Enantioselective Copper(II)-Catalyzed Conjugate Addition of Indoles to β-Substituted Unsaturated Acyl Phosphonates

Enantioselective Construction of Cyclic Indolyl α-Amino Estersviaa Friedel-Crafts Alkylation Reaction

(2015) Liang Wu et al.   ADVANCED SYNTHESIS & CATALYSIS

Transition Metal-Catalyzed CH Activation of Indoles

(2015) Alexander H. Sandtorv   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Bis(oxazoline) Ligands Possessing C-5 gem-Disubstitution and Their Application in Asymmetric Friedel–Crafts Alkylations

(2015) Steven O’Reilly et al.   JOURNAL OF ORGANIC CHEMISTRY

Heteroarylidene-tethered bis(oxazoline) copper complexes catalyzed cascade reaction involving asymmetric Friedel–Crafts alkylation/N-hemiacetalization of indoles with β,γ-unsaturated α-ketoester

(2015) Hong-Li Ma et al.   TETRAHEDRON

Enantioselective Friedel–Crafts reaction of 4,7-dihydroindoles with β-CF3-β-disubstituted nitroalkenes

(2015) Hao Wu et al.   Organic Chemistry Frontiers

Chemistry of α-Oxoesters: A Powerful Tool for the Synthesis of Heterocycles

(2014) Bagher Eftekhari-Sis et al.   CHEMICAL REVIEWS

Asymmetric Friedel–Crafts Alkylation of α-Substituted β-Nitroacrylates: Access to β2,2-Amino Acids Bearing Indolic All-Carbon Quaternary Stereocenters

(2014) Jian-Quan Weng et al.   ORGANIC LETTERS

Direct Catalytic Asymmetric Synthesis of N-Heterocycles from Commodity Acid Chlorides by Employing α,β-Unsaturated Acylammonium Salts

(2013) Sreekumar Vellalath et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Synthesis of Pyrroloindolones by N-Heterocyclic Carbene Catalyzed [2+3] Annulation of α-Chloroaldehydes with Nitrovinylindoles

(2013) Qijian Ni et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Friedel-Crafts Alkylation/N-Hemiacetalization Cascade Reaction with Indoles

(2013) Hong-Gang Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Friedel–Crafts alkylation for synthesis of 2-substituted indole derivatives

(2013) Yulong Zhang et al.   CHEMICAL COMMUNICATIONS

Asymmetric synthesis of 3,4-annulated indoles through an organocatalytic cascade approach

(2013) Lorenzo Caruana et al.   CHEMICAL COMMUNICATIONS

Cu(OTf)2-Catalyzed Asymmetric Friedel–Crafts Alkylation Reaction of Indoles with Arylidene Malonates Using Bis(sulfonamide)-Diamine Ligands

(2013) Jing Wu et al.   JOURNAL OF ORGANIC CHEMISTRY

Highly Enantioselective Construction of Trifluoromethylated All-Carbon Quaternary Stereocenters via Nickel-Catalyzed Friedel–Crafts Alkylation Reaction

(2013) Jian-Rong Gao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

One-Pot Asymmetric Synthesis of Seven-Membered Carbocycles Cyclohepta[b]indoles via a Sequential Organocatalytic Michael/Double Friedel–Crafts Alkylation Reaction

(2013) Nitin S. Dange et al.   ORGANIC LETTERS

Highly enantioselective Friedel–Crafts alkylation of indoles and pyrrole with β,γ-unsaturated α-ketoesters catalyzed by heteroarylidene-tethered bis(oxazoline) copper complexes

(2012) Lei Liu et al.   CHEMICAL COMMUNICATIONS

Indoles in Multicomponent Processes (MCPs)

(2012) Morteza Shiri   CHEMICAL REVIEWS

Exploiting the Electrophilic Properties of Indole Intermediates: New Options in Designing Asymmetric Reactions

(2011) Charles C. J. Loh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enhanced Efficiency of Thiourea Catalysts by External Brønsted Acids in the Friedel-Crafts Alkylation of Indoles

(2011) Eugenia Marqués-López et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Highly enantioselective Friedel–Crafts reaction of indoles with N-sulfonyl aldimines catalyzed by heteroarylidene malonate-type bis(oxazoline) copper(II) complexes

(2011) Lei Liu et al.   TETRAHEDRON-ASYMMETRY

Development of Diphenylamine-Linked Bis(imidazoline) Ligands and Their Application in Asymmetric Friedel-Crafts Alkylation of Indole Derivatives with Nitroalkenes

(2010) Han Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Friedel–Crafts alkylation reaction of indoles with α,β-unsaturated acyl phosphonates catalyzed by chiral phosphoric acid

(2010) Prabhakar Bachu et al.   CHEMICAL COMMUNICATIONS

Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

(2010) Anna J. Kochanowska-Karamyan et al.   CHEMICAL REVIEWS

Monodentate N-Ligand-Directed Bifunctional Transition-Metal Catalysis: Highly Enantioselective Friedel-Crafts Alkylation of Indoles with Nitroalkenes

(2010) Fengfeng Guo et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalyzed Asymmetric Friedel-Crafts Reactions

(2010) Vincent Terrasson et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Acyl Phosphonates: Good Hydrogen Bond Acceptors and Ester/Amide Equivalents in Asymmetric Organocatalysis

(2010) Hao Jiang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Simple indole alkaloids and those with a nonrearranged monoterpenoid unit

(2010) Minoru Ishikura et al.   NATURAL PRODUCT REPORTS

Enantioselective Friedel–Crafts alkylation of indole derivatives catalyzed by new Yb(OTf)3-pyridylalkylamine complexes as chiral Lewis acids

(2010) Guillaume Grach et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Asymmetric Binary-Acid Catalysis with Chiral Phosphoric Acid and MgF2: Catalytic Enantioselective Friedel−Crafts Reactions of β,γ-Unsaturated α-Ketoesters

(2010) Jian Lv et al.   ORGANIC LETTERS

Highly Enantioselective Friedel–Crafts Reaction of Indole with Alkylidenemalonates Catalyzed by Heteroarylidene Malonate-Derived Bis(oxazoline) Copper(II) Complexes

(2009) Yan-Jin Sun et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Friedel–Crafts reaction of N-heterocycles and nitroalkenes catalyzed by imidazoline–aminophenol–Cu complex

(2009) Naota Yokoyama et al.   CHEMICAL COMMUNICATIONS

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Enantioselective Friedel-Crafts Alkylation of Indoles with Alkylidene Malonates Catalyzed byN,N′-Dioxide-Scandium(III) Complexes: Asymmetric Synthesis ofβ-Carbolines

(2009) Yanling Liu et al.   CHEMISTRY-A EUROPEAN JOURNAL

From Nature to Drug Discovery: The Indole Scaffold as a ‘Privileged Structure’

(2009) Fernando de Sa Alves et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

AgAsF6/Sm(OTf)3Promoted Reversal of Enantioselectivity for the Asymmetric Friedel−Crafts Alkylations of Indoles with β,γ-Unsaturated α-Ketoesters

(2009) Yanling Liu et al.   ORGANIC LETTERS

N,N′-Dioxide–scandium(III) complex catalyzed highly enantioselective Friedel–Crafts alkylation of indole to alkylidene malonates

(2009) Yanling Liu et al.   TETRAHEDRON

Chiral Phosphoric Acid Catalyzed Enantioselective Friedel–Crafts Alkylation of Indoles with Nitroalkenes: Cooperative Effect of 3 Å Molecular Sieves

(2008) Junji Itoh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Asymmetric Friedel–Crafts Alkylation of Indoles with Methyl (E)-2-Oxo-4-aryl-3-butenoates Catalyzed by Sc(OTf)3/pybox

(2008) Giovanni Desimoni et al.   CHEMISTRY-A EUROPEAN JOURNAL

Asymmetric Friedel–Crafts Alkylation of Electron‐Rich N‐Heterocycles with Nitroalkenes Catalyzed by Diphenylamine‐Tethered Bis(oxazoline) and Bis(thiazoline) ZnIIComplexes

(2008) Han Liu et al.   Chemistry-An Asian Journal

Catalytic Enantioselective Additions of Indoles to Nitroalkenes

(2008) Madhu Ganesh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

BINAM and H8-BINAM-based chiral imines and Zn(OTf)2-catalyzed enantioselective Friedel–Crafts alkylation of indoles with nitroalkenes

(2008) Zhi-Liang Yuan et al.   TETRAHEDRON-ASYMMETRY

Asymmetric Brønsted Acid Catalysis: Enantioselective Nucleophilic Substitutions and 1,4-Additions

(2007) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Enantiopure (S)-Indolylglycine by Organocatalyzed Friedel–Crafts Alkylation of Indole

(2007) Martin J. Wanner et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY