Metal-free, high yielding synthesis of unsymmetrical biaryl, bi(heteroaryl), aryl vinyl, aryl alkyl sulfones via coupling of aryne with sulfinic acid salts

Discovery of Vinyl Sulfones as a Novel Class of Neuroprotective Agents toward Parkinson’s Disease Therapy

(2014) Seo Yeon Woo et al.   JOURNAL OF MEDICINAL CHEMISTRY

Sulfonylation of Five-Membered Heterocycles via an SNAr Reaction

(2013) Shuai Liang et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine-Catalyzed Regioselective 2-Sulfonylation of Indoles with Sodium Sulfinates

(2013) Fuhong Xiao et al.   ORGANIC LETTERS

Recent advances in transition-metal-free carbon–carbon and carbon–heteroatom bond-forming reactions using arynes

(2012) Anup Bhunia et al.   CHEMICAL SOCIETY REVIEWS

A one-pot regioselective synthetic route to vinyl sulfones from terminal epoxides in aqueous media

(2012) Ruchi Chawla et al.   GREEN CHEMISTRY

1,2-Dibromotetrachloroethane: An Ozone-Friendly Reagent for the in Situ Ramberg–Bäcklund Rearrangement and Its Use in the Formal Synthesis of E-Resveratrol

(2012) Stefan C. Söderman et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Synthesis of Diaryl Sulfones from Arylsulfinic Acid Salts and Diaryliodonium Salts

(2012) Natalie Umierski et al.   ORGANIC LETTERS

Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: New Cyclic Substituents at Indole-2-carboxamide

(2011) Giuseppe La Regina et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6Receptor (5-HT6R) Antagonists

(2011) Alexandre V. Ivachtchenko et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Graphical Journey of Innovative Organic Architectures That Have Improved Our Lives

(2010) Nicholas A. McGrath et al.   JOURNAL OF CHEMICAL EDUCATION

5-Piperazinyl-3-sulfonylindazoles as Potent and Selective 5-Hydroxytryptamine-6 Antagonists

(2010) Kevin G. Liu et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Practical, One-Pot Synthesis of Sulfonylated Pyridines

(2010) Kevin M. Maloney et al.   ORGANIC LETTERS

Herbicidal 4-hydroxyphenylpyruvate dioxygenase inhibitors—A review of the triketone chemistry story from a Syngenta perspective

(2009) Renaud Beaudegnies et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Palladium-catalyzed coupling of vinyl tosylates with arylsulfinate salts

(2009) Diana C. Reeves et al.   TETRAHEDRON LETTERS