Analogues of the HIV-Tat peptide containing Nη-modified arginines as potent inhibitors of protein arginine N-methyltransferases

Kinetic Mechanism of Protein Arginine Methyltransferase 6 (PRMT6)

(2012) Obiamaka Obianyo et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Epigenetic protein families: a new frontier for drug discovery

(2012) Cheryl H. Arrowsmith et al.   NATURE REVIEWS DRUG DISCOVERY

Structural basis for CARM1 inhibition by indole and pyrazole inhibitors

(2011) John S. Sack et al.   BIOCHEMICAL JOURNAL

A Protein ArginineN-Methyltransferase 1 (PRMT1) and 2 Heteromeric Interaction Increases PRMT1 Enzymatic Activity

(2011) Magnolia L. Pak et al.   BIOCHEMISTRY

A Transient Kinetic Analysis of PRMT1 Catalysis

(2011) You Feng et al.   BIOCHEMISTRY

Peptidic Partial Bisubstrates as Inhibitors of the Protein Arginine N-Methyltransferases

(2011) Peter 't Hart et al.   CHEMBIOCHEM

Structural insights into protein arginine symmetric dimethylation by PRMT5

(2011) L. Sun et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Translocation of HIV TAT peptide and analogues induced by multiplexed membrane and cytoskeletal interactions

(2011) A. Mishra et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Nη-Substituted Arginyl Peptide Inhibitors of Protein ArginineN-Methyltransferases

(2010) Ted M. Lakowski et al.   ACS Chemical Biology

Dysregulation of PRMT1 and PRMT6, Type I arginine methyltransferases, is involved in various types of human cancers

(2010) Masanori Yoshimatsu et al.   INTERNATIONAL JOURNAL OF CANCER

Protein arginine methyltransferase 6 regulates multiple aspects of gene expression

(2010) Matthew J. Harrison et al.   NUCLEIC ACIDS RESEARCH

Förster resonance energy transfer measurements of cofactor-dependent effects on protein arginineN-methyltransferase homodimerization

(2010) Dylan Thomas et al.   PROTEIN SCIENCE

Kinetic analysis of human protein arginine N-methyltransferase 2: formation of monomethyl- and asymmetric dimethyl-arginine residues on histone H4

(2009) Ted M. Lakowski et al.   BIOCHEMICAL JOURNAL

para-Nitrophenyl Sulfate Activation of Human Sulfotransferase 1A1 Is Consistent with Intercepting theE·PAP Complex and Reformation ofE·PAPS

(2009) Eduard Tyapochkin et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Type I Arginine Methyltransferases PRMT1 and PRMT-3 Act Distributively

(2009) Knut Kölbel et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Protein Arginine Methylation in Mammals: Who, What, and Why

(2009) Mark T. Bedford et al.   MOLECULAR CELL

Protein methyltransferases as a target class for drug discovery

(2009) Robert A. Copeland et al.   NATURE REVIEWS DRUG DISCOVERY

Kinetic Mechanism of Protein Arginine Methyltransferase 1†

(2008) Obiamaka Obianyo et al.   BIOCHEMISTRY

Chemical mechanisms of histone lysine and arginine modifications

(2008) Brian C. Smith et al.   Biochimica et Biophysica Acta-Gene Regulatory Mechanisms

A Kinetic Study of Human Protein ArginineN-Methyltransferase 6 Reveals a Distributive Mechanism

(2008) Ted M. Lakowski et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Preparation ofNG-Substitutedl-Arginine Analogues Suitable for Solid Phase Peptide Synthesis

(2008) Nathaniel I. Martin et al.   JOURNAL OF ORGANIC CHEMISTRY