Synthesis and biological activity of novel 4-aminoquinoline/1,2,3-triazole hybrids against Leishmania amazonensis
出版年份 2021 全文链接
标题
Synthesis and biological activity of novel 4-aminoquinoline/1,2,3-triazole hybrids against Leishmania amazonensis
作者
关键词
Leishmania, Antileishmanial activity, Quinoline, 1,2,3-triazolic derivative, Apoptosis, Necrosis
出版物
BIOMEDICINE & PHARMACOTHERAPY
Volume 141, Issue -, Pages 111857
出版商
Elsevier BV
发表日期
2021-07-14
DOI
10.1016/j.biopha.2021.111857
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- The ultimate fate determinants of drug induced cell-death mechanisms in trypanosomatids
- (2021) Payel Das et al. International Journal for Parasitology-Drugs and Drug Resistance
- Synthesis and Biological Evaluation of New 1,2,3‐Triazolyl‐Pyrazolyl‐Quinoline Derivatives as Potential Antimicrobial Agents
- (2020) Prashant P. Thakare et al. ChemistrySelect
- Differential lethal action of C17:2 and C17:0 anacardic acid derivatives in Trypanosoma cruzi – A mechanistic study
- (2020) Eric Umehara et al. BIOORGANIC CHEMISTRY
- Cell death pathways in pathogenic trypanosomatids: lessons of (over)kill
- (2019) Rubem Figueiredo Sadok Menna-Barreto Cell Death & Disease
- Comprehensive review on the anti-bacterial activity of 1,2,3-triazole hybrids
- (2019) Bo Zhang EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Insights into the current status of privileged N-heterocycles as antileishmanial agents
- (2019) Nima Razzaghi-Asl et al. MOLECULAR DIVERSITY
- A semi-synthetic neolignan derivative from dihydrodieugenol B selectively affects the bioenergetic system of Leishmania infantum and inhibits cell division
- (2019) Maiara Amaral et al. Scientific Reports
- Activity and Cell-Death Pathway in Leishmania infantum Induced by Sugiol: Vectorization Using Yeast Cell Wall Particles Obtained From Saccharomyces cerevisiae
- (2019) Débora Botura Scariot et al. Frontiers in Cellular and Infection Microbiology
- 1,2,3-Triazole-containing hybrids as leads in medicinal chemistry: A recent overview
- (2019) Khurshed Bozorov et al. BIOORGANIC & MEDICINAL CHEMISTRY
- 4-Aminoquinoline-based compounds as antileishmanial agents that inhibit the energy metabolism of Leishmania
- (2019) José Ignacio Manzano et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Resveratrol analogues present effective antileishmanial activity against promastigotes and amastigotes from distinct Leishmania species by multitarget action in the parasites
- (2019) Luciana Maria Ribeiro Antinarelli et al. JOURNAL OF PHARMACY AND PHARMACOLOGY
- Novel functionalized 1,2,3-triazole derivatives exhibit antileishmanial activity, increase in total and mitochondrial-ROS and depolarization of mitochondrial membrane potential of Leishmania amazonensis
- (2019) Raíssa Soares Meinel et al. CHEMICO-BIOLOGICAL INTERACTIONS
- Multi-target drugs active against leishmaniasis: A paradigm of drug repurposing
- (2019) Susana Santos Braga EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis of cinnamic acid derivatives and leishmanicidal activity against Leishmania braziliensis
- (2019) Michelle Peixoto Rodrigues et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis, biological activity, and mechanism of action of new 2-pyrimidinyl hydrazone and N-acylhydrazone derivatives, a potent and new classes of antileishmanial agents
- (2019) Elaine Soares Coimbra et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- 1,2,3-Triazole-containing hybrids as potential anticancer agents: Current developments, action mechanisms and structure-activity relationships
- (2019) Zhi Xu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and evaluation of novel triazolyl quinoline derivatives as potential antileishmanial agents
- (2018) Akanksha Upadhyay et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and leishmanicidal activity of eugenol derivatives bearing 1,2,3-triazole functionalities
- (2018) Róbson Ricardo Teixeira et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Leishmaniasis
- (2018) Sakib Burza et al. LANCET
- Atypical leishmaniasis: A global perspective with emphasis on the Indian subcontinent
- (2018) Lovlesh Thakur et al. PLoS Neglected Tropical Diseases
- Quinoline and quinolone dimers and their biological activities: An overview
- (2018) Xue-Mei Chu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Antileishmanial activity of a 4-hydrazinoquinoline derivative: Induction of autophagy and apoptosis-related processes and effectiveness in experimental cutaneous leishmaniasis
- (2018) Luciana Maria Ribeiro Antinarelli et al. EXPERIMENTAL PARASITOLOGY
- A review on quinoline derived scaffolds as Anti-HIV Agents
- (2018) Nisha Chokkar et al. MINI-REVIEWS IN MEDICINAL CHEMISTRY
- 4-Aminoquinoline-ferrocenyl-chalcone conjugates: Synthesis and anti-plasmodial evaluation
- (2017) Amandeep Singh et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Quinoline hybrids and their antiplasmodial and antimalarial activities
- (2017) Yuan-Qiang Hu et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Comprehensive review on various strategies for antimalarial drug discovery
- (2017) Mitali Mishra et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- The photodynamic action of pheophorbide a induces cell death through oxidative stress in Leishmania amazonensis
- (2017) Nathielle Miranda et al. JOURNAL OF PHOTOCHEMISTRY AND PHOTOBIOLOGY B-BIOLOGY
- Chemotherapy of leishmaniasis: present challenges
- (2017) SILVIA R. B. ULIANA et al. PARASITOLOGY
- Induction of Early Autophagic Process on Leishmania amazonensis by Synergistic Effect of Miltefosine and Innovative Semi-synthetic Thiosemicarbazone
- (2017) Débora B. Scariot et al. Frontiers in Microbiology
- Effect of quinoline based 1,2,3-triazole and its structural analogues on growth and virulence attributes of Candida albicans
- (2017) Mohammad Irfan et al. PLoS One
- Zinc depletion promotes apoptosis-like death in drug-sensitive and antimony-resistance Leishmania donovani
- (2017) Shalini Saini et al. Scientific Reports
- Novel Triazole-Quinoline Derivatives as Selective Dual Binding Site Acetylcholinesterase Inhibitors
- (2016) Susimaire Mantoani et al. MOLECULES
- Dibenzylideneacetones Are Potent Trypanocidal Compounds That Affect the Trypanosoma cruzi Redox System
- (2015) Danielle Lazarin-Bidóia et al. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
- PotentIn VitroAntiproliferative Synergism of Combinations of Ergosterol Biosynthesis Inhibitors against Leishmania amazonensis
- (2015) S. T. de Macedo-Silva et al. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
- In vitro and in vivo antileishmanial properties of a 2- n -propylquinoline hydroxypropyl β-cyclodextrin formulation and pharmacokinetics via intravenous route
- (2015) Kaluvu Balaraman et al. BIOMEDICINE & PHARMACOTHERAPY
- 4-Aminoquinoline Derivatives as Potential Antileishmanial Agents
- (2015) Luciana M. R. Antinarelli et al. Chemical Biology & Drug Design
- A review on anticancer potential of bioactive heterocycle quinoline
- (2015) Obaid Afzal et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- 4-Amino Bis-Pyridinium Derivatives as Novel Antileishmanial Agents
- (2014) Verónica Gómez-Pérez et al. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
- Quinoline: A promising antitubercular target
- (2014) Rangappa S. Keri et al. BIOMEDICINE & PHARMACOTHERAPY
- Synthesis of novel triazole-linked mefloquine derivatives: Biological evaluation against Plasmodium falciparum
- (2014) Anton R. Hamann et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- New Compounds Hybrids 1H-1,2,3-Triazole-Quinoline AgainstPlasmodium falciparum
- (2014) Núbia Boechat et al. Chemical Biology & Drug Design
- Antiplasmodial activity of chloroquine analogs against chloroquine-resistant parasites, docking studies and mechanisms of drug action
- (2014) Nicolli B de Souza et al. MALARIA JOURNAL
- 7-Chloro-4-quinolinyl Hydrazones: A Promising and Potent Class of Antileishmanial Compounds
- (2013) Elaine S. Coimbra et al. Chemical Biology & Drug Design
- Potent naphthoquinones against antimony-sensitive and -resistant Leishmania parasites: Synthesis of novel α- and nor-α-lapachone-based 1,2,3-triazoles by copper-catalyzed azide–alkyne cycloaddition
- (2013) Tiago T. Guimarães et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Mitochondrial Dysfunction Induces Formation of Lipid Droplets as a Generalized Response to Stress
- (2013) Seon-Jin Lee et al. Oxidative Medicine and Cellular Longevity
- In Vitro Activity of the Antifungal Azoles Itraconazole and Posaconazole against Leishmania amazonensis
- (2013) Sara Teixeira de Macedo-Silva et al. PLoS One
- Apoptosis-induced mitochondrial dysfunction causes cytoplasmic lipid droplet formation
- (2012) J Boren et al. CELL DEATH AND DIFFERENTIATION
- Mitochondrial damage contribute to epigallocatechin-3-gallate induced death in Leishmania amazonensis
- (2012) Job D.F. Inacio et al. EXPERIMENTAL PARASITOLOGY
- Cell death features induced in Leishmania major by 1,3,4-thiadiazole derivatives
- (2012) Sussan K. Ardestani et al. EXPERIMENTAL PARASITOLOGY
- Leishmaniasis Worldwide and Global Estimates of Its Incidence
- (2012) Jorge Alvar et al. PLoS One
- Redox-Active Antiparasitic Drugs
- (2011) Chinmay Pal et al. ANTIOXIDANTS & REDOX SIGNALING
- Synthesis of 4-aminoquinoline analogues and their platinum(II) complexes as new antileishmanial and antitubercular agents
- (2011) Arturene M.L. Carmo et al. BIOMEDICINE & PHARMACOTHERAPY
- Synthesis of quinoline coupled [1,2,3]-triazoles as a promising class of anti-tuberculosis agents
- (2011) K. Karthik Kumar et al. CARBOHYDRATE RESEARCH
- Synthesis of a Star Polymer Library with a Diverse Range of Highly Functionalized Macromolecular Architectures
- (2011) Jing M. Ren et al. MACROMOLECULES
- Synthesis and antimicrobial activity of 1,2,3-triazoles containing quinoline moiety
- (2010) V. Sumangala et al. ARCHIVES OF PHARMACAL RESEARCH
- Morphological and physiological changes in Leishmania promastigotes induced by yangambin, a lignan obtained from Ocotea duckei
- (2010) Rubens L. Monte Neto et al. EXPERIMENTAL PARASITOLOGY
- Secondary necrosis: The natural outcome of the complete apoptotic program
- (2010) Manuel T. Silva FEBS LETTERS
- Targeting essential pathways in trypanosomatids gives insights into protozoan mechanisms of cell death
- (2010) Despina Smirlis et al. Parasites & Vectors
- In Vitro Activities of ER-119884 and E5700, Two Potent Squalene Synthase Inhibitors, against Leishmania amazonensis: Antiproliferative, Biochemical, and Ultrastructural Effects
- (2008) J. C. Fernandes Rodrigues et al. ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
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