Discovery and structure–activity analysis of 4-((5-nitropyrimidin-4-yl)amino)benzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors

标题
Discovery and structure–activity analysis of 4-((5-nitropyrimidin-4-yl)amino)benzimidamide derivatives as novel protein arginine methyltransferase 1 (PRMT1) inhibitors
作者
关键词
PRMT1, Small molecule inhibitor, Epigenetics, Structure–activity relationship, Protein arginine methyltransferase
出版物
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Volume 25, Issue 22, Pages 5449-5453
出版商
Elsevier BV
发表日期
2015-07-05
DOI
10.1016/j.bmcl.2015.06.095

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