Modulating the function of ABCB1: in vitro and in vivo characterization of sitravatinib, a tyrosine kinase inhibitor
出版年份 2020 全文链接
标题
Modulating the function of ABCB1:
in vitro
and
in vivo
characterization of sitravatinib, a tyrosine kinase inhibitor
作者
关键词
-
出版物
Cancer Communications
Volume 40, Issue 7, Pages 285-300
出版商
Wiley
发表日期
2020-06-11
DOI
10.1002/cac2.12040
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- Sitravatinib, a Tyrosine Kinase Inhibitor, Inhibits the Transport Function of ABCG2 and Restores Sensitivity to Chemotherapy-Resistant Cancer Cells in vitro
- (2020) Yuqi Yang et al. Frontiers in Oncology
- Glesatinib, a c-MET/SMO Dual Inhibitor, Antagonizes P-glycoprotein Mediated Multidrug Resistance in Cancer Cells
- (2019) Qingbin Cui et al. Frontiers in Oncology
- Enhanced efficacy of sitravatinib in metastatic models of antiangiogenic therapy resistance
- (2019) Melissa Dolan et al. PLoS One
- Midostaurin Reverses ABCB1-Mediated Multidrug Resistance, an in vitro Study
- (2019) Ning Ji et al. Frontiers in Oncology
- Metabolic reprogramming and redox adaptation in sorafenib-resistant leukemia cells: detected by untargeted metabolomics and stable isotope tracing analysis
- (2019) Xin You et al. Cancer Communications
- Tepotinib reverses ABCB1-mediated multidrug resistance in cancer cells
- (2019) Zhuo-Xun Wu et al. BIOCHEMICAL PHARMACOLOGY
- Pathological transition as the arising mechanism for drug resistance in lung cancer
- (2019) Yueqing Chen et al. Cancer Communications
- Benzoyl indoles with metabolic stability as reversal agents for ABCG2-mediated multidrug resistance
- (2019) Chao-Yun Cai et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Derivative of 5-cyano-6-phenylpyrimidin antagonizes ABCB1- and ABCG2-mediated multidrug resistance
- (2019) Jing-Quan Wang et al. EUROPEAN JOURNAL OF PHARMACOLOGY
- Epidermal growth factor receptor (EGFR) inhibitor PD153035 reverses ABCG2-mediated multidrug resistance in non-small cell lung cancer: In vitro and in vivo
- (2018) Guan-Nan Zhang et al. CANCER LETTERS
- Radioresistant Cervical Cancers Are Sensitive to Inhibition of Glycolysis and Redox Metabolism
- (2018) Ramachandran Rashmi et al. CANCER RESEARCH
- Discovery of 5-Cyano-6-phenylpyrimidin Derivatives Containing an Acylurea Moiety as Orally Bioavailable Reversal Agents against P-Glycoprotein-Mediated Mutidrug Resistance
- (2018) Bo Wang et al. JOURNAL OF MEDICINAL CHEMISTRY
- Tumor-Independent Host Secretomes Induced By Angiogenesis and Immune-Checkpoint Inhibitors
- (2018) Michalis Mastri et al. MOLECULAR CANCER THERAPEUTICS
- Structure of a zosuquidar and UIC2-bound human-mouse chimeric ABCB1
- (2018) Amer Alam et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Ulixertinib (BVD-523) antagonizes ABCB1- and ABCG2-mediated chemotherapeutic drug resistance
- (2018) Ning Ji et al. BIOCHEMICAL PHARMACOLOGY
- Modulating ROS to overcome multidrug resistance in cancer
- (2018) Qingbin Cui et al. DRUG RESISTANCE UPDATES
- Outcomes of 219 chronic myeloid leukaemia patients with additional chromosomal abnormalities and/or tyrosine kinase domain mutations
- (2018) Mingming Xue et al. International Journal of Laboratory Hematology
- VS-4718 Antagonizes Multidrug Resistance in ABCB1- and ABCG2-Overexpressing Cancer Cells by Inhibiting the Efflux Function of ABC Transporters
- (2018) Ning Ji et al. Frontiers in Pharmacology
- Regorafenib antagonizes BCRP-mediated multidrug resistance in colon cancer
- (2018) Yun-Kai Zhang et al. CANCER LETTERS
- Second- and third-generation drugs for immuno-oncology treatment—The more the better?
- (2017) Wolfram C.M. Dempke et al. EUROPEAN JOURNAL OF CANCER
- Significance of preoperative prognostic nutrition index as prognostic predictors in patients with metastatic renal cell carcinoma with tyrosine kinase inhibitors as first-line target therapy
- (2017) Wen Cai et al. INTERNATIONAL UROLOGY AND NEPHROLOGY
- Uterine metastasis of lung adenocarcinoma under molecular target therapy with epidermal growth factor receptor tyrosine kinase inhibitors: A case report and review of the literature
- (2017) Mayu Shibata et al. JOURNAL OF OBSTETRICS AND GYNAECOLOGY RESEARCH
- pH-Sensitive Nano-Complexes Overcome Drug Resistance and Inhibit Metastasis of Breast Cancer by Silencing Akt Expression
- (2017) Jieying Yin et al. Theranostics
- Overcoming ABC transporter-mediated multidrug resistance: Molecular mechanisms and novel therapeutic drug strategies
- (2016) Wen Li et al. DRUG RESISTANCE UPDATES
- Alantolactone selectively ablates acute myeloid leukemia stem and progenitor cells
- (2016) Yahui Ding et al. Journal of Hematology & Oncology
- Patient-derived xenograft (PDX) tumors increase growth rate with time
- (2016) Alexander T. Pearson et al. Oncotarget
- DNA Repair and Cytokines: TGF-β, IL-6, and Thrombopoietin as Different Biomarkers of Radioresistance
- (2016) Lucia Centurione et al. Frontiers in Oncology
- Multidrug Resistance Proteins (MRPs) and Cancer Therapy
- (2015) Yun-Kai Zhang et al. AAPS Journal
- The modulation of ABC transporter-mediated multidrug resistance in cancer: A review of the past decade
- (2015) Rishil J. Kathawala et al. DRUG RESISTANCE UPDATES
- Significant blockade of multiple receptor tyrosine kinases by MGCD516 (Sitravatinib), a novel small molecule inhibitor, shows potent anti-tumor activity in preclinical models of sarcoma
- (2015) Parag P. Patwardhan et al. Oncotarget
- In vitro,in vivoandex vivocharacterization of ibrutinib: a potent inhibitor of the efflux function of the transporter MRP1
- (2014) Hui Zhang et al. BRITISH JOURNAL OF PHARMACOLOGY
- Down-regulation of c-fos by shRNA sensitizes adriamycin-resistant MCF-7/ADR cells to chemotherapeutic agents via P-glycoprotein inhibition and apoptosis augmentation
- (2013) Ruizan Shi et al. JOURNAL OF CELLULAR BIOCHEMISTRY
- Enzymatic features of the glucose metabolism in tumor cells
- (2011) Anique Herling et al. FEBS Journal
- Reversion of Multidrug Resistance in Tumor By Biocompatible Nanomaterials
- (2010) H. Zhang et al. MINI-REVIEWS IN MEDICINAL CHEMISTRY
- Lipid dependence of ABC transporter localization and function
- (2009) Karin Klappe et al. CHEMISTRY AND PHYSICS OF LIPIDS
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