Catalytic Asymmetric Synthesis of 3-Indolyl Methanamines Using Unprotected Indoles and N-Boc Imines under Basic Conditions

Enantioselective Construction of Cyclic Indolyl α-Amino Estersviaa Friedel-Crafts Alkylation Reaction

(2015) Liang Wu et al.   ADVANCED SYNTHESIS & CATALYSIS

Dual Catalysis for the Redox Annulation of Nitroalkynes with Indoles: Enantioselective Construction of Indolin-3-ones Bearing Quaternary Stereocenters

(2015) Ren-Rong Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

3-Pyrrolyl-oxindoles as efficient nucleophiles for organocatalytic asymmetric synthesis of structurally diverse 3,3′-disubstituted oxindole derivatives

(2015) Bao-Dong Cui et al.   CHEMICAL COMMUNICATIONS

Catalytic Enantioselective Reaction of α-Phenylthioacetonitriles with Imines Using Chiral Bis(imidazoline)-Palladium Catalysts

(2015) Masaru Kondo et al.   CHEMISTRY-A EUROPEAN JOURNAL

Chiral Bis(imidazolidine)-Derived NCN Pincer Rh Complex for Catalytic Asymmetric Mannich Reaction of Malononitrile withN-Boc Imines

(2015) Takayoshi Arai et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis, molecular modeling, and biological evaluation of novel RAD51 inhibitors

(2015) Jiewen Zhu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Telescoped Synthesis of 2-Acyl-1-aryl-1,2-dihydroisoquinolines and Their Inhibition of the Transcription Factor NF-κB

(2015) Tsai-Wen Chung et al.   ACS Combinatorial Science

Anticancer activity of VDR-coregulator inhibitor PS121912

(2014) Preetpal S. Sidhu et al.   CANCER CHEMOTHERAPY AND PHARMACOLOGY

Enantioselective Continuous-Flow Production of 3-Indolylmethanamines Mediated by an Immobilized Phosphoric Acid Catalyst

(2014) Laura Osorio-Planes et al.   CHEMISTRY-A EUROPEAN JOURNAL

Chiral BrOnsted Acid-Catalyzed Friedel-Crafts Reaction of Indoles

(2014) Pinaki Bhadury et al.   CURRENT ORGANIC CHEMISTRY

Asymmetric Phase-Transfer Catalysts Bearing Multiple Hydrogen-Bonding Donors: Highly Efficient Catalysts for Enantio- and Diastereoselective Nitro-Mannich Reaction of Amidosulfones

(2014) Bin Wang et al.   ORGANIC LETTERS

Development of Novel Vitamin D Receptor–Coactivator Inhibitors

(2014) Preetpal S. Sidhu et al.   ACS Medicinal Chemistry Letters

Chiral Phosphoric Acid-Catalyzed Asymmetric Aza-Friedel-Crafts Reaction of Indoles with CyclicN-Acylketimines: Enantioselective Synthesis of Trifluoromethyldihydroquinazolines

(2013) Ke-Feng Zhang et al.   ADVANCED SYNTHESIS & CATALYSIS

Thiourea-phosphonium salts from amino acids: cooperative phase-transfer catalysts in the enantioselective aza-Henry reaction

(2013) Dongdong Cao et al.   CHEMICAL COMMUNICATIONS

Enantioselective methodologies using N-carbamoyl-imines

(2013) Jan Vesely et al.   CHEMICAL SOCIETY REVIEWS

A Neutral, Chiral, Bis(imidazolidine)-Derived NCN-Type Palladium Pincer Complex with Catalytic Activity

(2013) Takayoshi Arai et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Enantioselective Decarboxylative Cyanoalkylation of Imines by Using Palladium Pincer Complexes withC2-Symmetric Chiral Bis(imidazoline)s

(2013) Kengo Hyodo et al.   CHEMISTRY-A EUROPEAN JOURNAL

Leaving Group and Regioselectivity Switches in the Aminoalkylation Reaction of Indoles and Related Heterocycles with α-Amido Sulfones

(2013) Gonzalo Blay et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Disulfonimide-Catalyzed Asymmetric Synthesis of β3-Amino Esters Directly from N-Boc-Amino Sulfones

(2013) Qinggang Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chiral Brønsted acid-catalyzed enantioselective addition of indoles to ketimines

(2013) Taichi Kano et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Construction of Spiro-tetrahydroquinolines via Intramolecular Dearomatization of Quinolines: Free of a Preinstalled Activation Group

(2013) Shou-Guo Wang et al.   ORGANIC LETTERS

Catalyst-free coupling of indole derivatives with 3,4-dihydroisoquinoline and related compounds

(2013) István Szatmári et al.   TETRAHEDRON LETTERS

Enantioselective Addition of Thiols to Imines Catalyzed by Thiourea–Quaternary Ammonium Salts

(2013) Hong-Yu Wang et al.   ACS Catalysis

A Novel Method for Synthesizing N-Alkoxycarbonyl Aryl α-Imino Esters and Their Applications in Enantioselective Transformations

(2012) Yu Qian et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Friedel–Crafts reactions between phenols and N-tosylaldimines catalyzed by a leucine-derived bifunctional catalyst

(2012) Guo-Xing Li et al.   CHEMICAL COMMUNICATIONS

The highly enantioselective addition of indoles and pyrroles to isatins-derived N-Boc ketimines catalyzed by chiral phosphoric acids

(2012) Jingchao Feng et al.   CHEMICAL COMMUNICATIONS

Double Axially Chiral Bisphosphorylimides Catalyzed Highly Enantioselective and Efficient Friedel-Crafts Reaction of Indoles with Imines

(2012) Kun Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Vanadium-catalyzed enantioselective Friedel–Crafts-type reactions

(2012) Shinobu Takizawa et al.   DALTON TRANSACTIONS

A New Family of Cinchona-Derived Bifunctional Asymmetric Phase-Transfer Catalysts: Application to the Enantio- and Diastereoselective Nitro-Mannich Reaction of Amidosulfones

(2012) Kayli M. Johnson et al.   ORGANIC LETTERS

Highly Enantioselective Nitro-Mannich Reaction Catalyzed by Cinchona Alkaloids and N-Benzotriazole Derived Ammonium Salts

(2012) Yu Wei et al.   ORGANIC LETTERS

Asymmetric aza-Friedel–Crafts reaction of indoles induced by O-pivaloylated d-galactosylamine as the chiral auxiliary

(2012) Haohao Yang et al.   TETRAHEDRON

Enantioselective Reaction of Imines and Benzyl Nitriles Using Palladium Pincer Complexes withC2-Symmetric Chiral Bis(imidazoline)s

(2011) Kengo Hyodo et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Enantioselective Formation of C−C Bonds by Addition to Imines and Hydrazones: A Ten-Year Update

(2011) Shu̅ Kobayashi et al.   CHEMICAL REVIEWS

Enantioselective Mannich reaction of a highly reactive Horner–Wadsworth–Emmons reagent with imines catalyzed by a bifunctional thiourea

(2011) Depeng Zhao et al.   Chemical Science

Controlling Stereoselectivity in the Aminocatalytic Enantioselective Mannich Reaction of Aldehydes with In Situ Generated N-Carbamoyl Imines

(2010) Patrizia Galzerano et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalyzed Asymmetric Friedel-Crafts Reactions

(2010) Vincent Terrasson et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Highly Enantio- and Diastereoselective Mannich Reactions of Glycine Schiff Bases within situGeneratedN-Boc-imines Catalyzed by a Cinchona Alkaloid Thiourea

(2010) Haile Zhang et al.   ORGANIC LETTERS

Catalytic Asymmetric Mannich Reactions of Sulfonylacetates

(2009) Carlo Cassani et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Aza-Baylis–Hillman-Type Reaction of α,β-Unsaturated Aldehydes with In Situ GeneratedN-Boc- andN-Cbz-Imines

(2009) Sylva Číhalová et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Asymmetric Formal [3 + 2] Cycloaddition with in Situ-GeneratedN-Carbamoyl Nitrones

(2009) Claudio Gioia et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Enantioselective Aza-Friedel-Crafts Alkylation of Pyrroles with N-(Heteroarenesulfonyl)imines

(2009) Shuichi Nakamura et al.   SYNLETT

Aminocatalytic Enantioselectiveanti-Mannich Reaction of Aldehydes with In Situ GeneratedN-Cbz andN-Boc Imines

(2008) Chiara Gianelli et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Brønsted Acid Catalyzed Isoindoline Synthesis: Enhancement of Enantiomeric Ratio by Stereoablative Kinetic Resolution

(2008) Dieter Enders et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

9-Thiourea Cinchona alkaloid supported on mesoporous silica as a highly enantioselective, recyclable heterogeneous asymmetric catalyst

(2008) Peng Yu et al.   CHEMICAL COMMUNICATIONS

Reactions of In Situ GeneratedN-Boc Nitrones with Aromatic and Heteroaromatic Grignard Reagents:  Application to the Synthesis of Zileuton

(2008) Xavier Guinchard et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Enantiopure (S)-Indolylglycine by Organocatalyzed Friedel–Crafts Alkylation of Indole

(2007) Martin J. Wanner et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY