Remarkably flexible quinazolinones—synthesis and biological applications

Polydopamine: An Amine Oxidase Mimicking Sustainable Catalyst for the Synthesis of Nitrogen Heterocycles under Aqueous Conditions

(2019) Shweta Anil Pawar et al.   ACS Sustainable Chemistry & Engineering

Palladium Catalyzed Cross -Dehydrogenative Coupling/Annulation Reaction: A Practical and Efficient Approach to Hydroxyisoindolo[1,2-b ]quinazolinone

(2019) Minoo Dabiri et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Identification of Promising Biofilm Inhibitory and Cytotoxic Quinazolin‐4‐one Derivatives: Synthesis, Evaluation, Molecular Docking and ADMET Studies

(2019) Siddique A. Ansari et al.   ChemistrySelect

Discovery of coumarin-dihydroquinazolinone analogs as niacin receptor 1 agonist with in-vivo anti-obesity efficacy

(2018) L. Ravithej Singh et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis and biological activities of 2,3-dihydroquinazolin-4(1 H )-one derivatives as TRPM2 inhibitors

(2018) Han Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis and biological evaluation of novel quinazoline-2,4-diones conjugated with different amino acids as potential chitin synthase inhibitors

(2018) Nada A. Noureldin et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Quinazoline and quinazolinone as important medicinal scaffolds: a comparative patent review (2011–2016)

(2018) Abdul Hameed et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Synthesis and evaluation of 2-substituted 4(3H)-quinazolinone thioether derivatives as monoamine oxidase inhibitors

(2018) Malikotsi A. Qhobosheane et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Isoxazolidine Conjugates of N3-Substituted 6-Bromoquinazolinones—Synthesis, Anti-Varizella-Zoster Virus, and Anti-Cytomegalovirus Activity

(2018) Magdalena Grabkowska-Drużyc et al.   MOLECULES

Design, synthesis and cytotoxic evaluation of novel imidazolone fused quinazolinone derivatives

(2017) Deepak Kumar et al.   Arabian Journal of Chemistry

One-pot synthesis of benzazoles and quinazolinones via iron pentacarbonyl mediated carbonylation of aryl iodides under microwave irradiation

(2017) Wun-Huei Lin et al.   Organic Chemistry Frontiers

A Quinazolinone based fluorescent chemosensor for selective detection of Fe(III) in aqueous media: Applications to pharmaceutical and environmental analysis

(2017) Pravin R. Dongare et al.   Inorganic and Nano-Metal Chemistry

Synthesis, anti-inflammatory, analgesic, COX-1/2 inhibitory activities and molecular docking studies of substituted 2-mercapto-4(3 H )-quinazolinones

(2016) Alaa A.-M. Abdel-Aziz et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antitumor evaluation of trimethoxyanilides based on 4(3 H )-quinazolinone scaffolds

(2016) Menshawy A. Mohamed et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Vasodilation and hypotension of a novel 3-benzylquinazolin- 4(3 H )-one derivative via the inhibition of calcium flux

(2016) Sen Li et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

Solvent-free copper-catalyzed three-component synthesis of 2-substituted quinazolin-4(3H)-ones

(2016) Mehdi Soheilizad et al.   MONATSHEFTE FUR CHEMIE

Advanced Synthetic Strategies for Constructing Quinazolinone Scaffolds

(2016) Umesh Kshirsagar et al.   SYNTHESIS-STUTTGART

Efficient synthesis of 2,3-dihydroquinazolin-4(1H)-ones catalyzed by titanium silicon oxide nanopowder in aqueous media

(2016) Ramamohan Mekala et al.   SYNTHETIC COMMUNICATIONS

Synthetic approaches, functionalization and therapeutic potential of quinazoline and quinazolinone skeletons: The advances continue

(2015) Imtiaz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of quinazolines and quinazolinones via palladium-mediated approach

(2015) Ibrahim M. Abdou et al.   HETEROCYCLIC COMMUNICATIONS

Recent developments in the chemistry of quinazolinone alkaloids

(2015) U. A. Kshirsagar   ORGANIC & BIOMOLECULAR CHEMISTRY

An environment-friendly synthesis of 4(3H)-quinazolinones

(2015) Haidong Wei et al.   TOXICOLOGICAL AND ENVIRONMENTAL CHEMISTRY

The chemistry and biology of febrifugine and halofuginone

(2014) Noel P. McLaughlin et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Recent advances in the structural library of functionalized quinazoline and quinazolinone scaffolds: Synthetic approaches and multifarious applications

(2014) Imtiaz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, Anti-microbial and Molecular Docking Studies of Quinazolin-4(3H)-one Derivatives

(2014) Yahia Mabkhot et al.   MOLECULES

Pd-Catalyzed Intramolecular Aerobic Oxidative C–H Amination of 2-Aryl-3-(arylamino)quinazolinones: Synthesis of Fluorescent Indazolo[3,2-b]quinazolinones

(2014) Weiguang Yang et al.   ORGANIC LETTERS

An Efficient Synthesis of 2-Substituted Quinazolin-4(3H)-ones Catalyzed by Iron(III) Chloride

(2014) Jayaprakash Sarva et al.   SYNLETT

Urea/Thiourea as Ammonia Surrogate: A Catalyst-Free Synthesis of 2-Substituted 2,3-Dihydroquinazolin-4(1H)-ones/Quinazoline-4(3H)-ones

(2014) P. Paradesi Naidu et al.   SYNTHETIC COMMUNICATIONS

Recent advances in 4(3H)-quinazolinone syntheses

(2014) Lin He et al.   RSC Advances

A Novel Quinazolinone Derivative as Fluorescence Quenching Off-On Sensor for High Selectivity of Fe3+

(2013) Ailin Yuan et al.   JOURNAL OF FLUORESCENCE

Discovery of a New Class of Natural Product-Inspired Quinazolinone Hybrid as Potent Antileishmanial agents

(2013) Moni Sharma et al.   JOURNAL OF MEDICINAL CHEMISTRY

Amino acid-based ionic liquid immobilized on α-Fe2O3-MCM-41: An efficient magnetic nanocatalyst and recyclable reaction media for the synthesis of quinazolin-4(3H)-one derivatives

(2013) Shahnaz Rostamizadeh et al.   JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL

Synthesis and crystal structure of bis [2-(4-methylphenyl)-1-phenethyl-4(1H)-quinazolinone] dichlorocopper (II)

(2012) G.Y.S.K. Swamy et al.   POLYHEDRON

Analogue-based design, synthesis and molecular docking analysis of 2,3-diaryl quinazolinones as non-ulcerogenic anti-inflammatory agents

(2011) E. Manivannan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Yb(OTf)3 catalyzed new cascade reaction: a facile assembly of fused quinazolinones

(2011) K. Siva Kumar et al.   CHEMICAL COMMUNICATIONS

Use of Structure-Based Design to Discover a Potent, Selective, In Vivo Active Phosphodiesterase 10A Inhibitor Lead Series for the Treatment of Schizophrenia

(2011) Christopher J. Helal et al.   JOURNAL OF MEDICINAL CHEMISTRY

One-Pot Synthesis of Quinazolinones via Iridium-Catalyzed Hydrogen Transfers

(2011) Jianguang Zhou et al.   JOURNAL OF ORGANIC CHEMISTRY

Cyanuric Chloride Catalyzed Mild Protocol for Synthesis of Biologically Active Dihydro/Spiro Quinazolinones and Quinazolinone-glycoconjugates

(2011) Moni Sharma et al.   JOURNAL OF ORGANIC CHEMISTRY

Green and One-Pot Three-Component Synthesis of 2,3-Dihydroquinazolin- 4(1H)-Ones Promoted by Citric Acid as Recoverable Catalyst in Water

(2011) Arash Ghorbani-Choghamarani et al.   LETTERS IN ORGANIC CHEMISTRY

Highly efficient solvent-free synthesis of quinazolin-4(3H)-ones and 2,3-dihydroquinazolin-4(1H)-ones using tetrabutylammonium bromide as novel ionic liquid catalyst

(2010) A. Davoodnia et al.   CHINESE CHEMICAL LETTERS

Novel 6,8-dibromo-4(3H)quinazolinone derivatives of anti-bacterial and anti-fungal activities

(2010) Mosaad S. Mohamed et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of some new 4(3H)-quinazolinone-2-carboxaldehyde thiosemicarbazones and their metal complexes and a study on their anticonvulsant, analgesic, cytotoxic and antimicrobial activities – Part-1

(2010) Mohsen M. Aly et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and antitumor activity of some 2, 3-disubstituted quinazolin-4(3H)-ones and 4, 6- disubstituted- 1, 2, 3, 4-tetrahydroquinazolin-2H-ones

(2010) Nagwa M. Abdel Gawad et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Iodine: Selectively promote the synthesis of mono substituted quinazolin-4(3H)-ones and 2,3-dihydroquinazolin-4(1H)-ones in one-pot

(2010) Li-Yan Zeng et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

[bmim]HSO4: an efficient and reusable catalyst for one-pot three-component synthesis of 2,3-dihydro-4(1H)-quinazolinones

(2010) Nitin B. Darvatkar et al.   Green Chemistry Letters and Reviews

Asymmetric Brønsted Acid Catalysis: Catalytic Enantioselective Synthesis of Highly Biologically Active Dihydroquinazolinones

(2008) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

New pyrazoline bearing 4(3H)-quinazolinone inhibitors of monoamine oxidase: Synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity

(2008) Nesrin Gökhan-Kelekçi et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A novel catalyst zinc(II) perfluorooctanoate [Zn(PFO)2]-catalyzed three-component one-pot reaction: Synthesis of quinazolinone derivatives in aqueous micellar media

(2008) Li-Min Wang et al.   JOURNAL OF FLUORINE CHEMISTRY

Direct Catalytic Asymmetric Synthesis of Cyclic Aminals from Aldehydes

(2008) Xu Cheng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Click Reaction: Highly Efficient Synthesis of 2,3-Dihydroquinazolin-4(1H)-ones

(2008) Ahmad Shaabani et al.   SYNTHETIC COMMUNICATIONS

Gallium(III) triflate-catalyzed one-pot selective synthesis of 2,3-dihydroquinazolin-4(1H)-ones and quinazolin-4(3H)-ones

(2008) Jiuxi Chen et al.   TETRAHEDRON LETTERS