covid-19 — Preliminary Report

(2020)   NEW ENGLAND JOURNAL OF MEDICINE

The VEGA suite of programs: an versatile platform for cheminformatics and drug design projects

(2020) Alessandro Pedretti et al.   BIOINFORMATICS

Hydrophobicity and self‐association (micellization) of bile salts with a lactone or lactam group in a steroid skeleton

(2020) Mihalj Poša et al.   JOURNAL OF PHYSICAL ORGANIC CHEMISTRY

GR Dimerization and the Impact of GR Dimerization on GR Protein Stability and Half-Life

(2019) Ann Louw   Frontiers in Immunology

Taurochenodeoxycholic Acid Inhibited AP-1 Activation via Stimulating Glucocorticoid Receptor

(2019) Lei Li et al.   MOLECULES

Identification of d -seco modified steroid derivatives with affinity for estrogen receptor α and β isoforms using a non-transcriptional fluorescent cell assay in yeast

(2018) Sofija S. Bekić et al.   STEROIDS

Therapeutic Mechanisms of Glucocorticoids

(2018) Jolien Vandewalle et al.   TRENDS IN ENDOCRINOLOGY AND METABOLISM

A screening assay for Selective Dimerizing Glucocorticoid Receptor Agonists and Modulators (SEDIGRAM) that are effective against acute inflammation

(2018) Jolien Souffriau et al.   Scientific Reports

Synthesis of Five Known Brassinosteroid Analogs from Hyodeoxycholic Acid and Their Activities as Plant-Growth Regulators

(2017) María Duran et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Synthesis of B- and C-ring-modified lithocholic acid analogues as potential sialyltransferase inhibitors

(2016) Hajjaj H.M. Abdu-Allah et al.   STEROIDS

Tissue-specific actions of FXR in metabolism and cancer

(2015) Raffaella Maria Gadaleta et al.   BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS

Selective glucocorticoid receptor modulation: New directions with non-steroidal scaffolds

(2015) Nora Sundahl et al.   PHARMACOLOGY & THERAPEUTICS

TGR5 and Immunometabolism: Insights from Physiology and Pharmacology

(2015) Alessia Perino et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Glucocorticoid receptor-dependent immunomodulatory effect of ursodeoxycholic acid on liver lymphocytes in mice

(2013) Toshimichi Takigawa et al.   AMERICAN JOURNAL OF PHYSIOLOGY-GASTROINTESTINAL AND LIVER PHYSIOLOGY

11β-Hydroxysteroid dehydrogenase type 1 contributes to the balance between 7-keto- and 7-hydroxy-oxysterols in vivo

(2013) Tijana Mitić et al.   BIOCHEMICAL PHARMACOLOGY

Diabetes Mellitus and Inflammation

(2013) Eric Lontchi-Yimagou et al.   Current Diabetes Reports

Synthesis and antiproliferative activity of C-homo-lactam derivatives of 7-deoxycholic acid

(2012) Yanmin Huang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A Role of the Bile Salt Receptor FXR in Atherosclerosis

(2010) Jurre Hageman et al.   ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY

AutoDock4 and AutoDockTools4: Automated docking with selective receptor flexibility

(2009) Garrett M. Morris et al.   JOURNAL OF COMPUTATIONAL CHEMISTRY