Ester to amide substitution improves selectivity, efficacy and kinetic behavior of a benzodiazepine positive modulator of GABA A receptors containing the α5 subunit

标题
Ester to amide substitution improves selectivity, efficacy and kinetic behavior of a benzodiazepine positive modulator of GABA A receptors containing the α5 subunit
作者
关键词
Amide compound, Receptor efficacy, Binding assay, Free brain concentration, Rat kinetics, Basic behavior
出版物
EUROPEAN JOURNAL OF PHARMACOLOGY
Volume 791, Issue -, Pages 433-443
出版商
Elsevier BV
发表日期
2016-09-16
DOI
10.1016/j.ejphar.2016.09.016

向作者/读者发起求助以获取更多资源

Reprint

联系作者

Publish scientific posters with Peeref

Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.

Learn More

Create your own webinar

Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.

Create Now