Synthesis and biological evaluation of 12 novel (-)-camphene-based 1,3,4-thiadiazoles against Mycobacterium tuberculosis

Hydrazone, benzohydrazones and isoniazid-acylhydrazones as potential antituberculosis agents

(2019) Eloísa G Sampiron et al.   Future Microbiology

The Role of Efflux Pumps in Tuberculosis Treatment and Their Promise as a Target in Drug Development: Unraveling the Black Box

(2018) Lindsey H.M. te Brake et al.   Annual Review of Pharmacology and Toxicology

Carvacrol activity & morphological changes in Mycobacterium tuberculosis

(2018) Sandra S Nakamura de Vasconcelos et al.   Future Microbiology

Synthesis of novel (-)-Camphene-based thiosemicarbazones and evaluation of anti-Mycobacterium tuberculosis activity

(2018) Mariana R. P. Souza et al.   NATURAL PRODUCT RESEARCH

2-Amino-1,3,4-thiadiazole as a potential scaffold for promising antimicrobial agents

(2018) Georgeta Serban et al.   Drug Design Development and Therapy

The host microbiome and impact of tuberculosis chemotherapy

(2018) Ronan F. O'Toole et al.   TUBERCULOSIS

Diversity and evolution of drug resistance mechanisms in Mycobacterium tuberculosis

(2017) Mashael Al-Saeedi et al.   Infection and Drug Resistance

Synthesis and evaluation of the trypanocidal activity of a series of 1,3,4-thiadiazoles derivatives of R-(+)-limonene benzaldehyde-thiosemicarbazones

(2016) Solange C. Martins et al.   MEDICINAL CHEMISTRY RESEARCH

Morphological changes and differentially expressed efflux pump genes in Mycobacterium tuberculosis exposed to a rifampicin and verapamil combination

(2016) Katiany R. Caleffi-Ferracioli et al.   TUBERCULOSIS

Synthesis and antimicrobial evaluation of novel 1,3,4-thiadiazole derivatives of 2-(4-formyl-2-methoxyphenoxy) acetic acid

(2016) Malleshappa N. Noolvi et al.   Arabian Journal of Chemistry

Ion Channel Blockers as Antimicrobial Agents, Efflux Inhibitors, and Enhancers of Macrophage Killing Activity against Drug Resistant Mycobacterium tuberculosis

(2016) Diana Machado et al.   PLoS One

Cyrhetrenyl and ferrocenyl 1,3,4-thiadiazole derivatives: Synthesis, characterization, crystal structures and in vitro antitubercular activity

(2015) Cristóbal Quintana et al.   INORGANIC CHEMISTRY COMMUNICATIONS

Detection of drug susceptibility in rapidly growing mycobacteria by resazurin broth microdilution assay

(2015) Aline Lemes Castilho et al.   JOURNAL OF MICROBIOLOGICAL METHODS

Antimycobacterial activity of chiral aminoalcohols with camphane scaffold

(2014) Zhanina Petkova et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Anti-Mycobacterium tuberculosis activity and cytotoxicity of Calophyllum brasiliense Cambess (Clusiaceae)

(2014) Claudia Terencio Agostinho Pires et al.   MEMORIAS DO INSTITUTO OSWALDO CRUZ

Characterization of Antibacterial and Hemolytic Activity of Synthetic Pandinin 2 Variants and Their Inhibition against Mycobacterium tuberculosis

(2014) Alexis Rodríguez et al.   PLoS One

Anti-mycobacterial activities of synthetic cationic α-helical peptides and their synergism with rifampicin

(2013) Jasmeet S. Khara et al.   BIOMATERIALS

Fast detection of drug interaction in Mycobacterium tuberculosis by a checkerboard resazurin method

(2013) Katiany R. Caleffi-Ferracioli et al.   TUBERCULOSIS

Evaluation of the microscopic observation drug susceptibility assay for detection of Mycobacterium tuberculosis resistance to pyrazinamide

(2011) L.D. Ghiraldi et al.   CLINICAL MICROBIOLOGY AND INFECTION

In-Silico ADME Models: A General Assessment of their Utility in Drug Discovery Applications

(2011) M. Paul Gleeson et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Efflux as a mechanism for drug resistance inMycobacterium tuberculosis: Table 1

(2011) Pedro Eduardo Almeida da Silva et al.   FEMS IMMUNOLOGY AND MEDICAL MICROBIOLOGY

Rapid detection of resistance to pyrazinamide in Mycobacterium tuberculosis using the resazurin microtitre assay

(2011) P. A. Z. Campanerut et al.   JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY

The challenge of new drug discovery for tuberculosis

(2011) Anil Koul et al.   NATURE

Amino Acid Derivatives, Part 4: Synthesis and Anti-HIV Activity of New Naphthalene Derivatives

(2010) Nawar S. Hamad et al.   ARCHIV DER PHARMAZIE

Synthesis and anticancer activity of 5-(3-indolyl)-1,3,4-thiadiazoles

(2010) Dalip Kumar et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2-Amino-5-sulfanyl-1,3,4-thiadiazoles: a novel series of anti-inflammatory and analgesic agents

(2009) Jitendra Sainy et al.   PHARMACEUTICAL CHEMISTRY JOURNAL

Biological activity of 1,2,3,4-tetrahydro-β-carboline-3-carboxamides against Trypanosoma cruzi

(2008) Rodrigo Hinojosa Valdez et al.   ACTA TROPICA