Novel 1,3,4-oxadiazoles as antitubercular agents with limited activity against drug-resistant tuberculosis

Identification and development of benzoxazole derivatives as novel bacterial glutamate racemase inhibitors

(2018) Prasanthi Malapati et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

A Facile Synthesis and Antituberculosis Properties of Almazole D and Its Enantiomer

(2017) Dhanaji M. Lade et al.   ChemistrySelect

SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules

(2017) Antoine Daina et al.   Scientific Reports

Synthesis, biological evaluation and molecular docking study of some novel indole and pyridine based 1,3,4-oxadiazole derivatives as potential antitubercular agents

(2016) N.C. Desai et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A study on pre-XDR & XDR tuberculosis & their prevalent genotypes in clinical isolates of Mycobacterium tuberculosis in north India

(2016) Amita Jain et al.   INDIAN JOURNAL OF MEDICAL RESEARCH

Development of 3,5-Dinitrobenzylsulfanyl-1,3,4-oxadiazoles and Thiadiazoles as Selective Antitubercular Agents Active Against Replicating and Nonreplicating Mycobacterium tuberculosis

(2016) Galina Karabanovich et al.   JOURNAL OF MEDICINAL CHEMISTRY

Isoniazid metabolism and hepatotoxicity

(2016) Pengcheng Wang et al.   Acta Pharmaceutica Sinica B

Benzothiazinethione is a potent preclinical candidate for the treatment of drug-resistant tuberculosis

(2016) Chao Gao et al.   Scientific Reports

Bedaquiline in the treatment of multidrug- and extensively drug-resistant tuberculosis

(2015) Alexander S. Pym et al.   EUROPEAN RESPIRATORY JOURNAL

Lead Optimization of a Novel Series of Imidazo[1,2-a]pyridine Amides Leading to a Clinical Candidate (Q203) as a Multi- and Extensively-Drug-Resistant Anti-tuberculosis Agent

(2014) Sunhee Kang et al.   JOURNAL OF MEDICINAL CHEMISTRY

P450-Mediated O-Demethylated Metabolite Is Responsible for Rat Hepatobiliary Toxicity of Pyridyltriazine-Containing PI3K Inhibitors

(2014) Raju Subramanian et al.   TOXICOLOGICAL SCIENCES

Sensititre MYCOTB MIC Plate for Testing Mycobacterium tuberculosis Susceptibility to First- and Second-Line Drugs

(2013) Jongseok Lee et al.   ANTIMICROBIAL AGENTS AND CHEMOTHERAPY

Discovery of Q203, a potent clinical candidate for the treatment of tuberculosis

(2013) Kevin Pethe et al.   NATURE MEDICINE

Molecular properties prediction and synthesis of novel 1,3,4-oxadiazole analogues as potent antimicrobial and antitubercular agents

(2011) Mohamed Jawed Ahsan et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Benzothiazinones Kill Mycobacterium tuberculosis by Blocking Arabinan Synthesis

(2009) V. Makarov et al.   SCIENCE