New insight into structure-activity of furan-based salicylate synthase (MbtI) inhibitors as potential antitubercular agents
出版年份 2019 全文链接
标题
New insight into structure-activity of furan-based salicylate synthase (MbtI) inhibitors as potential antitubercular agents
作者
关键词
-
出版物
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Volume 34, Issue 1, Pages 823-828
出版商
Informa UK Limited
发表日期
2019-03-20
DOI
10.1080/14756366.2019.1589462
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- Discovery and development of novel salicylate synthase (MbtI) furanic inhibitors as antitubercular agents
- (2018) Laurent R. Chiarelli et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Fluorine and Fluorinated Motifs in the Design and Application of Bioisosteres for Drug Design
- (2018) Nicholas A. Meanwell JOURNAL OF MEDICINAL CHEMISTRY
- New Chromane-Based Derivatives as Inhibitors of Mycobacterium tuberculosis Salicylate Synthase (MbtI): Preliminary Biological Evaluation and Molecular Modeling Studies
- (2018) Elena Pini et al. MOLECULES
- Global Epidemiology of Tuberculosis
- (2018) Katherine Floyd et al. SEMINARS IN RESPIRATORY AND CRITICAL CARE MEDICINE
- Nitro-Group-Containing Drugs
- (2018) Kunal Nepali et al. JOURNAL OF MEDICINAL CHEMISTRY
- Effectiveness and safety of bedaquiline-containing regimens in the treatment of MDR- and XDR-TB: a multicentre study
- (2017) Sergey E. Borisov et al. EUROPEAN RESPIRATORY JOURNAL
- Delamanid and bedaquiline to treat multidrug-resistant and extensively drug-resistant tuberculosis in children: a systematic review
- (2017) Lia D’Ambrosio et al. Journal of Thoracic Disease
- Iron Acquisition Pathways as Targets for Antitubercular Drugs
- (2016) Fiorella Meneghetti et al. CURRENT MEDICINAL CHEMISTRY
- Reliability analysis and optimization of the consensus docking approach for the development of virtual screening studies
- (2016) Giulio Poli et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Mycobacterium tuberculosis Low Molecular Weight Phosphatases (MPtpA and MPtpB): From Biological Insight to Inhibitors
- (2015) Luisa Fanzani et al. CURRENT MEDICINAL CHEMISTRY
- PAINS in the Assay: Chemical Mechanisms of Assay Interference and Promiscuous Enzymatic Inhibition Observed during a Sulfhydryl-Scavenging HTS
- (2015) Jayme L. Dahlin et al. JOURNAL OF MEDICINAL CHEMISTRY
- Receptor-based virtual screening evaluation for the identification of estrogen receptorβligands
- (2014) Tiziano Tuccinardi et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Advances in the development of new tuberculosis drugs and treatment regimens
- (2013) Alimuddin Zumla et al. NATURE REVIEWS DRUG DISCOVERY
- Synthesis, structure–activity relationships and stereochemical investigations of new tricyclic pyridazinone derivatives as potential STAT3 inhibitors
- (2013) Daniela Masciocchi et al. MedChemComm
- Resistance to fluoroquinolones and second-line injectable drugs: impact on multidrug-resistant TB outcomes
- (2012) Dennis Falzon et al. EUROPEAN RESPIRATORY JOURNAL
- Synthesis and evaluation of M. tuberculosis salicylate synthase (MbtI) inhibitors designed to probe plasticity in the active site
- (2012) Alexandra Manos-Turvey et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- The challenge of new drug discovery for tuberculosis
- (2011) Anil Koul et al. NATURE
- Inhibitors of the Salicylate Synthase (MbtI) from Mycobacterium tuberculosis Discovered by High-Throughput Screening
- (2010) Mahalakshmi Vasan et al. ChemMedChem
- Multidrug-resistant and extensively drug-resistant tuberculosis: a threat to global control of tuberculosis
- (2010) Neel R Gandhi et al. LANCET
- Mycobacterial Esx-3 is required for mycobactin-mediated iron acquisition
- (2009) M. S. Siegrist et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Synthesis of heterocycles from arylation products of unsaturated compounds: XVIII. 5-Arylfuran-2-carboxylic acids and their application in the synthesis of 1,2,4-thiadiazole, 1,3,4-oxadiazole, and [1,2,4]triazolo[3,4-b][1,3,4]thiadiazole derivatives
- (2009) Yu. I. Gorak et al. RUSSIAN JOURNAL OF ORGANIC CHEMISTRY
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreBecome a Peeref-certified reviewer
The Peeref Institute provides free reviewer training that teaches the core competencies of the academic peer review process.
Get Started