Brønsted Acid Catalyzed [3+2]-Cycloaddition of 2-Vinylindoles with In Situ Generated 2-Methide-2H-indoles: Highly Enantioselective Synthesis of Pyrrolo[1,2-a]indoles

Organocatalytic asymmetric reaction of indol-2-yl carbinols with enamides: synthesis of chiral 2-indole-substituted 1,1-diarylalkanes

(2015) Chao-You Liu et al.   CHEMICAL COMMUNICATIONS

Strategies for the asymmetric functionalization of indoles: an update

(2015) Renato Dalpozzo   CHEMICAL SOCIETY REVIEWS

Enantioselective construction of a 2,2′-bisindolylmethane scaffold via catalytic asymmetric reactions of 2-indolylmethanols with 3-alkylindoles

(2015) Yu-Xin Gong et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthetic Study toward the Misassigned (±)-Tronoharine

(2015) Xue Zhong et al.   ORGANIC LETTERS

Counter-Ion-Dependent Alkyne Iminium Ion Cyclization for Divergent Synthesis of N-Fused Indolylidine, Indole, and Indoline Derivatives Promoted by the Lewis/Bronsted Acid

(2015) Santosh J. Gharpure et al.   ORGANIC LETTERS

Enantioselective hydroacylation of N-vinylindole-2-carboxaldehydes

(2014) Avipsa Ghosh et al.   CHEMICAL COMMUNICATIONS

A metal free domino synthesis of 3-aroylindoles via two sp3 C–H activation

(2014) Anupal Gogoi et al.   CHEMICAL COMMUNICATIONS

Formal [3+3] cycloaddition of indol-2-yl carbinol with azadiene and the oxidative ring expansion reaction for the synthesis of indole azepinones

(2014) Xue Zhong et al.   CHEMICAL COMMUNICATIONS

Chiral phosphoramide-catalyzed enantioselective synthesis of 2,3′-diindolylarylmethanes from indol-2-yl carbinols and indoles

(2014) Shuai Qi et al.   CHEMICAL COMMUNICATIONS

Synthetic Approaches to 3-(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

(2014) Stefano Lancianesi et al.   CHEMICAL REVIEWS

Complete Field Guide to Asymmetric BINOL-Phosphate Derived Brønsted Acid and Metal Catalysis: History and Classification by Mode of Activation; Brønsted Acidity, Hydrogen Bonding, Ion Pairing, and Metal Phosphates

(2014) Dixit Parmar et al.   CHEMICAL REVIEWS

One-Pot Asymmetric Synthesis of Quaternary Pyrroloindolones through a Multicatalytic N-Allylation/Hydroacylation Sequence

(2014) Hong Lu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Pyrroloindolone Synthesis via a Cp*CoIII-Catalyzed Redox-Neutral Directed C–H Alkenylation/Annulation Sequence

(2014) Hideya Ikemoto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Imine and iminium precursors as versatile intermediates in enantioselective organocatalysis

(2014) Antti O. Kataja et al.   TETRAHEDRON

Microwave-assisted facile synthesis of [a]-annelated pyrazolopyrroloindoles via intramolecular azomethine imine 1,3-dipolar cycloaddition

(2014) Anand H. Shinde et al.   TETRAHEDRON LETTERS

Asymmetric Synthesis of Pyrroloindolones by N-Heterocyclic Carbene Catalyzed [2+3] Annulation of α-Chloroaldehydes with Nitrovinylindoles

(2013) Qijian Ni et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Friedel-Crafts Alkylation/N-Hemiacetalization Cascade Reaction with Indoles

(2013) Hong-Gang Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cu(OTf)2 catalysed [6+2] cycloaddition reaction for the synthesis of highly substituted pyrrolo[1,2-a]indoles: rapid construction of the yuremamine core

(2013) Dattatraya H. Dethe et al.   CHEMICAL COMMUNICATIONS

Synthesis of (±)-Actinophyllic Acid and Analogs: Applications of Cascade Reactions and Diverted Total Synthesis

(2013) Brett A. Granger et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pd(II)-catalyzed intramolecular aminopalladation/direct C–H arylation under aerobic conditions: synthesis of pyrrolo[1,2-a]indoles

(2013) Tiffany Piou et al.   TETRAHEDRON

AsymmetricN-Allylation of Indoles Through the Iridium-Catalyzed Allylic Alkylation/Oxidation of Indolines

(2012) Wen-Bo Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Thermally induced [3+2] cyclization of aniline-tethered alkylidenecyclopropanes: a facile synthetic protocol of pyrrolo[1,2-a]indoles

(2012) Kai Chen et al.   CHEMICAL COMMUNICATIONS

Quadruple Domino Organocatalysis: An Asymmetric Aza-Michael/Michael/Michael/Aldol Reaction Sequence Leading to Tetracyclic Indole Structures with Six Stereocenters

(2012) Dieter Enders et al.   CHEMISTRY-A EUROPEAN JOURNAL

Al-Catalyzed Facile Construction of Quaternary CC Bonds by the Allylic Substitution of Tertiary Alcohols: A Concise and Formal Synthesis of (±)-Mersicarpine

(2012) Xue Zhong et al.   CHEMISTRY-A EUROPEAN JOURNAL

Biomimetic Synthesis of the Antimalarial Flindersial Alkaloids

(2012) Ravikrishna Vallakati et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Complementary Asymmetric Routes to (R)-2-(7-Hydroxy-2,3-dihydro-1H-pyrrolo[1,2-a]indol-1-yl)acetate

(2012) Thomas O. Schrader et al.   ORGANIC LETTERS

Indole synthesis – something old, something new

(2012) Martyn Inman et al.   Chemical Science

Modulating the Acidity: Highly Acidic Brønsted Acids in Asymmetric Catalysis

(2011) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acids in enantioselective carbonyl activations – activation modes and applications

(2011) Magnus Rueping et al.   CHEMICAL SOCIETY REVIEWS

Biomimetic Total Syntheses of Flinderoles B and C

(2011) Dattatraya H. Dethe et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diastereoselective Intramolecular Friedel–Crafts Cyclizations of Substituted Methyl 2-(1H-indole-1-carbonyl)acrylates: Efficient Access to Functionalized 1H-Pyrrolo[1,2-a]indoles

(2011) Dadasaheb V. Patil et al.   ORGANIC LETTERS

Synthesis of flinderoles B and C by a gold-catalyzed allene hydroarylation

(2011) Rachel M. Zeldin et al.   Chemical Science

Chemoselective Cascade Synthesis of N-Fused Heterocycles via Silver(I) Triflate-Catalyzed Friedel-Crafts/N-C Bond Formation Sequence

(2010) Lu Hao et al.   ADVANCED SYNTHESIS & CATALYSIS

Chiral Phosphoric Acids as Versatile Catalysts for Enantioselective Carbon–Carbon Bond Forming Reactions

(2010) Masahiro Terada   BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

N-Heterocyclic Carbene Catalyzed Domino Reactions of Formylcyclopropane 1,1-Diesters: Construction of a 6-5-5 Tricyclic Pyrrolo[1,2-a]indole

(2010) Linxia Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Antiparasitic activity of alkaloids from plant species of Papua New Guinea and Australia

(2010) Liza S. Fernandez et al.   INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS

Chiral Phosphoric Acids as Versatile Catalysts for Enantioselective Transformations

(2010) Masahiro Terada   SYNTHESIS-STUTTGART

Palladium-Catalyzed Sequential Reactions via Allene Intermediates for the Rapid Synthesis of Fused Polycyclic Pyrrole Derivatives

(2009) Xian Huang et al.   ADVANCED SYNTHESIS & CATALYSIS

Chemoselective Asymmetric N-Allylic Alkylation of Indoles with Morita-Baylis-Hillman Carbonates

(2009) Hai-Lei Cui et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iridium-Catalyzed Regio- and Enantioselective N-Allylation of Indoles

(2009) Levi M. Stanley et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Organocatalytic N-Alkylation of Indole-2-carbaldehydes with α,β-Unsaturated Aldehydes: One-Pot Synthesis of Chiral Pyrrolo[1,2-a]indole-2-carbaldehydes

(2009) Liang Hong et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of β-heteroaryl propionates via trapping of carbocations with π-nucleophiles

(2009) Tsung-hao Fu et al.   TETRAHEDRON LETTERS

Binaphthol-derived phosphoric acid as a versatile catalyst for enantioselective carbon–carbon bond forming reactions

(2008) Masahiro Terada   CHEMICAL COMMUNICATIONS

Expedient Synthesis of Pyrrolo[1,2-a]indoles: Preparation of the Core of Yuremamine

(2008) Michael B. Johansen et al.   ORGANIC LETTERS

Flinderoles A−C: Antimalarial Bis-indole Alkaloids fromFlindersiaSpecies

(2008) Liza S. Fernandez et al.   ORGANIC LETTERS

An efficient synthesis of 9H-pyrrolo[1,2-a]indoles

(2008) Kasey Wood et al.   TETRAHEDRON LETTERS