Discovery, optimization and evaluation of 1-(indolin-1-yl)ethan-1-ones as novel selective TRIM24/BRPF1 bromodomain inhibitors
出版年份 2022 全文链接
标题
Discovery, optimization and evaluation of 1-(indolin-1-yl)ethan-1-ones as novel selective TRIM24/BRPF1 bromodomain inhibitors
作者
关键词
TRIM24, BRPF1, Bromodomain, Dual targeting inhibitor, Structure-guided design
出版物
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Volume 236, Issue -, Pages 114311
出版商
Elsevier BV
发表日期
2022-03-28
DOI
10.1016/j.ejmech.2022.114311
参考文献
相关参考文献
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